| GENE_SYMBOL |
DRUG_NAME |
Ki (nM) |
IC50 (nM) |
Kd (nM) |
EC50 (nM) |
Potency (nM) |
AC50 (nM) |
Datasource |
| PIK3CG |
N-[5-[3-[(4-hydroxyphenyl)sulfamoyl]-4-methoxyphenyl]-4-methyl-1,3-thiazol-2-yl]-2-(oxan-4-yl)acetamide |
NA |
200000 |
NA |
NA |
NA |
NA |
BindingDB |
| PIK3CG |
N-[5-[3-[(4-fluorophenyl)sulfamoyl]-4-methoxyphenyl]-4-methyl-1,3-thiazol-2-yl]-2-(oxan-4-yl)acetamide |
NA |
200000 |
NA |
NA |
NA |
NA |
BindingDB |
| PIK3CG |
N-[5-[3-[(4-hydroxy-2-methylphenyl)sulfamoyl]-4-methoxyphenyl]-4-methyl-1,3-thiazol-2-yl]-2-(oxan-4-yl)acetamide |
NA |
200000 |
NA |
NA |
NA |
NA |
BindingDB |
| PIK3CG |
5-[2-(tert-butylamino)-4-methyl-1,3-thiazol-5-yl]-N-(4-hydroxycyclohexyl)-2-methoxybenzenesulfonamide |
NA |
200000 |
NA |
NA |
NA |
NA |
BindingDB |
| PIK3CG |
5-[2-[[(1R)-1-cyclohexylethyl]amino]-4-methyl-1,3-thiazol-5-yl]-2-methoxy-N-piperidin-4-ylbenzenesulfonamide |
NA |
200000 |
NA |
NA |
NA |
NA |
BindingDB |
| PIK3CG |
5-[2-(cyclohexylamino)-4-methyl-1,3-thiazol-5-yl]-N-cyclopentyl-2-methoxybenzenesulfonamide |
NA |
200000 |
NA |
NA |
NA |
NA |
BindingDB |
| PIK3CG |
N-(cyclohexylmethyl)-5-[2-(cyclohexylmethylamino)-4-methyl-1,3-thiazol-5-yl]-2-methoxybenzenesulfonamide |
NA |
200000 |
NA |
NA |
NA |
NA |
BindingDB |
| PIK3CG |
N-(4-hydroxycyclohexyl)-2-methoxy-5-[4-methyl-2-(propan-2-ylamino)-1,3-thiazol-5-yl]benzenesulfonamide |
NA |
200000 |
NA |
NA |
NA |
NA |
BindingDB |
| PIK3CG |
N-[5-[3-[(3-hydroxy-5-methylphenyl)sulfamoyl]-4-methoxyphenyl]-4-methyl-1,3-thiazol-2-yl]-2-(oxan-4-yl)acetamide |
NA |
200000 |
NA |
NA |
NA |
NA |
BindingDB |
| PIK3CG |
3-cyclopentyl-N-[5-[4-methoxy-3-(piperidin-4-ylsulfamoyl)phenyl]-4-methyl-1,3-thiazol-2-yl]propanamide |
NA |
200000 |
NA |
NA |
NA |
NA |
BindingDB |
| PIK3CG |
5-[2-(2-cyclohexylethylamino)-4-methyl-1,3-thiazol-5-yl]-N-(3-hydroxycyclopentyl)-2-methoxybenzenesulfonamide |
NA |
200000 |
NA |
NA |
NA |
NA |
BindingDB |
| PIK3CG |
N-[5-[5-[(2,4-difluorophenyl)sulfamoyl]-6-methoxypyridin-3-yl]-4-methyl-1,3-thiazol-2-yl]-2-(oxan-4-yl)acetamide |
NA |
200000 |
NA |
NA |
NA |
NA |
BindingDB |
| PIK3CG |
5-[2-[[(1R)-1-cyclohexylethyl]amino]-4-methyl-1,3-thiazol-5-yl]-2-methoxy-N-piperidin-3-ylbenzenesulfonamide |
NA |
200000 |
NA |
NA |
NA |
NA |
BindingDB |
| PIK3CG |
3-[[2-Methoxy-5-[4-methyl-2-[[2-(oxan-4-yl)acetyl]amino]-1,3-thiazol-5-yl]pyridin-3-yl]sulfonylamino]benzoic acid |
NA |
200000 |
NA |
NA |
NA |
NA |
BindingDB |
| PIK3CG |
5-[2-(cyclohexylmethylamino)-4-methyl-1,3-thiazol-5-yl]-N-cyclopropyl-2-methoxybenzenesulfonamide |
NA |
200000 |
NA |
NA |
NA |
NA |
BindingDB |
| PIK3CG |
8-Ethyl-11-(4-methoxyphenyl)-13-morpholin-4-yl-6,8,10,12-tetrazatricyclo[7.4.0.02,6]trideca-1(13),9,11-triene-7-thione |
NA |
125800 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| PIK3CG |
11-(3-Methoxyphenyl)-13-morpholin-4-yl-8-phenyl-6,8,10,12-tetrazatricyclo[7.4.0.02,6]trideca-1(13),9,11-triene-7-thione |
NA |
465500 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| PIK3CG |
11-(4-Methoxyphenyl)-13-morpholin-4-yl-8-phenyl-6,8,10,12-tetrazatricyclo[7.4.0.02,6]trideca-1(13),9,11-triene-7-thione |
NA |
345900 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| PIK3CG |
13-Morpholin-4-yl-11-(morpholin-4-ylmethyl)-8-phenyl-6,8,10,12-tetrazatricyclo[7.4.0.02,6]trideca-1(13),9,11-triene-7-thione |
NA |
781500 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| PIK3CG |
13-Morpholin-4-yl-11-(1-morpholin-4-ylethyl)-8-phenyl-6,8,10,12-tetrazatricyclo[7.4.0.02,6]trideca-1(13),9,11-triene-7-thione |
NA |
967700 |
NA |
NA |
NA |
NA |
BindingDB|TTD |