| GENE_SYMBOL |
DRUG_NAME |
Ki (nM) |
IC50 (nM) |
Kd (nM) |
EC50 (nM) |
Potency (nM) |
AC50 (nM) |
Datasource |
| PIK3CG |
1-(cyclopropylmethyl)-4-[2-[[(1S)-1-(oxan-4-yl)ethyl]amino]-1,3-benzothiazol-6-yl]pyridin-2-one |
NA |
199526.23 |
NA |
NA |
NA |
NA |
TTD |
| PIK3CG |
2,4-Diamino-6-[[1-(5,8-dichloro-3-cyclobutyl-4-oxoquinazolin-2-yl)cyclopropyl]amino]pyrimidine-5-carbonitrile |
NA |
229000|524000 |
NA |
NA |
NA |
NA |
BindingDB |
| PIK3CG |
6-(1H-indol-4-yl)-1H-indazole |
NA |
158489.32 |
NA |
NA |
NA |
NA |
TTD |
| PIK3CG |
2-Methylpyrazolo[1,5-a]pyrimidine-3-carbonitrile |
NA |
773000 |
NA |
NA |
NA |
NA |
BindingDB|ChEMBL|TTD |
| PIK3CG |
1-[2-[4-(4,6-dimorpholin-4-yl-1,3,5-triazin-2-yl)anilino]-3H-benzimidazole-5-carbonyl]piperidine-4-carboxamide |
NA |
849000 |
NA |
NA |
NA |
NA |
BindingDB |
| PIK3CG |
PI3K/mTOR Inhibitor-6 |
NA |
444000 |
NA |
NA |
NA |
NA |
BindingDB |
| PIK3CG |
N-[(2S)-1-amino-1-oxopropan-2-yl]-2-[4-(4,6-dimorpholin-4-yl-1,3,5-triazin-2-yl)anilino]-3H-benzimidazole-5-carboxamide |
NA |
645000 |
NA |
NA |
NA |
NA |
BindingDB |
| PIK3CG |
5-(Benzylamino)pyrimido[4,5-c]quinoline-8-carboxylic acid |
NA |
5300000 |
NA |
NA |
NA |
NA |
BindingDB |
| PIK3CG |
6-Hydroxy-5-((2-methyl-4-((2-methylphenyl)diazenyl)phenyl)diazenyl)-2-naphthalenesulfonic acid |
NA |
2415000 |
NA |
NA |
NA |
NA |
TTD |
| PIK3CG |
4-[(2S,3aS,7aS)-2-(5-fluoro-4-oxo-3-pyridin-3-ylquinazolin-2-yl)-2,3,3a,4,5,6,7,7a-octahydroindol-1-yl]-2,6-diaminopyrimidine-5-carbonitrile |
NA |
364000 |
NA |
NA |
NA |
NA |
BindingDB |
| PIK3CG |
4-[(2S,3aS,7aS)-2-(5-chloro-3-morpholin-4-yl-4-oxoquinazolin-2-yl)-2,3,3a,4,5,6,7,7a-octahydroindol-1-yl]-2,6-diaminopyrimidine-5-carbonitrile |
NA |
312000 |
NA |
NA |
NA |
NA |
BindingDB |
| PIK3CG |
4-[(2S,3aS,7aS)-2-[5-chloro-3-(3-fluorophenyl)-4-oxoquinazolin-2-yl]-2,3,3a,4,5,6,7,7a-octahydroindol-1-yl]-2,6-diaminopyrimidine-5-carbonitrile |
NA |
280000 |
NA |
NA |
NA |
NA |
BindingDB |
| PIK3CG |
Theophylline |
NA |
2904000|800000 |
NA |
NA |
NA |
NA |
BindingDB|PubChem|TTD |
| PIK3CG |
2-(7-Oxobenzo[a]phenalen-3-yl)sulfinylacetic acid |
NA |
1570000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| PIK3CG |
7-(4-Ethoxyphenylamino)-4-hydroxynaphthalene-2-sulfonic acid |
NA |
992000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| PIK3CG |
3-(4-Butoxy-3-methoxyphenyl)pentanedioic acid |
NA |
134000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| PIK3CG |
6-(6-Methoxynaphthalen-2-yl)-2-methyl-6-oxohexanoic acid |
NA |
5184000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| PIK3CG |
Caffeine |
NA |
3630000|1000000 |
NA |
NA |
NA |
NA |
BindingDB|PubChem|TTD |
| PIK3CG |
3-(4-Morpholino-1-methyl-1H-pyrazolo[3,4-d]pyrimidine-6-yl)phenol |
NA |
717300 |
NA |
NA |
NA |
NA |
BindingDB |
| PIK3CG |
2,2'-((3-Chlorophenyl)methylene)bis(sulfanediyl)dibenzoic acid |
NA |
187000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |