| GENE_SYMBOL |
DRUG_NAME |
Ki (nM) |
IC50 (nM) |
Kd (nM) |
EC50 (nM) |
Potency (nM) |
AC50 (nM) |
Datasource |
| PIK3CG |
6-(Benzyloxy)-5-methoxy-1H-indole-2-carboxylic acid |
NA |
105000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| PIK3CG |
n,o-Bis[(benzyloxy)carbonyl]tyrosine |
NA |
324000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| PIK3CG |
5,7-Dimethyl-(1,2,4)triazolo(1,5-a)pyrimidin-2-amine |
NA |
1600000 |
NA |
NA |
NA |
NA |
TTD |
| PIK3CG |
3-(3,4-Dimethoxy-phenyl)-3-(3,4,5-trimethoxy-phenyl)-propionic acid |
NA |
6074000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| PIK3CG |
4-(5-oxo-3-pentadecyl-4-phenyldiazenyl-4H-pyrazol-1-yl)benzenesulfonic acid |
NA |
241000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| PIK3CG |
4-[(4-Carboxy-2,5-dimethyl-phenyl)disulfanyl]-2,5-dimethyl-benzoic acid |
NA |
1460000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| PIK3CG |
5,7-Dimethylpyrazolo[1,5-a]pyrimidin-2-amine |
NA |
915000 |
NA |
NA |
NA |
NA |
BindingDB|ChEMBL|TTD |
| PIK3CG |
4-(1,3-Benzodioxol-5-yl)-2-(3,4-dimethoxyphenyl)-4-oxobutanoic acid |
NA |
234000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| PIK3CG |
5-Chloro-2-[2-[3-[(3-fluorosulfonylphenyl)carbamoylamino]anilino]-2-oxoethoxy]benzoic acid |
NA |
9157000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| PIK3CG |
3-[4-(Benzyloxy)-3-methoxyphenyl]pentanedioic acid |
NA |
5876000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| PIK3CG |
Benzoxazole, 2-amino-6-chloro- |
NA |
380000 |
NA |
NA |
NA |
NA |
BindingDB|ChEMBL|TTD |
| PIK3CG |
6-Hydroxy-5-[[2-methoxy-4-[(4-sulfophenyl)diazenyl]phenyl]diazenyl]naphthalene-2-sulfonic acid |
NA |
2437000 |
NA |
NA |
NA |
NA |
TTD |
| PIK3CG |
3-(2,3,10,11-Tetramethoxyisoquinolino[2,1-b]isoquinolin-7-ium-8-yl)propanoic acid |
NA |
7333000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| PIK3CG |
6-Bromoimidazo[1,2-a]pyridin-2-amine |
NA |
156000 |
NA |
NA |
NA |
NA |
BindingDB|ChEMBL|TTD |
| PIK3CG |
(5-Hydroxyindolo(1,2-a)quinazolin-7-yl)acetic acid |
NA |
200000 |
NA |
NA |
NA |
NA |
TTD |
| PIK3CG |
7-Chloro-5-methyl-[1,2,4]triazolo[1,5-a]pyrimidine |
NA |
1670000 |
NA |
NA |
NA |
NA |
TTD |
| PIK3CG |
N-[(3,4-Dimethoxyphenyl)methyl]-2-[5-(quinolin-6-YL)-1,3,4-oxadiazol-2-YL]acetamide |
NA |
152200 |
NA |
NA |
NA |
NA |
BindingDB |
| PIK3CG |
|
NA |
2437000 |
NA |
NA |
NA |
NA |
BindingDB |
| PIK3CG |
|
NA |
2415000 |
NA |
NA |
NA |
NA |
BindingDB |
| PIK3CG |
2-Propan-2-ylpyrazolo[1,5-a]pyrimidine-3-carbonitrile |
NA |
395000 |
NA |
NA |
NA |
NA |
BindingDB|ChEMBL|TTD |