| GENE_SYMBOL |
DRUG_NAME |
Ki (nM) |
IC50 (nM) |
Kd (nM) |
EC50 (nM) |
Potency (nM) |
AC50 (nM) |
Datasource |
| PIK3CG |
|
NA |
1498000 |
NA |
NA |
NA |
NA |
BindingDB |
| PIK3CG |
{2-[(3-Ethyl-4-oxo-2-thioxo-1,3-thiazolidin-5-ylidene)methyl]-4-nitrophenoxy}acetic acid |
NA |
612000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| PIK3CG |
2-cyclopentyl-N-[5-[3-[(4-hydroxyphenyl)sulfamoyl]-4-methoxyphenyl]-4-methyl-1,3-thiazol-2-yl]acetamide |
NA |
200000 |
NA |
NA |
NA |
NA |
BindingDB |
| PIK3CG |
1-(4'-Chloro-phenylazo)-2-naphthol-6-sulfonic acid |
NA |
1498000 |
NA |
NA |
NA |
NA |
TTD |
| PIK3CG |
5-[2-(cycloheptylamino)-4-methyl-1,3-thiazol-5-yl]-N-(2,6-dimethylphenyl)-2-methoxybenzenesulfonamide |
NA |
200000 |
NA |
NA |
NA |
NA |
BindingDB |
| PIK3CG |
2-cyclopentyl-N-[5-[4-methoxy-3-[(6-methylpyridin-3-yl)sulfamoyl]phenyl]-4-methyl-1,3-thiazol-2-yl]acetamide |
NA |
200000 |
NA |
NA |
NA |
NA |
BindingDB |
| PIK3CG |
(2S)-4-(1,3-benzodioxol-5-yl)-4-oxo-2-[(3,4,5-trimethoxyphenyl)methyl]butanoic acid |
NA |
575000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| PIK3CG |
3-butyl-2-(7H-purin-6-ylsulfanylmethyl)quinazolin-4-one |
NA |
217800 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| PIK3R1 |
5-(4,6-Dimorpholin-4-yl-1,3,5-triazin-2-yl)-3-(trifluoromethyl)pyridin-2-amine |
4300000 |
NA |
NA |
NA |
NA |
NA |
BindingDB |
| PIK3R1 |
Wortmannin |
NA |
147000000 |
NA |
NA |
NA |
NA |
BindingDB |
| PIK3R2 |
(S)-1-(3-(2-(1-((6-amino-5-cyanopyrimidin-4-yl)amino)ethyl)-4-oxoquinazolin-3(4H)-yl)phenyl)-3-ethylurea |
NA |
340000 |
NA |
NA |
NA |
NA |
BindingDB |
| PIK3R2 |
(S)-1-(3-(2-(1-((6-amino-5-cyanopyrimidin-4-yl)amino)ethyl)-7-fluoro-4-oxoquinazolin-3(4H)-yl)phenyl)-3-ethylurea |
NA |
2600000 |
NA |
NA |
NA |
NA |
BindingDB |
| PIK3R2 |
(S)-1-(3-(2-(1-((6-amino-5-cyanopyrimidin-4-yl)amino)ethyl)-5-chloro-4-oxoquinazolin-3(4H)-yl)phenyl)-3-(2,2,2-trifluoroethyl)urea |
NA |
420000 |
NA |
NA |
NA |
NA |
BindingDB |
| PIK3R2 |
(S)-1-(3-(2-(1-((6-amino-5-cyanopyrimidin-4-yl)amino)ethyl)-5-chloro-4-oxoquinazolin-3(4H)-yl)phenyl)-3-(2-cyanophenyl)urea |
NA |
4800000 |
NA |
NA |
NA |
NA |
BindingDB |
| PIK3R2 |
(S)-1-(3-(2-(1-((6-amino-5-cyanopyrimidin-4-yl)amino)ethyl)-5-methoxy-4-oxoquinazolin-3(4H)-yl)phenyl)-3-ethylurea |
NA |
6600000 |
NA |
NA |
NA |
NA |
BindingDB |
| PIK3R2 |
(S)-1-(3-(2-(1-((4-amino-6-methyl-1,3,5-triazin-2-yl)amino)ethyl)-5-chloro-4-oxoquinazolin-3(4H)-yl)phenyl)-3-ethylurea |
NA |
5500000 |
NA |
NA |
NA |
NA |
BindingDB |
| PIK3R2 |
3-[5-chloro-2-[(1S)-1-[(2,6-diamino-5-cyanopyrimidin-4-yl)amino]ethyl]-4-oxoquinazolin-3-yl]-2-methylbenzamide |
NA |
526000 |
NA |
NA |
NA |
NA |
BindingDB |
| PIK3R2 |
1-[3-[2-[(2S)-1-(6-amino-5-cyanopyrimidin-4-yl)pyrrolidin-2-yl]-5-chloro-4-oxoquinazolin-3-yl]phenyl]-3-pyridin-2-ylurea |
NA |
420000 |
NA |
NA |
NA |
NA |
BindingDB |
| PIK3R2 |
(S)-1-(3-(2-(1-((6-amino-5-cyanopyrimidin-4-yl)amino)ethyl)-5-chloro-4-oxoquinazolin-3(4H)-yl)-4-chlorophenyl)-3-ethylurea |
NA |
210000|610000 |
NA |
NA |
NA |
NA |
BindingDB |
| PIK3R2 |
(S)-1-(3-(2-(1-((6-amino-5-cyanopyrimidin-4-yl)amino)ethyl)-8-chloro-4-oxoquinazolin-3(4H)-yl)phenyl)-3-(3-hydroxypropyl)urea |
NA |
220000 |
NA |
NA |
NA |
NA |
BindingDB |