| GENE_SYMBOL |
DRUG_NAME |
Ki (nM) |
IC50 (nM) |
Kd (nM) |
EC50 (nM) |
Potency (nM) |
AC50 (nM) |
Datasource |
| PRKCE |
2-(N-[2,6-dihydroxy-4-[4-[(4-hydroxybenzoyl)amino]pyrrolidin-3-yl]oxycarbonylbenzoyl]anilino)acetic acid |
NA |
150000 |
NA |
NA |
NA |
NA |
TTD |
| PRKCE |
[(4R)-3-[(4-hydroxybenzoyl)amino]azepan-4-yl] 3,5-dihydroxy-4-(1-hydroxynaphthalene-2-carbonyl)benzoate |
NA |
150000 |
NA |
NA |
NA |
NA |
TTD |
| PRKCE |
(1S,3aS,5aR,5bR,9S,11aR)-9-hydroxy-5a,5b,8,8,11a-pentamethyl-1-propan-2-yl-1,2,3,4,5,6,7,7a,9,10,11,11b,12,13,13a,13b-hexadecahydrocyclopenta[a]chrysene-3a-carboxylic acid |
NA |
150000 |
NA |
NA |
NA |
NA |
TTD |
| PRKCE |
betulinic acid 3-O-sulfonate potassium salt |
NA |
150000 |
NA |
NA |
NA |
NA |
TTD |
| PRKCE |
4-Phenyl-[1]benzofuro[2,3-b]pyridine-3,6-diol |
1000000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| PRKCE |
Harmine |
NA |
250000 |
NA |
NA |
NA |
NA |
PubChem |
| PRKCE |
Betulinic Acid |
NA |
150000 |
NA |
NA |
NA |
NA |
PubChem|TTD |
| PRKCE |
Platanic Acid |
NA |
150000 |
NA |
NA |
NA |
NA |
TTD |
| PRKCE |
Betulin |
NA |
150000 |
NA |
NA |
NA |
NA |
PubChem|TTD |
| PRKCE |
Edotecarin |
NA |
200000 |
NA |
NA |
NA |
NA |
PubChem |
| PRKCG |
N-(4-methoxybenzyl)benzofuro[2,3-b]pyridin-4-amine |
1000000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| PRKCG |
4-Phenyl-[1]benzofuro[2,3-b]pyridine-3,6-diol |
1000000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| PRKCG |
Harmine |
NA |
250000 |
NA |
NA |
NA |
NA |
PubChem |
| PRKCG |
Edotecarin |
NA |
200000 |
NA |
NA |
NA |
NA |
PubChem |
| PRKCH |
Harmine |
NA |
250000 |
NA |
NA |
NA |
NA |
PubChem |
| PRKCH |
Edotecarin |
NA |
200000 |
NA |
NA |
NA |
NA |
PubChem |
| PRKCI |
4-Chloro-1H-pyrrolo[2,3-b]pyridine |
NA |
1300000 |
NA |
NA |
NA |
NA |
ChEMBL|TTD |
| PRKCI |
5-Aminobenzimidazole |
NA |
728000 |
NA |
NA |
NA |
NA |
ChEMBL|TTD |
| PRKCI |
6-(1H-pyrrolo[2,3-b]pyridin-4-yl)-3,4-dihydro-2H-1,4-benzoxazine |
NA |
148000 |
NA |
NA |
NA |
NA |
ChEMBL|TTD |
| PRKCI |
4-(1H-indol-6-yl)-1H-pyrrolo[2,3-b]pyridine |
NA |
384000 |
NA |
NA |
NA |
NA |
TTD |