| GENE_SYMBOL |
DRUG_NAME |
Ki (nM) |
IC50 (nM) |
Kd (nM) |
EC50 (nM) |
Potency (nM) |
AC50 (nM) |
Datasource |
| PRKCI |
1-methyl-5-(1H-pyrrolo[2,3-b]pyridin-4-yl)benzimidazole |
NA |
384000 |
NA |
NA |
NA |
NA |
TTD |
| PRKCI |
5-(1H-pyrrolo[2,3-b]pyridin-4-yl)-2,3-dihydroisoindol-1-one |
NA |
105000 |
NA |
NA |
NA |
NA |
ChEMBL|TTD |
| PRKCI |
2-methyl-6-(1H-pyrrolo[2,3-b]pyridin-4-yl)-1H-benzimidazole |
NA |
215000 |
NA |
NA |
NA |
NA |
ChEMBL|TTD |
| PRKCI |
6-methoxy-2-[5-(1H-pyrrolo[2,3-b]pyridin-4-yl)pyrazolo[1,5-a]pyridin-3-yl]-3H-isoindol-1-one |
NA |
384000 |
NA |
NA |
NA |
NA |
TTD |
| PRKCI |
1-(azetidin-3-yl)-6-(1H-pyrrolo[2,3-b]pyridin-4-yl)benzimidazole |
NA |
188000 |
NA |
NA |
NA |
NA |
ChEMBL|TTD |
| PRKCI |
4-imidazo[1,5-a]pyridin-7-yl-1H-pyrrolo[2,3-b]pyridine |
NA |
221000 |
NA |
NA |
NA |
NA |
ChEMBL|TTD |
| PRKCI |
3-amino-N-(2,6-dimethylpyridin-4-yl)pyrazine-2-carboxamide |
NA |
263000 |
NA |
NA |
NA |
NA |
ChEMBL|TTD |
| PRKCI |
3-amino-N-(1H-pyrrolo[2,3-b]pyridin-4-yl)pyrazine-2-carboxamide |
NA |
384000 |
NA |
NA |
NA |
NA |
TTD |
| PRKCI |
3-amino-N-(2-bromopyridin-4-yl)pyrazine-2-carboxamide |
NA |
384000 |
NA |
NA |
NA |
NA |
TTD |
| PRKCI |
4-Bromo-1H-pyrrolo[2,3-b]pyridine |
NA |
615000 |
NA |
NA |
NA |
NA |
ChEMBL|TTD |
| PRKCI |
1H-Pyrrolo[2,3-b]pyridine-4-carboxamide |
NA |
384000 |
NA |
NA |
NA |
NA |
TTD |
| PRKCI |
4-pyridin-2-yl-1H-pyrrolo[2,3-b]pyridine |
NA |
374000 |
NA |
NA |
NA |
NA |
ChEMBL|TTD |
| PRKCI |
N-methyl-(5-pyrid-4-ylthien-2-yl)methylamine |
NA |
229000 |
NA |
NA |
NA |
NA |
ChEMBL|TTD |
| PRKCI |
4-Chloro-5-methyl-1H-pyrrolo[2,3-b]pyridine |
NA |
452000 |
NA |
NA |
NA |
NA |
ChEMBL|TTD |
| PRKCI |
2,3-Dihydro-1-benzofuran-5-carbothioamide |
NA |
927000 |
NA |
NA |
NA |
NA |
ChEMBL|TTD |
| PRKCI |
1-methyl-1H-indol-5-amine |
NA |
1312000 |
NA |
NA |
NA |
NA |
ChEMBL|TTD |
| PRKCI |
1-(3-Amino-4-(methylamino)phenyl)ethanone |
NA |
1423000 |
NA |
NA |
NA |
NA |
ChEMBL|TTD |
| PRKCI |
(3-(Pyridin-4-yl)phenyl)methanol |
NA |
2216000 |
NA |
NA |
NA |
NA |
ChEMBL|TTD |
| PRKCI |
3-amino-N-(pyridin-4-ylmethyl)pyrazine-2-carboxamide |
NA |
384000 |
NA |
NA |
NA |
NA |
TTD |
| PRKCI |
3-Pyridinecarboxamide, 2-amino-N-phenyl- |
NA |
424000 |
NA |
NA |
NA |
NA |
ChEMBL|TTD |