| GENE_SYMBOL |
DRUG_NAME |
Ki (nM) |
IC50 (nM) |
Kd (nM) |
EC50 (nM) |
Potency (nM) |
AC50 (nM) |
Datasource |
| PRKCI |
4-Amino-2-[(Diethylamino)Methyl]Phenol |
NA |
1570000 |
NA |
NA |
NA |
NA |
ChEMBL|TTD |
| PRKCI |
6-Hydroxy-3,4-dihydro-1(2H)-naphthalenone |
NA |
1677000 |
NA |
NA |
NA |
NA |
ChEMBL|TTD |
| PRKCI |
N-(4-methoxybenzyl)benzofuro[2,3-b]pyridin-4-amine |
1000000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| PRKCI |
4-Phenyl-[1]benzofuro[2,3-b]pyridine-3,6-diol |
1000000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| PRKCI |
3-amino-N-(3-bromopyridin-4-yl)pyrazine-2-carboxamide |
NA |
384000 |
NA |
NA |
NA |
NA |
TTD |
| PRKCI |
Harmine |
NA |
250000 |
NA |
NA |
NA |
NA |
PubChem |
| PRKCI |
4-(4-bromo-1H-pyrazol-1-yl)-1H-pyrrolo[2,3-b]pyridine |
NA |
201000 |
NA |
NA |
NA |
NA |
ChEMBL|TTD |
| PRKCI |
3-(1H-pyrrolo[2,3-b]pyridin-4-yl)benzamide |
NA |
371000 |
NA |
NA |
NA |
NA |
ChEMBL|TTD |
| PRKCI |
2-amino-5-bromo-N-(pyridin-4-yl)nicotinamide |
NA |
384000 |
NA |
NA |
NA |
NA |
TTD |
| PRKCI |
1-(2,6-Dihydroxy-3-propylphenyl)ethanone |
NA |
1556000 |
NA |
NA |
NA |
NA |
ChEMBL|TTD |
| PRKCI |
2-Amino-5-(3-carbamoyl-phenyl)-N-pyridin-4-yl-nicotinamide |
NA |
384000 |
NA |
NA |
NA |
NA |
TTD |
| PRKCI |
Phthalazinone |
NA |
589000 |
NA |
NA |
NA |
NA |
ChEMBL|TTD |
| PRKCI |
Edotecarin |
NA |
200000 |
NA |
NA |
NA |
NA |
PubChem |
| PRKCQ |
(1,2,4)Triazino(3,4-c)(1,4)benzoxazin-2(1H)-one, 3,5-dihydro- |
NA |
453000 |
NA |
NA |
NA |
NA |
BindingDB|ChEMBL|TTD |
| PRKCQ |
Harmine |
NA |
250000 |
NA |
NA |
NA |
NA |
PubChem |
| PRKCQ |
Edotecarin |
NA |
200000 |
NA |
NA |
NA |
NA |
PubChem |
| PRKCZ |
2-[2,6-dihydroxy-4-[(3R,4R)-3-[(4-hydroxybenzoyl)amino]oxepan-4-yl]oxycarbonylbenzoyl]-3-hydroxybenzoic acid |
NA |
150000 |
NA |
NA |
NA |
NA |
TTD |
| PRKCZ |
2-[2,6-dihydroxy-4-[(3S,4R)-3-[(4-hydroxybenzoyl)amino]thiepan-4-yl]oxycarbonylbenzoyl]-3-hydroxybenzoic acid |
NA |
121000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| PRKCZ |
4-(2-Carboxy-6-hydroxy-benzoyl)-3,5-dihydroxy-benzoic acid (3S,4S)-3-(4-hydroxy-benzoylamino)-azepan-4-yl ester |
NA |
150000 |
NA |
NA |
NA |
NA |
TTD |
| PRKCZ |
2-[2,6-dihydroxy-4-[(3S,4R)-3-[(4-hydroxybenzoyl)amino]-1,1-dioxothiepan-4-yl]oxycarbonylbenzoyl]-3-hydroxybenzoic acid |
NA |
150000 |
NA |
NA |
NA |
NA |
TTD |