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Drugs And Genes
Negative Drug Target Genes
GENE_SYMBOL DRUG_NAME Ki (nM) IC50 (nM) Kd (nM) EC50 (nM) Potency (nM) AC50 (nM) Datasource
PRSS1 Benzylamine 299916251.9|299916000 NA NA NA NA|NA NA|NA BindingDB|PubChem|TTD
PRSS1 4-Methoxybenzylamine 1000000000 NA NA NA NA|NA NA|NA BindingDB|TTD
PRSS1 [2-[(3,5-dimethyl-1-phenylpyrazol-4-yl)amino]-2-oxoethyl] 2-(1H-indol-3-yl)acetate NA 150000 NA NA NA NA BindingDB
PRSS1 Cyclohexanemethylamine NA NA 1148154 NA NA NA BindingDB
PRSS1 4-Phenylbutylamine NA NA 19952623 NA NA NA BindingDB
PRSS1 2-(6-cyano-3-(2,2-difluoro-2-(pyridin-2-yl)ethylamino)-2-oxopyrazin-1(2H)-yl)-N-((3-fluoropyridin-2-yl)methyl)acetamide 213000 NA NA NA NA NA BindingDB|TTD
PRSS1 tert-butyl (3S)-4-[[3-(1-aminoisoquinolin-6-yl)-1-oxo-1-piperidin-1-ylpropan-2-yl]amino]-3-[(4-methoxy-2,3,6-trimethylphenyl)sulfonylamino]-4-oxobutanoate NA 378000 NA NA NA NA BindingDB|TTD
PRSS1 2-(6-Methyl-2-oxo-3-phenethylamino-2H-pyrazin-1-yl)-N-pyridin-2-ylmethyl-acetamide 1000000 NA NA NA NA NA TTD
PRSS1 N-Imidazo[1,2-a]pyridin-7-ylmethyl-2-(6-methyl-2-oxo-3-phenethylamino-2H-pyrazin-1-yl)-acetamide 120000 NA NA NA NA NA BindingDB|TTD
PRSS1 (4-Benzyloxy-benzyl)-pyridin-4-yl-amine 233000 NA NA NA NA NA BindingDB|TTD
PRSS1 N-(1H-Indol-5-ylmethyl)-2-[6-methyl-2-oxo-3-(2-pyridin-2-yl-ethylamino)-2H-pyrazin-1-yl]-acetamide 290000 NA NA NA NA NA BindingDB|TTD
PRSS1 GW-813893 NA 158000 NA NA NA NA PubChem
PRSS1 2-[3-(2,2-Difluoro-2-pyridin-2-yl-ethylamino)-6-methyl-2-oxo-2H-pyrazin-1-yl]-N-(4-methyl-pyridin-2-ylmethyl)-acetamide 431000 NA NA NA NA NA BindingDB|TTD
PRSS1 Dpoc-4088 202000 NA NA NA NA NA BindingDB|PubChem|TTD
PRSS1 CGH-1484A free base 153000 NA NA NA NA NA BindingDB|TTD
PRSS2 Xeruborbactam NA 1000000 NA NA NA NA PubChem
PRSS2 Vaborbactam NA 1000000 NA NA NA NA PubChem
PRSS2 Baicalin NA 1000000 NA NA NA NA PubChem
PRSS2 GW-813893 NA 158000 NA NA NA NA PubChem
PRSS2 Dpoc-4088 202000 NA NA NA NA NA PubChem