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Drugs And Genes
Negative Drug Target Genes
GENE_SYMBOL DRUG_NAME Ki (nM) IC50 (nM) Kd (nM) EC50 (nM) Potency (nM) AC50 (nM) Datasource
PSENEN MG 132 NA 200000 NA NA NA NA BindingDB
PSENEN 9-octyl-2-(2H-tetrazol-5-ylmethoxy)carbazole NA 102000 NA NA NA NA TTD
PSENEN 2-(9-Octylcarbazol-2-yl)oxyacetamide NA 104000 NA NA NA NA TTD
PSENEN 2-(9-Octylcarbazol-2-yl)oxyacetonitrile NA 105000 NA NA NA NA TTD
PSENEN 4-[4-[(Z)-(5-chloro-2-oxo-1H-indol-3-ylidene)methyl]-2-methoxyphenoxy]butanenitrile NA 160000 NA NA NA NA TTD
PSENEN Tarenflurbil NA 307000 NA NA NA NA PubChem|TTD
PSENEN 2-Acetylamino-4-methyl-pentanoic acid [1-(1-formyl-butylcarbamoyl)-3-methyl-butyl]-amide NA 200000 NA NA NA NA BindingDB
PSMB1 4-[4-[3-(Cyclopropylmethyl)-4-oxophthalazin-1-yl]phenoxy]butyl-triphenylphosphanium NA 133100 NA NA NA NA BindingDB
PSMB1 4-[4-[3-(Cyclobutylmethyl)-4-oxophthalazin-1-yl]phenoxy]butyl-triphenylphosphanium NA 125200 NA NA NA NA BindingDB
PSMB1 4-[4-[3-[4-(Methylamino)phenyl]-4-oxophthalazin-1-yl]phenoxy]butyl-triphenylphosphanium NA 130900 NA NA NA NA BindingDB
PSMB1 Tricyclohexyl-[4-[4-[3-[4-(diethylamino)phenyl]-4-oxophthalazin-1-yl]phenoxy]butyl]phosphanium NA 124800 NA NA NA NA BindingDB
PSMB1 4-[4-(4-Oxo-3-phenylphthalazin-1-yl)phenoxy]butyl-triphenylphosphanium NA 102700 NA NA NA NA BindingDB
PSMB10 N-((S)-3-Hydroxy-1-(((S)-1-((R)-2-methyloxiran-2-YL)-1-oxo-3-phenylpropan-2-YL)amino)-1-oxopropan-2-YL)-6-oxo-1,6-dihydropyridine-2-carboxamide NA 250000 NA NA NA NA TTD
PSMB10 4,5-Anhydro-1,2-dideoxy-2-[[(2S)-2-[[(1,6-dihydro-6-oxo-2-pyridinyl)carbonyl]amino]-3-(4-methoxyphenyl)-1-oxopropyl]amino]-4-C-methyl-1-phenyl-D-erythro-3-pentulose NA 250000 NA NA NA NA TTD
PSMB10 N-[(2S)-1-[[(2S)-1-[(2R)-2-methyloxiran-2-yl]-1-oxo-3-phenylpropan-2-yl]amino]-1-oxopropan-2-yl]-6-oxo-1H-pyridine-2-carboxamide NA 250000 NA NA NA NA TTD
PSMB10 methyl 3-[[(2S)-3-[(3R)-3-hydroxy-2-oxo-1H-indol-3-yl]-2-[[(2S)-2-[[(2S)-2-[(2-methylpropan-2-yl)oxycarbonylamino]-3-(4-phenylmethoxyphenyl)propanoyl]amino]propanoyl]amino]propanoyl]amino]propanoate NA 106000 NA NA NA NA TTD
PSMB2 (2S)-N-[(2S)-1-[[(2S)-1-[5-[4-(dimethylamino)phenyl]-1,3,4-oxadiazol-2-yl]-4-methyl-1-oxopentan-2-yl]amino]-1-oxopropan-2-yl]-N'-(2,2-dimethylpropyl)-2-[(4-methylphenyl)sulfonylamino]butanediamide 290000 NA NA NA NA NA BindingDB
PSMB2 4-[4-[3-(2-Methylpropyl)-4-oxophthalazin-1-yl]phenoxy]butyl-triphenylphosphanium NA 276200 NA NA NA NA BindingDB
PSMB2 4-[4-[3-(Cyclopropylmethyl)-4-oxophthalazin-1-yl]phenoxy]butyl-triphenylphosphanium NA 588700 NA NA NA NA BindingDB
PSMB2 4-[4-[3-(Cyclobutylmethyl)-4-oxophthalazin-1-yl]phenoxy]butyl-triphenylphosphanium NA 475200 NA NA NA NA BindingDB