| GENE_SYMBOL |
DRUG_NAME |
Ki (nM) |
IC50 (nM) |
Kd (nM) |
EC50 (nM) |
Potency (nM) |
AC50 (nM) |
Datasource |
| PRSS3 |
Xeruborbactam |
NA |
1000000 |
NA |
NA |
NA |
NA |
PubChem |
| PRSS3 |
Vaborbactam |
NA |
1000000 |
NA |
NA |
NA |
NA |
PubChem |
| PRSS3 |
Baicalin |
NA |
1000000 |
NA |
NA |
NA |
NA |
PubChem |
| PRSS3 |
2-(6-Hydroxy-4-methyl-1,3-benzothiazol-2-yl)guanidine |
794000 |
NA |
NA |
NA |
NA |
NA |
BindingDB |
| PRSS3 |
ethyl 2-[(2E)-2-carbamimidoylimino-6-hydroxy-1,3-benzothiazol-3-yl]acetate |
168000 |
NA |
NA |
NA |
NA |
NA |
BindingDB |
| PRSS3 |
2-(5-Chloro-6-hydroxy-1,3-benzothiazol-2-yl)guanidine |
476000 |
NA |
NA |
NA |
NA |
NA |
BindingDB |
| PRSS3 |
2-[(2E)-2-carbamimidoylimino-6-hydroxy-1,3-benzothiazol-3-yl]-N-ethylacetamide |
1094000 |
NA |
NA |
NA |
NA |
NA |
BindingDB |
| PRSS3 |
GW-813893 |
NA |
158000 |
NA |
NA |
NA |
NA |
PubChem |
| PRSS3 |
Dpoc-4088 |
202000 |
NA |
NA |
NA |
NA |
NA |
PubChem |
| PRTN3 |
6-(((5-(cyclopropanecarboxamido)-1,3,4-thiadiazol-2-yl)thio)methyl)-4-oxo-4H-pyran-3-yl 3-fluorobenzoate |
NA |
134000 |
NA |
NA |
NA |
NA |
TTD |
| PRTN3 |
2-[(5-amino-1H-1,2,4-triazol-3-yl)sulfanyl]-N-(3,5-dichlorophenyl)-2-phenylacetamide |
NA |
139000 |
NA |
NA |
NA |
NA |
TTD |
| PSEN1 |
N-[(3,4-dichlorophenyl)methyl]-N-propan-2-ylnaphthalene-2-carboxamide |
NA |
135000 |
NA |
NA |
NA |
NA |
TTD |
| PSEN1 |
9-octyl-2-(2H-tetrazol-5-ylmethoxy)carbazole |
NA |
102000 |
NA |
NA |
NA |
NA |
TTD |
| PSEN1 |
2-(9-Octylcarbazol-2-yl)oxyacetamide |
NA |
104000 |
NA |
NA |
NA |
NA |
TTD |
| PSEN1 |
2-(9-Octylcarbazol-2-yl)oxyacetonitrile |
NA |
105000 |
NA |
NA |
NA |
NA |
TTD |
| PSEN1 |
4-[4-[(Z)-(5-chloro-2-oxo-1H-indol-3-ylidene)methyl]-2-methoxyphenoxy]butanenitrile |
NA |
160000 |
NA |
NA |
NA |
NA |
TTD |
| PSEN1 |
Tarenflurbil |
NA |
307000 |
NA |
NA |
NA |
NA |
BindingDB|PubChem|TTD |
| PSEN2 |
Tarenflurbil |
NA |
307000 |
NA |
NA |
NA |
NA |
PubChem |
| PSENEN |
N-[(3,4-dichlorophenyl)methyl]-N-propan-2-ylnaphthalene-2-carboxamide |
NA |
135000 |
NA |
NA |
NA |
NA |
TTD |
| PSENEN |
[1-(1-Formyl-butylcarbamoyl)-3-methyl-butyl]-carbamic acid benzyl ester |
NA |
200000 |
NA |
NA |
NA |
NA |
BindingDB |