| GENE_SYMBOL |
DRUG_NAME |
Ki (nM) |
IC50 (nM) |
Kd (nM) |
EC50 (nM) |
Potency (nM) |
AC50 (nM) |
Datasource |
| PSMB5 |
1-[(1S,9R)-11-benzoyl-6-oxo-7,11-diazatricyclo[7.3.1.02,7]trideca-2,4-dien-5-yl]-3-(3-cyanophenyl)urea |
NA |
201000 |
NA |
NA |
NA |
NA |
BindingDB |
| PSMB5 |
1-(3-cyanophenyl)-3-[(1S,9R)-6-oxo-11-(pyridine-3-carbonyl)-7,11-diazatricyclo[7.3.1.02,7]trideca-2,4-dien-5-yl]urea |
NA |
440000 |
NA |
NA |
NA |
NA |
BindingDB |
| PSMB5 |
1-[(1S,9R)-11-acetyl-6-oxo-7,11-diazatricyclo[7.3.1.02,7]trideca-2,4-dien-5-yl]-3-(3-cyanophenyl)urea |
NA |
491000 |
NA |
NA |
NA |
NA |
BindingDB |
| PSMB5 |
Gallic Acid |
NA |
7100000 |
NA |
NA |
NA |
NA |
BindingDB|PubChem|TTD |
| PSMB5 |
Bortezomib |
NA |
512861000 |
NA |
NA |
NA |
NA |
PubChem |
| PSMB5 |
N-[(Phenylmethoxy)carbonyl]-L-leucyl-N-[(1S)-1-cyano-3-methylbutyl]-L-leucinamide |
450000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| PSMB5 |
N-[(2S)-1-[[(1R)-3-methyl-1-[(1S,2S,8S)-2,9,9-trimethyl-3,5-dioxa-4-boratricyclo[6.1.1.02,6]decan-4-yl]butyl]amino]-1-oxo-3-phenylpropan-2-yl]pyrazine-2-carboxamide |
NA |
524807460.3 |
NA |
NA |
NA |
NA |
TTD |
| PSMB5 |
Epigallocatechin |
NA |
1200000 |
NA |
NA |
NA |
NA |
BindingDB|PubChem|TTD |
| PSMB5 |
3-(5-methyl-7-oxo-3-phenyl-7H-furo[3,2-g]chromen-6-yl)propanoic acid |
NA |
172200 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| PSMB8 |
(2S)-3-[4-(aminomethyl)phenyl]-2-[[(2S)-2-[[(2S)-2-[[(2S)-2-amino-3-phenylpropanoyl]amino]-4-methylpentanoyl]amino]-4-methylpentanoyl]amino]propane-1-sulfonyl fluoride |
NA |
136500 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| PSMB8 |
N-(3-methyl-2-sulfanylidene-1H-benzimidazol-5-yl)acetamide |
NA |
149000 |
NA |
NA |
NA |
NA |
BindingDB|ChEMBL |
| PSMB8 |
N-(2-sulfanylidene-3H-1,3-benzoxazol-7-yl)benzamide |
NA |
129000 |
NA |
NA |
NA |
NA |
BindingDB|ChEMBL |
| PSMB8 |
2-pyridin-3-yl-N-(2-sulfanylidene-3H-1,3-benzoxazol-7-yl)acetamide |
NA |
156000 |
NA |
NA |
NA |
NA |
BindingDB|ChEMBL |
| PSMB8 |
(2R)-N-(3-methyl-2-sulfanylidene-1H-benzimidazol-5-yl)pyrrolidine-2-carboxamide |
NA |
109000 |
NA |
NA |
NA |
NA |
BindingDB|ChEMBL |
| PSMB8 |
N-(2-Sulfanylidene-2,3-dihydro-1,3-benzothiazol-6-yl)acetamide |
NA |
130000 |
NA |
NA |
NA |
NA |
BindingDB|ChEMBL |
| PSMB8 |
2-Benzimidazolethiol |
NA |
114000 |
NA |
NA |
NA |
NA |
BindingDB|ChEMBL |
| PTAFR |
Loratadine |
NA |
135000 |
NA |
NA |
NA |
NA |
BindingDB|PubChem|TTD |
| PTGER1 |
3-(2-((E)-3-(4-(benzyloxy)-3-methoxyphenyl)prop-1-enyl)phenyl)acrylic acid |
151350 |
NA |
NA |
NA |
NA |
NA |
TTD |
| PTGER2 |
7-{(R)-2-[(E)-3-Hydroxy-3-(1-phenyl-cyclopropyl)-propenyl]-5-oxo-pyrrolidin-1-yl}-heptanoic acid |
164000 |
NA |
NA |
NA |
NA |
NA |
BindingDB |
| PTGER3 |
7-{(R)-2-[(E)-3-Hydroxy-3-(3-trifluoromethyl-phenyl)-propenyl]-5-oxo-pyrrolidin-1-yl}-heptanoic acid |
131000 |
NA |
NA |
NA |
NA |
NA |
TTD |