| GENE_SYMBOL |
DRUG_NAME |
Ki (nM) |
IC50 (nM) |
Kd (nM) |
EC50 (nM) |
Potency (nM) |
AC50 (nM) |
Datasource |
| PTGER4 |
11-Deoxy-8-azaprostaglandin E(1) |
NA |
NA |
NA |
200000 |
NA |
NA |
BindingDB|TTD |
| PTGES |
3-(5-{[3-(2-Anilino-2-oxoethyl)-2,4-dioxo-1,3-thiazolidin-5-ylidene]methyl}-2-furyl)-4-methylbenzoic acid |
NA |
160000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| PTGES |
2-(4-Bromophenyl)-2-oxoethyl 1,3-dioxo-2-(4-phenoxyphenyl)-5-isoindolinecarboxylate |
NA |
200000 |
NA |
NA |
NA |
NA |
BindingDB |
| PTGES |
|
NA |
130000 |
NA |
NA |
NA |
NA |
BindingDB |
| PTGES |
(2E,5Z)-5-{3-bromo-4-[(4-nitrobenzyl)oxy]benzylidene}-3-(4-methoxybenzyl)-2-(phenylimino)-1,3-thiazolidin-4-one |
NA |
120000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| PTGES |
3,4,5-tris(benzyloxy)-N'-{4-nitrobenzylidene}benzohydrazide |
NA |
200000 |
NA |
NA |
NA |
NA |
BindingDB |
| PTGIS |
1H-Imidazole, 1-(2-phenoxyethyl)- |
NA |
1000000 |
NA |
NA |
NA |
NA |
TTD |
| PTGIS |
[4-(2-Imidazol-1-yl-ethoxy)-phenyl]-acetic acid ethyl ester |
NA |
1000000 |
NA |
NA |
NA |
NA |
TTD |
| PTGIS |
N-[4-(2-Imidazol-1-yl-ethoxy)-phenyl]-acetamide |
NA |
1000000 |
NA |
NA |
NA |
NA |
TTD |
| PTGIS |
5-[4-(2-Imidazol-1-yl-ethoxy)-phenyl]-1H-tetrazole |
NA |
1000000 |
NA |
NA |
NA |
NA |
TTD |
| PTGIS |
3-Imidazol-1-ylmethyl-1H-indole |
NA |
650000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| PTGIS |
Imidazole |
NA |
4000000 |
NA |
NA |
NA |
NA |
BindingDB|PubChem|TTD |
| PTGS1 |
6-formyl-2-trifluoromethyl-2H-chromene-3-carboxylic acid |
NA |
500000 |
NA |
NA |
NA |
NA |
TTD |
| PTGS1 |
4-(1-(4-(Aminosulfonyl)phenyl)-3-(trifluoromethyl)-1H-pyrazol-5-yl)benzoic acid |
NA |
250000 |
NA |
NA |
NA |
NA |
TTD |
| PTGS1 |
2-(5-Methoxy-1H-benzoimidazol-2-ylsulfanylmethyl)-3-pentadecyl-phenol |
NA |
384000 |
NA |
NA |
NA |
NA |
TTD |
| PTGS1 |
4-(4-Azido-phenyl)-3-phenyl-5H-furan-2-one |
NA |
159720 |
NA |
NA |
NA |
NA |
TTD |
| PTGS1 |
2-Butyl-1,3-dimethyl-5-[(4-phenylpiperazin-1-yl)methyl]pyrrolo[3,4-c]pyrrole-4,6-dione |
NA |
124400 |
NA |
NA |
NA |
NA |
TTD |
| PTGS1 |
5-[1-(4-Methanesulfonyl-phenyl)-4-trifluoromethyl-1H-imidazol-2-yl]-2-methyl-pyridine |
NA |
1000000 |
NA |
NA |
NA |
NA |
TTD |
| PTGS1 |
Osthol |
NA |
200000 |
NA |
NA |
NA |
NA |
PubChem|TTD |
| PTGS1 |
2-(2-Methoxy-6-pentadecyl-benzylsulfanyl)-benzothiazole |
NA |
500000 |
NA |
NA |
NA |
NA |
TTD |