| GENE_SYMBOL |
DRUG_NAME |
Ki (nM) |
IC50 (nM) |
Kd (nM) |
EC50 (nM) |
Potency (nM) |
AC50 (nM) |
Datasource |
| PTGS1 |
4-[2-(6-Methyl-pyridin-2-yl)-4-trifluoromethyl-imidazol-1-yl]-benzenesulfonamide |
NA |
1000000 |
NA |
NA |
NA |
NA |
TTD |
| PTGS1 |
Pyridine,2-methyl-6-[1-[4-(methylsulfonyl)phenyl]-4-(trifluoromethyl)-1h-imidazol-2-yl]- |
NA |
1000000 |
NA |
NA |
NA |
NA |
TTD |
| PTGS1 |
5-(4-Methanesulfonyl-phenyl)-2,3-dimethyl-4-phenyl-2,3-dihydro-isoxazole |
NA |
258110 |
NA |
NA |
NA |
NA |
TTD |
| PTGS1 |
4-[2-(2-Methyl-thiazol-4-yl)-4-trifluoromethyl-imidazol-1-yl]-benzenesulfonamide |
NA |
1000000 |
NA |
NA |
NA |
NA |
TTD |
| PTGS1 |
1-(4-Methanesulfonyl-phenyl)-2-o-tolyl-4-trifluoromethyl-1H-imidazole |
NA |
577000 |
NA |
NA |
NA |
NA |
TTD |
| PTGS1 |
Benzeneacetic acid, 2-[(3,5-dichlorophenyl)amino]- |
NA |
12589254.12 |
NA |
NA |
NA |
NA |
TTD |
| PTGS1 |
2-Carboxy-5-Maleimidophenyl Acetate |
NA |
300000 |
NA |
NA |
NA |
NA |
TTD |
| PTGS1 |
Oleanolic Acid |
NA |
380000 |
NA |
NA |
NA |
NA |
PubChem|TTD |
| PTGS1 |
2-[1-(4-Methanesulfonyl-phenyl)-4-trifluoromethyl-1H-imidazol-2-yl]-3-methyl-pyridine |
NA |
1000000 |
NA |
NA |
NA |
NA |
TTD |
| PTGS1 |
2-(3-Chloro-5-methyl-phenyl)-1-(4-methanesulfonyl-phenyl)-4-trifluoromethyl-1H-imidazole |
NA |
1000000 |
NA |
NA |
NA |
NA |
TTD |
| PTGS1 |
7-(2,5-dioxo-2,5-dihydro-1H-pyrrol-1-yl)heptanoic acid |
NA |
570000 |
NA |
NA |
NA |
NA |
TTD |
| PTGS1 |
4-[2-(2-Methyl-thiazol-5-yl)-4-trifluoromethyl-imidazol-1-yl]-benzenesulfonamide |
NA |
1000000 |
NA |
NA |
NA |
NA |
TTD |
| PTGS1 |
4-[5-(7-Methyl-benzo[1,3]dioxol-5-yl)-3-trifluoromethyl-pyrazol-1-yl]-benzenesulfonamide |
NA |
674000 |
NA |
NA |
NA |
NA |
TTD |
| PTGS1 |
4-(5-Pyridin-4-yl-3-trifluoromethyl-pyrazol-1-yl)-benzenesulfonamide |
NA |
209000 |
NA |
NA |
NA |
NA |
TTD |
| PTGS1 |
4,6-Dimethyl-5-phenyl-2-[(4-phenylpiperazin-1-yl)methyl]pyrrolo[3,4-c]pyrrole-1,3-dione |
NA |
129600 |
NA |
NA |
NA |
NA |
TTD |
| PTGS1 |
4-[2-(5-Bromo-pyridin-3-yl)-4-trifluoromethyl-imidazol-1-yl]-benzenesulfonamide |
NA |
1000000 |
NA |
NA |
NA |
NA |
TTD |
| PTGS1 |
4-[2-(5-Methyl-isoxazol-3-yl)-4-trifluoromethyl-imidazol-1-yl]-benzenesulfonamide |
NA |
1000000 |
NA |
NA |
NA |
NA |
TTD |
| PTGS1 |
4-[2-(5-Methyl-pyridin-2-yl)-4-trifluoromethyl-imidazol-1-yl]-benzenesulfonamide |
NA |
302000 |
NA |
NA |
NA |
NA |
TTD |
| PTGS1 |
1-[1-(4-Methanesulfonyl-phenyl)-4-trifluoromethyl-1H-imidazol-2-yl]-isoquinoline |
NA |
1000000 |
NA |
NA |
NA |
NA |
TTD |
| PTGS1 |
4'',5''-Difluoro-2''-(6-methyl-pyridin-3-yl)-biphenyl-4-sulfonic acid amide |
NA |
265000 |
NA |
NA |
NA |
NA |
TTD |