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Drugs And Genes
Negative Drug Target Genes
GENE_SYMBOL DRUG_NAME Ki (nM) IC50 (nM) Kd (nM) EC50 (nM) Potency (nM) AC50 (nM) Datasource
PTGS1 1-[4-(Methylsulfonyl)phenyl]-2-(2-methylthiazole-4-yl)-4-(trifluoromethyl)-1H-imidazole NA 1000000 NA NA NA NA TTD
PTGS1 2-(3-chloro-4-methoxyphenyl)-1-[4-(methylsulfonyl)phenyl]-4-trifluoromethyl-1H-imidazole NA 296000 NA NA NA NA TTD
PTGS1 3-Bromo-5-[1-(4-methanesulfonyl-phenyl)-4-trifluoromethyl-1H-imidazol-2-yl]-pyridine NA 1000000 NA NA NA NA TTD
PTGS1 2-[2-(2,5-Dioxopyrrol-1-yl)ethoxy]benzoic acid NA 250000 NA NA NA NA TTD
PTGS1 5-methyl-2-[1-[4-(methylsulfonyl)phenyl]-4-trifluoromethyl-1H-imidazol-2-yl]pyridine NA 1000000 NA NA NA NA TTD
PTGS1 3-[1-(4-Methanesulfonyl-phenyl)-4-trifluoromethyl-1H-imidazol-2-yl]-5-methyl-pyridine NA 1000000 NA NA NA NA TTD
PTGS1 [1-(4-Methanesulfonyl-phenyl)-2-pyridin-3-yl-1H-imidazol-4-yl]-methanol NA 1000000 NA NA NA NA TTD
PTGS1 1-(4-Methanesulfonyl-phenyl)-2-(3-methyl-thiophen-2-yl)-4-trifluoromethyl-1H-imidazole NA 1000000 NA NA NA NA TTD
PTGS1 3'-Hydroxydiclofenac NA 100000000 NA NA NA NA TTD
PTGS1 3-(4-Chloro-phenoxy)-2-(4-methanesulfonyl-phenyl)-6-methyl-pyran-4-one NA 207000 NA NA NA NA TTD
PTGS1 3-(4-Bromo-phenoxy)-2-(4-methanesulfonyl-phenyl)-6-methyl-pyran-4-one NA 119000 NA NA NA NA TTD
PTGS1 6,8-dimethyl-2-(trifluoromethyl)-2H-chromene-3-carboxylic Acid NA 169000 NA NA NA NA TTD
PTGS1 2-[[2-Anilinoethyl(methyl)amino]methyl]-4,6-dimethyl-[1,2]thiazolo[5,4-b]pyridin-3-one NA 173780.08 NA NA NA NA TTD
PTGS1 4'-Hydroxydiclofenac NA 7079460|7079457.84 NA NA NA NA PubChem|TTD
PTGS1 (R)-7-tert-butyl-6-chloro-2-(trifluoromethyl)-2H-chromene-3-carboxylic acid NA 136000 NA NA NA NA TTD
PTGS1 2-[[4-(2-Fluorophenyl)piperazin-1-yl]methyl]-4,6-dimethyl-[1,2]thiazolo[5,4-b]pyridin-3-one NA 141253.75 NA NA NA NA TTD
PTGS1 3-(4-Chloro-phenyl)-5-hydroxy-4-(4-methanesulfonyl-phenyl)-5-methyl-5H-furan-2-one NA 105000 NA NA NA NA TTD
PTGS1 1-[4-(Methylsulfonyl)phenyl]-2-(4-methyl-2-pyridinyl)-4-(trifluoromethyl)-1H-imidazole NA 1000000 NA NA NA NA TTD
PTGS1 2-(3-Fluoro-phenyl)-1-(4-methanesulfonyl-phenyl)-4-trifluoromethyl-1H-imidazole NA 1000000 NA NA NA NA TTD
PTGS1 2-(4-Bromo-thiophen-2-yl)-1-(4-methanesulfonyl-phenyl)-4-trifluoromethyl-1H-imidazole NA 1000000 NA NA NA NA TTD