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Drugs And Genes
Negative Drug Target Genes
GENE_SYMBOL DRUG_NAME Ki (nM) IC50 (nM) Kd (nM) EC50 (nM) Potency (nM) AC50 (nM) Datasource
PTPN1 5-(Biphenyl-3-yl-difluoro-methyl)-1-sodium-1H-tetrazole NA 195000 NA NA NA NA BindingDB
PTPN1 Sodium; biphenyl-3-yl-difluoro-acetate NA 435000 NA NA NA NA BindingDB
PTPN1 2-Fluoro-2-(naphthalen-2-yloxy)-malonic acid NA 320000 NA NA NA NA BindingDB
PTPN1 {3-[(1Z)-3-(allyloxy)-3-oxoprop-1-enyl]phenyl}(difluoro)methylphosphonate; diammonium salt NA|8000000 12200000|NA NA NA NA NA BindingDB
PTPN1 2-(2-methyl-4,5-disulfophenyl)-3-oxo-1H-pyrazole-5-carboxylic acid NA 118000 NA NA NA NA BindingDB
PTPN1 NA 460000 NA NA NA NA BindingDB
PTPN1 3-Phenylsalicylic acid NA 859000 NA NA NA NA BindingDB|TTD
PTPN1 1-(4-Hydroxy-3-methoxyphenyl)-3-(naphthalen-2-yl)prop-2-en-1-one NA 123030 NA NA NA NA BindingDB|TTD
PTPN1 (2S)-N-[(1S)-1-carbamoyl-2-{4-[(5S)-1,1,3-trioxo-1$l^{6},2-thiazolidin-5-yl]phenyl}ethyl]-2-acetamido-3-phenylpropanamide NA 179887 NA NA NA NA BindingDB
PTPN1 N-acetyl-L-phenylalanyl-4-(difluoro(phosphono)methyl)-L-phenylalaninamide NA 1749847 NA NA NA NA BindingDB
PTPN1 4-Bromo-3-(carboxymethoxy)thiophene-2-carboxylic acid 160000 NA NA NA NA NA BindingDB|TTD
PTPN1 2-[4-[4-(2-Benzyl-1-benzothiophen-3-yl)phenyl]-2-(4-methoxyphenyl)phenoxy]acetic acid NA 79400000 NA NA NA NA BindingDB
PTPN1 5-[4'-(2-Benzyl-benzofuran-3-yl)-biphenyl-4-yloxysulfonyl]-2-hydroxy-benzoic acid NA 27500000|27542287.03 NA NA NA NA BindingDB|TTD
PTPN1 [4''-(2-Butyl-benzofuran-3-ylmethyl)-biphenyl-4-yloxy]-acetic acid NA 870000000 NA NA NA NA BindingDB
PTPN1 3-[4'-(2-Benzyl-benzofuran-3-yl)-biphenyl-4-yloxysulfonyl]-benzoic acid NA 104000000 NA NA NA NA BindingDB
PTPN1 4-[4'-(2-Benzyl-benzo[b]thiophen-3-yl)-3,5-dibromo-biphenyl-4-yloxysulfonyl]-2-hydroxy-benzoic acid NA 30100000 NA NA NA NA BindingDB
PTPN1 2-(Naphthalen-2-yl)-2-oxoacetic acid NA 190000 NA NA NA NA BindingDB|TTD
PTPN1 Benzoic acid, 2-[(carboxycarbonyl)(2,3-dimethylphenyl)amino]- 293000 NA NA NA NA NA BindingDB
PTPN1 4''-((2-Butylbenzofuran-3-yl)methyl)biphenyl-4-ol NA 851000000 NA NA NA NA BindingDB
PTPN1 (2-Butyl-benzofuran-3-yl)-(4'-hydroxy-biphenyl-4-yl)-methanone NA 3980000|3981071.71 NA NA NA NA BindingDB|TTD