| GENE_SYMBOL |
DRUG_NAME |
Ki (nM) |
IC50 (nM) |
Kd (nM) |
EC50 (nM) |
Potency (nM) |
AC50 (nM) |
Datasource |
| PTPN1 |
3,5-Dibromo-4''-[(2-butyl-benzofuran-3-yl)-hydroxy-methyl]-biphenyl-4-ol |
NA |
707000000 |
NA |
NA |
NA |
NA |
BindingDB |
| PTPN1 |
2-[4-[4-(2-Benzyl-1-benzothiophen-3-yl)phenyl]-2-bromo-6-(4-methoxyphenyl)phenoxy]acetic acid |
NA |
28800000 |
NA |
NA |
NA |
NA |
BindingDB |
| PTPN1 |
2-[4-[4-(2-Benzylbenzo[b]thiophen-3-yl)phenyl]-2,6-di(4-methoxyphenyl)phenoxy]acetic acid |
NA |
25100000 |
NA |
NA |
NA |
NA |
BindingDB |
| PTPN11 |
Oleanolic Acid |
NA |
120000 |
NA |
NA |
NA |
NA |
PubChem |
| PTPN11 |
3-[(3-Acetyl-2-methyl-1-benzofuran-5-yl)sulfamoyl]benzoic acid |
NA |
176000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| PTPN11 |
4-[5-[5-(1H-indol-3-ylmethyl)-1,2,4-oxadiazol-3-yl]thiophen-2-yl]aniline |
NA |
120000 |
NA |
NA |
NA |
NA |
TTD |
| PTPN11 |
4-[3-[5-(1H-indol-3-ylmethyl)-1,2,4-oxadiazol-3-yl]phenyl]aniline |
NA |
120000 |
NA |
NA |
NA |
NA |
TTD |
| PTPN11 |
5-(1H-indol-3-ylmethyl)-3-[6-(4-propoxyphenyl)pyridin-2-yl]-1,2,4-oxadiazole |
NA |
120000 |
NA |
NA |
NA |
NA |
TTD |
| PTPN11 |
5-(1H-indol-3-ylmethyl)-3-[5-(3-methylphenyl)thiophen-2-yl]-1,2,4-oxadiazole |
NA |
120000 |
NA |
NA |
NA |
NA |
TTD |
| PTPN11 |
3-[5-(4-ethylphenyl)thiophen-2-yl]-5-(1H-indol-3-ylmethyl)-1,2,4-oxadiazole |
NA |
120000 |
NA |
NA |
NA |
NA |
TTD |
| PTPN11 |
5-(1H-indol-3-ylmethyl)-3-[5-(4-propylphenyl)thiophen-2-yl]-1,2,4-oxadiazole |
NA |
120000 |
NA |
NA |
NA |
NA |
TTD |
| PTPN11 |
3-[5-(4-butylphenyl)thiophen-2-yl]-5-(1H-indol-3-ylmethyl)-1,2,4-oxadiazole |
NA |
120000 |
NA |
NA |
NA |
NA |
TTD |
| PTPN11 |
3-[5-(4-ethoxyphenyl)thiophen-2-yl]-5-(1H-indol-3-ylmethyl)-1,2,4-oxadiazole |
NA |
120000 |
NA |
NA |
NA |
NA |
TTD |
| PTPN11 |
5-(1H-indol-3-ylmethyl)-3-[5-(4-propoxyphenyl)thiophen-2-yl]-1,2,4-oxadiazole |
NA |
120000 |
NA |
NA |
NA |
NA |
TTD |
| PTPN11 |
methyl 4-[4-[5-[5-(1H-indol-3-ylmethyl)-1,2,4-oxadiazol-3-yl]thiophen-2-yl]phenoxy]butanoate |
NA |
120000 |
NA |
NA |
NA |
NA |
TTD |
| PTPN11 |
3-(5-bromothiophen-2-yl)-5-(1H-indol-3-ylmethyl)-1,2,4-oxadiazole |
NA |
120000 |
NA |
NA |
NA |
NA |
TTD |
| PTPN11 |
3-(3-bromophenyl)-5-(1H-indol-3-ylmethyl)-1,2,4-oxadiazole |
NA |
120000 |
NA |
NA |
NA |
NA |
TTD |
| PTPN11 |
4-[3-[5-(1H-indol-3-ylmethyl)-1,2,4-oxadiazol-3-yl]phenyl]phenol |
NA |
120000 |
NA |
NA |
NA |
NA |
TTD |
| PTPN11 |
5-(1H-indol-3-ylmethyl)-3-[3-(2-methylphenyl)phenyl]-1,2,4-oxadiazole |
NA |
120000 |
NA |
NA |
NA |
NA |
TTD |
| PTPN11 |
5-(1H-indol-3-ylmethyl)-3-[3-(3-methylphenyl)phenyl]-1,2,4-oxadiazole |
NA |
120000 |
NA |
NA |
NA |
NA |
TTD |