| GENE_SYMBOL |
DRUG_NAME |
Ki (nM) |
IC50 (nM) |
Kd (nM) |
EC50 (nM) |
Potency (nM) |
AC50 (nM) |
Datasource |
| PTPN11 |
5-(1H-indol-3-ylmethyl)-3-[3-(4-propylphenyl)phenyl]-1,2,4-oxadiazole |
NA |
120000 |
NA |
NA |
NA |
NA |
TTD |
| PTPN11 |
3-[3-(4-butylphenyl)phenyl]-5-(1H-indol-3-ylmethyl)-1,2,4-oxadiazole |
NA |
120000 |
NA |
NA |
NA |
NA |
TTD |
| PTPN11 |
3-(6-bromopyridin-2-yl)-5-(1H-indol-3-ylmethyl)-1,2,4-oxadiazole |
NA |
120000 |
NA |
NA |
NA |
NA |
TTD |
| PTPN11 |
5-(1H-indol-3-ylmethyl)-3-[5-(2-methylphenyl)thiophen-2-yl]-1,2,4-oxadiazole |
NA |
120000 |
NA |
NA |
NA |
NA |
TTD |
| PTPN11 |
3-[3-(4-ethoxyphenyl)phenyl]-5-(1H-indol-3-ylmethyl)-1,2,4-oxadiazole |
NA |
120000 |
NA |
NA |
NA |
NA |
TTD |
| PTPN11 |
5-(1H-indol-3-ylmethyl)-3-[3-(4-propoxyphenyl)phenyl]-1,2,4-oxadiazole |
NA |
120000 |
NA |
NA |
NA |
NA |
TTD |
| PTPN11 |
methyl 4-[4-[3-[5-(1H-indol-3-ylmethyl)-1,2,4-oxadiazol-3-yl]phenyl]phenoxy]butanoate |
NA |
120000 |
NA |
NA |
NA |
NA |
TTD |
| PTPN11 |
5-(1H-indol-3-ylmethyl)-3-[6-(2-methylphenyl)pyridin-2-yl]-1,2,4-oxadiazole |
NA |
120000 |
NA |
NA |
NA |
NA |
TTD |
| PTPN11 |
5-(1H-indol-3-ylmethyl)-3-[6-(3-methylphenyl)pyridin-2-yl]-1,2,4-oxadiazole |
NA |
120000 |
NA |
NA |
NA |
NA |
TTD |
| PTPN11 |
3-[6-(4-butylphenyl)pyridin-2-yl]-5-(1H-indol-3-ylmethyl)-1,2,4-oxadiazole |
NA |
120000 |
NA |
NA |
NA |
NA |
TTD |
| PTPN11 |
3-[6-(4-ethoxyphenyl)pyridin-2-yl]-5-(1H-indol-3-ylmethyl)-1,2,4-oxadiazole |
NA |
120000 |
NA |
NA |
NA |
NA |
TTD |
| PTPN11 |
3-(1,1,1,3,3,3-Hexafluoro-2-hydroxypropan-2-yl)naphthalen-2-ol |
NA |
114800 |
NA |
NA |
NA |
NA |
TTD |
| PTPN11 |
2-(1,1,1,3,3,3-Hexafluoro-2-hydroxypropan-2-yl)-5-phenylphenol |
NA |
500000 |
NA |
NA |
NA |
NA |
TTD |
| PTPN11 |
2-(1,1,1,3,3,3-Hexafluoro-2-hydroxypropan-2-yl)-4-phenylphenol |
NA |
392200 |
NA |
NA |
NA |
NA |
TTD |
| PTPN11 |
2-(1,1,1,3,3,3-Hexafluoro-2-hydroxypropan-2-yl)-6-phenylphenol |
NA |
136000 |
NA |
NA |
NA |
NA |
TTD |
| PTPN11 |
(2E,5E)-5-[(4-nitrophenyl)methylidene]-2-(1,3-thiazol-2-ylimino)-1,3-thiazolidin-4-one |
473600 |
NA |
NA |
NA |
NA |
NA |
TTD |
| PTPN11 |
(2E,5E)-5-[(4-hydroxyphenyl)methylidene]-2-(1,3-thiazol-2-ylimino)-1,3-thiazolidin-4-one |
388000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| PTPN11 |
(2E,5E)-5-[(3-nitrophenyl)methylidene]-2-(1,3-thiazol-2-ylimino)-1,3-thiazolidin-4-one |
547500 |
NA |
NA |
NA |
NA |
NA |
TTD |
| PTPN11 |
(2E,5E)-5-[(3-chlorophenyl)methylidene]-2-(1,3-thiazol-2-ylimino)-1,3-thiazolidin-4-one |
1088200 |
NA |
NA |
NA |
NA |
NA |
TTD |
| PTPN11 |
(2E,5E)-5-[(4-hydroxy-3-methoxyphenyl)methylidene]-2-[(4-phenyl-1,3-thiazol-2-yl)imino]-1,3-thiazolidin-4-one |
103200 |
NA |
NA |
NA |
NA |
NA |
TTD |