| GENE_SYMBOL |
DRUG_NAME |
Ki (nM) |
IC50 (nM) |
Kd (nM) |
EC50 (nM) |
Potency (nM) |
AC50 (nM) |
Datasource |
| PTPN11 |
4-[6-[5-(1H-indol-3-ylmethyl)-1,2,4-oxadiazol-3-yl]pyridin-2-yl]phenol |
NA |
120000 |
NA |
NA |
NA |
NA |
TTD |
| PTPN11 |
2-(1,1,1,3,3,3-Hexafluoro-2-hydroxypropan-2-yl)-4-methylphenol |
NA |
201800 |
NA |
NA |
NA |
NA |
TTD |
| PTPN11 |
|
473600 |
NA |
NA |
NA |
NA |
NA |
BindingDB |
| PTPN11 |
|
388000 |
NA |
NA |
NA |
NA |
NA |
BindingDB |
| PTPN11 |
|
547500 |
NA |
NA |
NA |
NA |
NA |
BindingDB |
| PTPN11 |
|
1088200 |
NA |
NA |
NA |
NA |
NA |
BindingDB |
| PTPN11 |
|
103200 |
NA |
NA |
NA |
NA |
NA |
BindingDB |
| PTPN11 |
(2E)-3-[3-chloro-4-(4-fluorophenyl)phenyl]prop-2-enoic acid |
NA |
500000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| PTPN11 |
Estramustine |
NA |
300000 |
NA |
NA |
NA |
NA |
PubChem|TTD |
| PTPN11 |
2-(2-Hydroxy-1,1,1,3,3,3-hexafluoropropyl)-1-naphthol |
NA |
500000 |
NA |
NA |
NA |
NA |
TTD |
| PTPN11 |
4-[Acetyl(6,7,8,9-tetrahydrodibenzofuran-2-yl)sulfamoyl]benzoic acid |
NA |
181000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| PTPN11 |
Genipin |
NA |
500000 |
NA |
NA |
NA |
NA |
PubChem |
| PTPN11 |
US8623906, XW2-038G |
NA |
143600 |
NA |
NA |
NA |
NA |
BindingDB |
| PTPN11 |
3-Ethynyl-6-hydroxy-1-methyl-2-phenyl-1H-indole-5-carboxylic Acid |
NA |
212000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| PTPN11 |
Ethoxy-[[3-[[[ethoxy(hydroxy)phosphoryl]-(2-hydroxyphenyl)methyl]amino]propylamino]-(2-hydroxyphenyl)methyl]phosphinic acid |
NA |
10000000 |
NA |
NA |
NA |
NA |
TTD |
| PTPN11 |
Azane;[[4-[2-[[4-[difluoro(phosphono)methyl]phenyl]methoxy]ethoxymethyl]phenyl]-difluoromethyl]phosphonic acid |
NA |
152000 |
NA |
NA |
NA |
NA |
TTD |
| PTPN11 |
{3(S)-Methylcarbamoyl-2-[3-(3-sulfoamino-phenyl)-propionyl]-1,2,3,4-tetrahydro-isoquinolin-7-YL}-sulfamic acid |
NA |
500000 |
NA |
NA |
NA |
NA |
TTD |
| PTPN11 |
(6R,8'R,9'S,13'S,14'S)-N,N-bis(2-chloroethyl)-3'-methoxy-13'-methyl-2-oxospiro[1,3,2lambda5-oxazaphosphinane-6,17'-7,8,9,11,12,14,15,16-octahydro-6H-cyclopenta[a]phenanthrene]-2-amine |
NA |
300000 |
NA |
NA |
NA |
NA |
TTD |
| PTPN11 |
Ethoxy-[[2-[[[ethoxy(hydroxy)phosphoryl]-(2-hydroxyphenyl)methyl]amino]ethylamino]-(2-hydroxyphenyl)methyl]phosphinic acid |
NA |
10000000 |
NA |
NA |
NA |
NA |
TTD |
| PTPN11 |
Phosphonic acid, P,Pa(2)-[1,6-hexanediylbis[imino[(2-hydroxyphenyl)methylene]]]bis-, P,Pa(2)-diethyl ester |
NA |
10000000 |
NA |
NA |
NA |
NA |
TTD |