| GENE_SYMBOL |
DRUG_NAME |
Ki (nM) |
IC50 (nM) |
Kd (nM) |
EC50 (nM) |
Potency (nM) |
AC50 (nM) |
Datasource |
| PTPN11 |
sodium;(2S)-2-[[[ethoxy(hydroxy)phosphoryl]-(2-hydroxyphenyl)methyl]amino]-3-(1H-indol-3-yl)propanoate |
NA |
10000000 |
NA |
NA |
NA |
NA |
TTD |
| PTPN11 |
2-[(S)-(4-chloroanilino)-diethoxyphosphorylmethyl]phenol |
NA |
10000000 |
NA |
NA |
NA |
NA |
TTD |
| PTPN11 |
Estradiol |
NA |
300000 |
NA |
NA |
NA |
NA |
PubChem|TTD |
| PTPN11 |
Vanadate(3-) |
NA |
209000 |
NA |
NA |
NA |
NA |
BindingDB |
| PTPN11 |
alpha,alpha-Bis(trifluoromethyl)benzyl alcohol |
NA |
500000 |
NA |
NA |
NA |
NA |
TTD |
| PTPN11 |
5-Oxo-1-(4-sulfophenyl)-2,5-dihydro-1H-pyrazole-3-carboxylic acid |
NA |
155000 |
NA |
NA |
NA |
NA |
BindingDB |
| PTPN11 |
(2S)-2-[[[ethoxy(hydroxy)phosphoryl]-(2-hydroxyphenyl)methyl]amino]-3-hydroxypropanoate |
NA |
191000 |
NA |
NA |
NA |
NA |
BindingDB |
| PTPN11 |
(2S)-2-[[[ethoxy(hydroxy)phosphoryl]-(2-hydroxyphenyl)methyl]amino]-3-(1H-imidazol-5-yl)propanoate |
NA |
210000 |
NA |
NA |
NA |
NA |
BindingDB |
| PTPN11 |
tetra ammonium [(4-{2-[4-(Difluoro-phosphono-methyl)-benzyloxy]-ethoxymethyl}-phenyl)-difluoro-methyl]-phosphonic acid |
NA |
152000 |
NA |
NA |
NA |
NA |
BindingDB |
| PTPN2 |
Oleanolic Acid |
NA |
120000 |
NA |
NA |
NA |
NA |
PubChem |
| PTPN2 |
2-Hydroxy-5-(5-(((1-hydroxy-2,2,6,6-tetramethylpiperidin-4-yl)amino)methyl)furan-2-yl)benzoic acid |
NA |
685000 |
NA |
NA |
NA |
NA |
BindingDB |
| PTPN2 |
(E)-2,2,6,6-tetramethyl-4-(3-(5-(3-nitrophenyl)furan-2-yl)acrylamido)piperidin-1-olate |
NA |
260000 |
NA |
NA |
NA |
NA |
BindingDB |
| PTPN2 |
Pyrrospirone N |
NA |
130000 |
NA |
NA |
NA |
NA |
BindingDB |
| PTPN2 |
2-[(5Z)-4-oxo-5-[[4-(4-phenylbutoxy)phenyl]methylidene]-2-sulfanylidene-1,3-thiazolidin-3-yl]acetic acid |
NA |
192700 |
NA |
NA |
NA |
NA |
BindingDB |
| PTPN2 |
5,5''-Methylenebis(2-hydroxybiphenyl-3-carboxylic acid) |
NA |
291000 |
NA |
NA |
NA |
NA |
BindingDB |
| PTPN2 |
5-Benzyl-2-hydroxybiphenyl-3-carboxylic acid |
NA |
540000 |
NA |
NA |
NA |
NA |
BindingDB |
| PTPN2 |
2-{4-[2-Acetamido-2-({4-[3-hydroxy-2-(methoxycarbonyl)phenoxy]butyl}carbamoyl)ethyl]-2-hydroxyphenoxy}acetic acid |
182000 |
NA |
NA |
NA |
NA |
NA |
BindingDB |
| PTPN2 |
({4-[(2S)-2-{[(tert-butoxy)carbonyl]amino}-2-({4-[3-hydroxy-2-(methoxycarbonyl)phenoxy]butyl}carbamoyl)ethyl]phenyl}carbamoyl)formic acid |
141000 |
NA |
NA |
NA |
NA |
NA |
BindingDB |
| PTPN2 |
5,5''-Methylenebis(4-hydroxybiphenyl-3-carboxylic acid) |
NA |
156000 |
NA |
NA |
NA |
NA |
BindingDB |
| PTPN2 |
4-Oxo-6-phenyl-4H-chromene-3-carbaldehyde |
NA |
240000 |
NA |
NA |
NA |
NA |
BindingDB |