| GENE_SYMBOL |
DRUG_NAME |
Ki (nM) |
IC50 (nM) |
Kd (nM) |
EC50 (nM) |
Potency (nM) |
AC50 (nM) |
Datasource |
| PTPN2 |
(2S)-2-amino-N-[(2R)-1-[[2-(2,3-dihydro-1H-inden-1-ylamino)-2-oxoethyl]amino]-1-oxopropan-2-yl]-3-(4-hydroxyphenyl)propanamide |
NA |
101900 |
NA |
NA |
NA |
NA |
BindingDB |
| PTPN2 |
1-Oxobenzo[f]chromene-2-carbaldehyde |
NA |
780000 |
NA |
NA |
NA |
NA |
BindingDB |
| PTPN2 |
[4-[3-[(S)-(3,4-dichlorophenyl)-hydroxymethyl]phenyl]benzoyl]-trihydroxyphosphanium |
170000 |
NA |
NA |
NA |
NA |
NA |
BindingDB |
| PTPN2 |
[4-[3-[(R)-(3,4-dichlorophenyl)-hydroxymethyl]phenyl]benzoyl]-trihydroxyphosphanium |
164000 |
NA |
NA |
NA |
NA |
NA |
BindingDB |
| PTPN2 |
(2S)-2-[[[ethoxy(hydroxy)phosphoryl]-(2-hydroxyphenyl)methyl]amino]-3-hydroxypropanoate |
NA |
123000 |
NA |
NA |
NA |
NA |
BindingDB |
| PTPN2 |
(2S)-2-[[[ethoxy(hydroxy)phosphoryl]-(2-hydroxyphenyl)methyl]amino]-3-(1H-imidazol-5-yl)propanoate |
NA |
178000 |
NA |
NA |
NA |
NA |
BindingDB |
| PTPN2 |
ammonium N-{4-[4-ethoxy-2,2-bis(methoxycarbonyl)-4-oxobutyl]phenyl}sulfamate |
NA |
109000 |
NA |
NA |
NA |
NA |
BindingDB |
| PTPN2 |
Benzoic acid, 2-[(carboxycarbonyl)(2,3-dimethylphenyl)amino]- |
164000 |
NA |
NA |
NA |
NA |
NA |
BindingDB |
| PTPN2 |
5-(3-(3-(3-Hydroxy-2-(methoxycarbonyl)phenoxy)prop-1-enyl)phenyl)isoxazole-3-carboxylic acid |
202000 |
NA |
NA |
NA |
NA |
NA |
BindingDB |
| PTPN22 |
Cefsulodin |
NA |
200000 |
NA |
NA |
NA |
NA |
PubChem |
| PTPN4 |
[(4-{4-[4-(Difluoro-phosphono-methyl)-benzyloxy]-phenoxymethyl}-phenyl)-difluoro-methyl]-phosphonic acid |
NA |
146000 |
NA |
NA |
NA |
NA |
BindingDB |
| PTPN5 |
4-(5-bromo-1,3-dioxo-1,3-dihydro-2H-isoindol-2-yl)-2-hydroxybenzoic acid |
NA |
273200 |
NA |
NA |
NA |
NA |
BindingDB |
| PTPN5 |
1-[3-Piperidin-4-yl-5-(trifluoromethyl)phenyl]guanidine |
NA |
NA |
800000|8e+05 |
NA |
NA |
NA |
BindingDB|ChEMBL |
| PTPN5 |
N-[4-(1,3-benzoxazol-2-yl)phenyl]-3-chlorobenzenesulfonamide |
NA |
545000 |
NA |
NA |
NA |
NA |
BindingDB |
| PTPN5 |
1,1''-Biphenyl-3-yl(difluoro)methylphosphonate |
337000 |
NA |
NA |
NA |
NA |
NA |
BindingDB |
| PTPN5 |
[Difluoro-(3-phenylphenyl)methyl]phosphonic acid |
337000 |
NA |
NA |
NA |
NA |
NA |
ChEMBL |
| PTPN5 |
Biphenyl-4-yldifluoromethylphosphonic acid |
120000 |
NA |
NA |
NA |
NA |
NA |
BindingDB|ChEMBL |
| PTPN5 |
[Difluoro-[3-(4-methylphenyl)phenyl]methyl]phosphonic acid |
205000 |
NA |
NA |
NA |
NA |
NA |
BindingDB|ChEMBL |
| PTPN5 |
[Difluoro-[3-(4-propan-2-ylphenyl)phenyl]methyl]phosphonic acid |
222000 |
NA |
NA |
NA |
NA |
NA |
BindingDB|ChEMBL |
| PTPN5 |
[Difluoro-[3-(3-methylphenyl)phenyl]methyl]phosphonic acid |
137000 |
NA |
NA |
NA |
NA |
NA |
BindingDB|ChEMBL |