| GENE_SYMBOL |
DRUG_NAME |
Ki (nM) |
IC50 (nM) |
Kd (nM) |
EC50 (nM) |
Potency (nM) |
AC50 (nM) |
Datasource |
| PTPN5 |
[Difluoro-[3-(2-hydroxyphenyl)phenyl]methyl]phosphonic acid |
168000 |
NA |
NA |
NA |
NA |
NA |
BindingDB|ChEMBL |
| PTPN5 |
[Difluoro-[3-(2-methoxyphenyl)phenyl]methyl]phosphonic acid |
271000 |
NA |
NA |
NA |
NA |
NA |
BindingDB|ChEMBL |
| PTPN5 |
[[3-(3-Ethyl-2-hydroxyphenyl)phenyl]-difluoromethyl]phosphonic acid |
124000 |
NA |
NA |
NA |
NA |
NA |
BindingDB|ChEMBL |
| PTPN5 |
[[4-(2-Cyanophenyl)phenyl]-difluoromethyl]phosphonic acid |
375000 |
NA |
NA |
NA |
NA |
NA |
BindingDB|ChEMBL |
| PTPN5 |
[[4-(3-Cyanophenyl)phenyl]-difluoromethyl]phosphonic acid |
400000|4e+05 |
NA |
NA |
NA |
NA |
NA |
BindingDB|ChEMBL |
| PTPN5 |
[[4-(4-Cyanophenyl)phenyl]-difluoromethyl]phosphonic acid |
617000 |
NA |
NA |
NA |
NA |
NA |
BindingDB|ChEMBL |
| PTPN5 |
[Difluoro-[4-(3-propan-2-yloxyphenyl)phenyl]methyl]phosphonic acid |
200000|2e+05 |
NA |
NA |
NA |
NA |
NA |
BindingDB|ChEMBL |
| PTPN5 |
[Difluoro-[4-(4-propan-2-yloxyphenyl)phenyl]methyl]phosphonic acid |
231000 |
NA |
NA |
NA |
NA |
NA |
BindingDB|ChEMBL |
| PTPN5 |
[Difluoro-[4-(3-propan-2-ylphenyl)phenyl]methyl]phosphonic acid |
132000 |
NA |
NA |
NA |
NA |
NA |
BindingDB|ChEMBL |
| PTPN5 |
[Difluoro-[4-(4-propan-2-ylphenyl)phenyl]methyl]phosphonic acid |
185000 |
NA |
NA |
NA |
NA |
NA |
BindingDB|ChEMBL |
| PTPN5 |
[Difluoro-[4-[2-(methanesulfonamido)phenyl]phenyl]methyl]phosphonic acid |
673000 |
NA |
NA |
NA |
NA |
NA |
BindingDB |
| PTPN5 |
[Difluoro-[4-[3-(methanesulfonamido)phenyl]phenyl]methyl]phosphonic acid |
113000 |
NA |
NA |
NA |
NA |
NA |
BindingDB |
| PTPN5 |
[Difluoro-[4-[4-(1-hydroxyethyl)phenyl]phenyl]methyl]phosphonic acid |
450000 |
NA |
NA |
NA |
NA |
NA |
BindingDB|ChEMBL |
| PTPN5 |
[[4-(3-Anilinophenyl)phenyl]-difluoromethyl]phosphonic acid |
112000 |
NA |
NA |
NA |
NA |
NA |
BindingDB |
| PTPN6 |
Oleanolic Acid |
NA |
120000 |
NA |
NA |
NA |
NA |
PubChem |
| PTPN6 |
4-[5-[5-(1H-indol-3-ylmethyl)-1,2,4-oxadiazol-3-yl]thiophen-2-yl]aniline |
NA |
120000 |
NA |
NA |
NA |
NA |
TTD |
| PTPN6 |
4-[3-[5-(1H-indol-3-ylmethyl)-1,2,4-oxadiazol-3-yl]phenyl]aniline |
NA |
120000 |
NA |
NA |
NA |
NA |
TTD |
| PTPN6 |
5-(1H-indol-3-ylmethyl)-3-[6-(4-propoxyphenyl)pyridin-2-yl]-1,2,4-oxadiazole |
NA |
120000 |
NA |
NA |
NA |
NA |
TTD |
| PTPN6 |
5-(1H-indol-3-ylmethyl)-3-[5-(3-methylphenyl)thiophen-2-yl]-1,2,4-oxadiazole |
NA |
120000 |
NA |
NA |
NA |
NA |
TTD |
| PTPN6 |
3-[5-(4-ethylphenyl)thiophen-2-yl]-5-(1H-indol-3-ylmethyl)-1,2,4-oxadiazole |
NA |
120000 |
NA |
NA |
NA |
NA |
TTD |