| GENE_SYMBOL |
DRUG_NAME |
Ki (nM) |
IC50 (nM) |
Kd (nM) |
EC50 (nM) |
Potency (nM) |
AC50 (nM) |
Datasource |
| PTPN6 |
5-(1H-indol-3-ylmethyl)-3-[5-(4-propylphenyl)thiophen-2-yl]-1,2,4-oxadiazole |
NA |
120000 |
NA |
NA |
NA |
NA |
TTD |
| PTPN6 |
3-[5-(4-butylphenyl)thiophen-2-yl]-5-(1H-indol-3-ylmethyl)-1,2,4-oxadiazole |
NA |
120000 |
NA |
NA |
NA |
NA |
TTD |
| PTPN6 |
3-[5-(4-ethoxyphenyl)thiophen-2-yl]-5-(1H-indol-3-ylmethyl)-1,2,4-oxadiazole |
NA |
120000 |
NA |
NA |
NA |
NA |
TTD |
| PTPN6 |
5-(1H-indol-3-ylmethyl)-3-[5-(4-propoxyphenyl)thiophen-2-yl]-1,2,4-oxadiazole |
NA |
120000 |
NA |
NA |
NA |
NA |
TTD |
| PTPN6 |
methyl 4-[4-[5-[5-(1H-indol-3-ylmethyl)-1,2,4-oxadiazol-3-yl]thiophen-2-yl]phenoxy]butanoate |
NA |
120000 |
NA |
NA |
NA |
NA |
TTD |
| PTPN6 |
3-(5-bromothiophen-2-yl)-5-(1H-indol-3-ylmethyl)-1,2,4-oxadiazole |
NA |
120000 |
NA |
NA |
NA |
NA |
TTD |
| PTPN6 |
3-(3-bromophenyl)-5-(1H-indol-3-ylmethyl)-1,2,4-oxadiazole |
NA |
120000 |
NA |
NA |
NA |
NA |
TTD |
| PTPN6 |
4-[3-[5-(1H-indol-3-ylmethyl)-1,2,4-oxadiazol-3-yl]phenyl]phenol |
NA |
120000 |
NA |
NA |
NA |
NA |
TTD |
| PTPN6 |
5-(1H-indol-3-ylmethyl)-3-[3-(2-methylphenyl)phenyl]-1,2,4-oxadiazole |
NA |
120000 |
NA |
NA |
NA |
NA |
TTD |
| PTPN6 |
5-(1H-indol-3-ylmethyl)-3-[3-(3-methylphenyl)phenyl]-1,2,4-oxadiazole |
NA |
120000 |
NA |
NA |
NA |
NA |
TTD |
| PTPN6 |
5-(1H-indol-3-ylmethyl)-3-[3-(4-propylphenyl)phenyl]-1,2,4-oxadiazole |
NA |
120000 |
NA |
NA |
NA |
NA |
TTD |
| PTPN6 |
3-[3-(4-butylphenyl)phenyl]-5-(1H-indol-3-ylmethyl)-1,2,4-oxadiazole |
NA |
120000 |
NA |
NA |
NA |
NA |
TTD |
| PTPN6 |
3-(6-bromopyridin-2-yl)-5-(1H-indol-3-ylmethyl)-1,2,4-oxadiazole |
NA |
120000 |
NA |
NA |
NA |
NA |
TTD |
| PTPN6 |
5-(1H-indol-3-ylmethyl)-3-[5-(2-methylphenyl)thiophen-2-yl]-1,2,4-oxadiazole |
NA |
120000 |
NA |
NA |
NA |
NA |
TTD |
| PTPN6 |
3-[3-(4-ethoxyphenyl)phenyl]-5-(1H-indol-3-ylmethyl)-1,2,4-oxadiazole |
NA |
120000 |
NA |
NA |
NA |
NA |
TTD |
| PTPN6 |
5-(1H-indol-3-ylmethyl)-3-[3-(4-propoxyphenyl)phenyl]-1,2,4-oxadiazole |
NA |
120000 |
NA |
NA |
NA |
NA |
TTD |
| PTPN6 |
methyl 4-[4-[3-[5-(1H-indol-3-ylmethyl)-1,2,4-oxadiazol-3-yl]phenyl]phenoxy]butanoate |
NA |
120000 |
NA |
NA |
NA |
NA |
TTD |
| PTPN6 |
5-(1H-indol-3-ylmethyl)-3-[6-(2-methylphenyl)pyridin-2-yl]-1,2,4-oxadiazole |
NA |
120000 |
NA |
NA |
NA |
NA |
TTD |
| PTPN6 |
5-(1H-indol-3-ylmethyl)-3-[6-(3-methylphenyl)pyridin-2-yl]-1,2,4-oxadiazole |
NA |
120000 |
NA |
NA |
NA |
NA |
TTD |
| PTPN6 |
3-[6-(4-butylphenyl)pyridin-2-yl]-5-(1H-indol-3-ylmethyl)-1,2,4-oxadiazole |
NA |
120000 |
NA |
NA |
NA |
NA |
TTD |