Navigator

      Support By : Li-lab

Drugs And Genes
Negative Drug Target Genes
GENE_SYMBOL DRUG_NAME Ki (nM) IC50 (nM) Kd (nM) EC50 (nM) Potency (nM) AC50 (nM) Datasource
PTPN1 4'-[(2-Butyl-benzofuran-3-yl)-hydroxymethyl]-biphenyl-4-ol NA 229000000 NA NA NA NA BindingDB
PTPN1 4-[4'-(2-Benzyl-benzofuran-3-yl)-biphenyl-4-yloxysulfonyl]-benzoic acid NA 75800000 NA NA NA NA BindingDB
PTPN1 (2R)-2-[4-[4-(2-benzyl-1-benzothiophen-3-yl)phenyl]-2-bromophenoxy]-3-phenylpropanoic acid NA 58800000 NA NA NA NA BindingDB
PTPN1 6-[(2-Butyl-benzofuran-3-yl)-hydroxy-methyl]-naphthalen-2-ol NA 912000000 NA NA NA NA BindingDB
PTPN1 4'-[5-Methyl-2-(4-trifluoromethyl-phenyl)-oxazol-4-yl]-biphenyl-4-ol NA 12500000|12589254.12 NA NA NA NA BindingDB|TTD
PTPN1 1-Bromo-6-[(2-butyl-benzofuran-3-yl)-hydroxy-methyl]-naphthalen-2-ol NA 478000000 NA NA NA NA BindingDB
PTPN1 {4'-[(2-Butyl-benzofuran-3-yl)-hydroxy-methyl]-biphenyl-4-yloxy}-acetic acid NA 537000000 NA NA NA NA BindingDB
PTPN1 (2R)-2-[4-[4-[2-[(2,4-dimethoxyphenyl)methyl]-1-benzothiophen-3-yl]phenyl]phenoxy]-3-phenylpropanoic acid NA 85100000 NA NA NA NA BindingDB
PTPN1 (2S)-2-[4-[4-(2-benzyl-1-benzofuran-3-yl)phenyl]-2-bromophenoxy]-3-phenylpropanoic acid NA 56200000 NA NA NA NA BindingDB
PTPN1 4-[4'-(2-Benzyl-benzofuran-3-yl)-3,5-dimethyl-biphenyl-4-yloxysulfonyl]-2-hydroxy-benzoic acid NA 38900000 NA NA NA NA BindingDB
PTPN1 2-[1-Bromo-6-[5-methyl-2-[4-(trifluoromethyl)phenyl]-1,3-oxazol-4-yl]naphthalen-2-yl]oxy-3-phenylpropanoic acid NA 190000000|190546071.8 NA NA NA NA BindingDB|TTD
PTPN1 4-[4'-(2-Benzyl-benzofuran-3-yl)-3-nitro-biphenyl-4-yloxysulfonyl]-2-hydroxy-benzoic acid NA 39800000 NA NA NA NA BindingDB
PTPN1 Benzothiophene derivative NA 28100000 NA NA NA NA BindingDB
PTPN1 4-[4''-(2-Benzyl-benzofuran-3-yl)-3-cyclopentyl-biphenyl-4-yloxysulfonyl]-2-hydroxy-benzoic acid NA 28100000 NA NA NA NA BindingDB
PTPN1 1-Bromo-6-(2-butyl-benzofuran-3-ylmethyl)-naphthalen-2-ol NA 331000000 NA NA NA NA BindingDB
PTPN1 2-[4'-(2-Benzyl-benzofuran-3-yl)-biphenyl-4-yloxy]-3-phenyl-propionic acid NA 275000000 NA NA NA NA BindingDB
PTPN1 (2S)-2-[4'-(2-Benzyl-benzofuran-3-yl)-biphenyl-4-yloxy]-3-phenyl-propionic acid NA 323000000 NA NA NA NA BindingDB
PTPN1 Subelliptenone G NA 148300 NA NA NA NA BindingDB|TTD
PTPN1 4-[4'-(2-Benzyl-benzo[b]thiophen-3-yl)-3-bromo-biphenyl-4-yloxysulfonyl]-2-hydroxy-benzoic acid NA 23900000 NA NA NA NA BindingDB
PTPN1 6-(2-Butyl-benzofuran-3-ylmethyl)-naphthalen-2-ol NA 676000000 NA NA NA NA BindingDB