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Drugs And Genes
Negative Drug Target Genes
GENE_SYMBOL DRUG_NAME Ki (nM) IC50 (nM) Kd (nM) EC50 (nM) Potency (nM) AC50 (nM) Datasource
PTPN6 sodium;(2R)-2-[[[ethoxy(hydroxy)phosphoryl]-(2-hydroxyphenyl)methyl]amino]-3-sulfanylpropanoate NA 10000000 NA NA NA NA TTD
PTPN6 sodium;(2S)-2-[[[ethoxy(hydroxy)phosphoryl]-(2-hydroxyphenyl)methyl]amino]-3-(1H-imidazol-5-yl)propanoate NA 167000 NA NA NA NA TTD
PTPN6 sodium;(2S)-2-[[[ethoxy(hydroxy)phosphoryl]-(2-hydroxyphenyl)methyl]amino]-3-phenylpropanoate NA 10000000 NA NA NA NA TTD
PTPN6 sodium;(2S)-2-[[[ethoxy(hydroxy)phosphoryl]-(2-hydroxyphenyl)methyl]amino]-3-(4-hydroxyphenyl)propanoate NA 10000000 NA NA NA NA TTD
PTPN6 2-[(S)-(2-chloroanilino)-diethoxyphosphorylmethyl]phenol NA 10000000 NA NA NA NA TTD
PTPN6 [(S)-(4-hydroxyanilino)-(2-hydroxyphenyl)methyl]phosphonic acid NA 10000000 NA NA NA NA TTD
PTPN6 2-[(S)-(4-bromoanilino)-diethoxyphosphorylmethyl]phenol NA 10000000 NA NA NA NA TTD
PTPN6 2-[(S)-diethoxyphosphoryl-(4-nitroanilino)methyl]phenol NA 10000000 NA NA NA NA TTD
PTPN6 sodium;(2S)-2-[[[ethoxy(hydroxy)phosphoryl]-(2-hydroxyphenyl)methyl]amino]-3-(1H-indol-3-yl)propanoate NA 10000000 NA NA NA NA TTD
PTPN6 2-[(S)-(4-chloroanilino)-diethoxyphosphorylmethyl]phenol NA 10000000 NA NA NA NA TTD
PTPN6 Vanadate(3-) NA 138000 NA NA NA NA BindingDB
PTPN6 Estradiol Phosphate NA 300000 NA NA NA NA TTD
PTPN6 H-Leu-Val-hPhe-Tyr(PO3H2)-Asn-Leu-Gly-Glu-OH NA NA NA 140000 NA NA TTD
PTPN6 (2S)-2-[[[ethoxy(hydroxy)phosphoryl]-(2-hydroxyphenyl)methyl]amino]-3-hydroxypropanoate NA 129000 NA NA NA NA BindingDB
PTPN6 (2S)-2-[[[ethoxy(hydroxy)phosphoryl]-(2-hydroxyphenyl)methyl]amino]-3-(1H-imidazol-5-yl)propanoate NA 167000 NA NA NA NA BindingDB
PTPN7 Enoxolone NA 300000 NA NA NA NA PubChem
PTPN7 (E)-2,2,6,6-tetramethyl-4-(3-(5-(3-nitrophenyl)furan-2-yl)acrylamido)piperidin-1-olate NA 211000 NA NA NA NA BindingDB
PTPN7 Estramustine Phosphate NA 152700 NA NA NA NA BindingDB|PubChem
PTPN7 (6R,7R)-3-[(4-carbamoylpyridin-1-ium-1-yl)methyl]-8-oxo-7-[(2-phenyl-2-sulfoacetyl)amino]-5-thia-1-azabicyclo[4.2.0]oct-2-ene-2-carboxylic acid NA 250000 NA NA NA NA BindingDB
PTPN7 Cefsulodin NA 250000 NA NA NA NA PubChem