| GENE_SYMBOL |
DRUG_NAME |
Ki (nM) |
IC50 (nM) |
Kd (nM) |
EC50 (nM) |
Potency (nM) |
AC50 (nM) |
Datasource |
| PTPN9 |
Cefsulodin |
NA |
350000 |
NA |
NA |
NA |
NA |
PubChem |
| PTPRA |
5-(3-Butyramidophenyl)isoxazole-3-carboxylic acid |
634000 |
NA |
NA |
NA |
NA |
NA |
ChEMBL |
| PTPRA |
2-(Oxalyl-Amino)-Benzoic Acid |
870000 |
NA |
NA |
NA |
NA |
NA |
PubChem |
| PTPRA |
Cefsulodin |
NA |
200000 |
NA |
NA |
NA |
NA |
PubChem |
| PTPRB |
3-(Carboxyformamido)thiophene-2-carboxylic acid |
160000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| PTPRB |
2-(Oxalyl-Amino)-4,5,6,7-Tetrahydro-Thieno[2,3-C]Pyridine-3-Carboxylic Acid |
560000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| PTPRB |
((4-(4-(4-(Difluoro-Phosphono-Methyl)-Phenyl)-Butyl)-Phenyl)-Difluoro-Methyl)-Phosphonic Acid |
NA |
342000 |
NA |
NA |
NA |
NA |
TTD |
| PTPRB |
Azane;[[4-[2-[[4-[difluoro(phosphono)methyl]phenyl]methoxy]ethoxymethyl]phenyl]-difluoromethyl]phosphonic acid |
NA |
300000 |
NA |
NA |
NA |
NA |
TTD |
| PTPRB |
10,13-dimethyl-17-[2-(6-sulfanylidene-3H-purin-9-yl)acetyl]-1,2,6,7,8,9,11,12,14,15,16,17-dodecahydrocyclopenta[a]phenanthren-3-one |
NA |
135000 |
NA |
NA |
NA |
NA |
TTD |
| PTPRB |
Sdccgsbi-0050247.P002 |
NA |
200000 |
NA |
NA |
NA |
NA |
TTD |
| PTPRB |
Cefsulodin |
NA |
200000 |
NA |
NA |
NA |
NA |
PubChem |
| PTPRB |
(1-Amino-2-phenylethyl)phosphonic acid |
NA |
139000 |
NA |
NA |
NA |
NA |
TTD |
| PTPRC |
Oxalyl-aryl-amino benzoic acid-based inhibitor 19 |
300000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| PTPRC |
2-[{4-[(2S)-2-{[(Allyloxy)carbonyl]amino}-3-({4-[3-hydroxy-2-(methoxycarbonyl)phenoxy]butyl}amino)-3-oxopropyl]phenyl}(carboxycarbonyl)amino]benzoic acid |
200000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| PTPRC |
Difluoro(1-naphthyl)methylphosphonic acid |
NA |
1000000 |
NA |
NA |
NA |
NA |
TTD |
| PTPRC |
Phosphonic acid, (difluoro-2-naphthalenylmethyl)- |
NA |
1000000 |
NA |
NA |
NA |
NA |
TTD |
| PTPRC |
[(4-{3-[4-(Difluoro-phosphono-methyl)-benzyloxy]-phenoxymethyl}-phenyl)-difluoro-methyl]-phosphonic acid |
NA |
108000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| PTPRC |
Benzo[b]thieno[2,3-d]thiophene-2-carboxylic acid, 3-(carboxymethoxy)- |
1250000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| PTPRC |
3-(1,1,1,3,3,3-Hexafluoro-2-hydroxypropan-2-yl)naphthalen-2-ol |
NA |
112400 |
NA |
NA |
NA |
NA |
TTD |
| PTPRC |
2-(1,1,1,3,3,3-Hexafluoro-2-hydroxypropan-2-yl)-5-phenylphenol |
NA |
500000 |
NA |
NA |
NA |
NA |
TTD |