| GENE_SYMBOL |
DRUG_NAME |
Ki (nM) |
IC50 (nM) |
Kd (nM) |
EC50 (nM) |
Potency (nM) |
AC50 (nM) |
Datasource |
| PTPRC |
2-(1,1,1,3,3,3-Hexafluoro-2-hydroxypropan-2-yl)-4-phenylphenol |
NA |
500000 |
NA |
NA |
NA |
NA |
TTD |
| PTPRC |
2-(1,1,1,3,3,3-Hexafluoro-2-hydroxypropan-2-yl)-6-phenylphenol |
NA |
157200 |
NA |
NA |
NA |
NA |
TTD |
| PTPRC |
2-(1,1,1,3,3,3-Hexafluoro-2-hydroxypropan-2-yl)-4-methylphenol |
NA |
207100 |
NA |
NA |
NA |
NA |
TTD |
| PTPRC |
4-(5-((3-Carboxy-4-hydroxyphenyl)amino)-5-oxopentanamido)-2,2,6,6-tetramethylpiperidin-1-olate |
NA |
1000000 |
NA |
NA |
NA |
NA |
TTD |
| PTPRC |
2-Hydroxy-5-(5-(((1-hydroxy-2,2,6,6-tetramethylpiperidin-4-yl)amino)methyl)furan-2-yl)benzoic acid |
NA |
1000000 |
NA |
NA |
NA |
NA |
TTD |
| PTPRC |
(E)-2,2,6,6-tetramethyl-4-(3-(5-(3-nitrophenyl)furan-2-yl)acrylamido)piperidin-1-olate |
NA |
1000000 |
NA |
NA |
NA |
NA |
TTD |
| PTPRC |
4-(5-((4-Hydroxy-3-(methoxycarbonyl)phenyl)amino)-5-oxopentanamido)-2,2,6,6-tetramethylpiperidin-1-olate |
NA |
1000000 |
NA |
NA |
NA |
NA |
TTD |
| PTPRC |
(E)-2,2,6,6-tetramethyl-4-(3-(5-(4-nitrophenyl)furan-2-yl)acrylamido)piperidin-1-olate |
NA |
1000000 |
NA |
NA |
NA |
NA |
TTD |
| PTPRC |
Methyl 2-hydroxy-5-(5-(((1-hydroxy-2,2,6,6-tetramethylpiperidin-4-yl)amino)methyl)furan-2-yl)benzoate |
NA |
1000000 |
NA |
NA |
NA |
NA |
TTD |
| PTPRC |
Pyrrospirone P |
NA |
190000 |
NA |
NA |
NA |
NA |
BindingDB |
| PTPRC |
4-Bromo-3-(Carboxymethoxy)-5-{3-[(3,3,5,5-Tetramethylcyclohexyl)amino]phenyl}thiophene-2-Carboxylic Acid |
151000 |
NA |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| PTPRC |
[7-(Phosphonomethyl)naphthalen-2-yl]methylphosphonic acid |
NA |
500000 |
NA |
NA |
NA |
NA |
TTD |
| PTPRC |
6-hydroxy-3-(1-(4-(naphthalen-1-ylamino)-4-oxobutyl)-1H-1,2,3-triazol-4-yl)-2-phenylbenzofuran-5-carboxylic acid |
NA |
186000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| PTPRC |
3-[(4-Chlorobenzyl)sulfanyl]-2-thiophenecarboxylic acid |
NA |
120000 |
NA |
NA |
NA |
NA |
TTD |
| PTPRC |
2-(2-Hydroxy-1,1,1,3,3,3-hexafluoropropyl)-1-naphthol |
NA |
500000 |
NA |
NA |
NA |
NA |
TTD |
| PTPRC |
4-Hydroxyphenylglyoxylic acid |
NA |
200000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| PTPRC |
5-Isopropoxy-2-(4-methylsulfanyl-pyridin-2-ylmethylsulfanyl)-1H-benzoimidazole |
NA |
1000000 |
NA |
NA |
NA |
NA |
TTD |
| PTPRC |
5-Isopropoxy-2-(pyridin-2-ylmethanesulfinyl)-1H-benzoimidazole |
NA |
120000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| PTPRC |
5-Isopropoxy-2-(4-methyl-pyridin-2-ylmethanesulfinyl)-1H-benzoimidazole |
NA |
380000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| PTPRC |
[7-(Phosphonatomethyl)-2-naphthyl]methylphosphonate |
NA |
500000 |
NA |
NA |
NA |
NA |
BindingDB |