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Drugs And Genes
Negative Drug Target Genes
GENE_SYMBOL DRUG_NAME Ki (nM) IC50 (nM) Kd (nM) EC50 (nM) Potency (nM) AC50 (nM) Datasource
PTPRC [[3-(3-Cyclohexyl-2-oxidanyl-phenyl)phenyl]-bis(fluoranyl)methyl]phosphonic acid 500000 NA NA NA NA NA TTD
PTPRC [4-[3-[(S)-(3,4-dichlorophenyl)-hydroxymethyl]phenyl]benzoyl]-trihydroxyphosphanium 270000 NA NA NA NA NA BindingDB
PTPRC [4-[3-[(R)-(3,4-dichlorophenyl)-hydroxymethyl]phenyl]benzoyl]-trihydroxyphosphanium 340000 NA NA NA NA NA BindingDB
PTPRC Ammonium; [7-(difluoro-phosphono-methyl)-naphthalen-2-yl]-difluoro-methanephosphonate NA 180000 NA NA NA NA BindingDB
PTPRC tetra ammonium [(4-{2-[4-(Difluoro-phosphono-methyl)-benzyloxy]-ethoxymethyl}-phenyl)-difluoro-methyl]-phosphonic acid NA 236000 NA NA NA NA BindingDB
PTPRC ammonium N-[4-(2-{[(benzyloxy)carbonyl]amino}-3-ethoxy-2-(methoxycarbonyl)-3-oxopropyl)phenyl]sulfamate NA 280000 NA NA NA NA BindingDB
PTPRC ammonium N-{4-[4-ethoxy-2,2-bis(methoxycarbonyl)-4-oxobutyl]phenyl}sulfamate NA 126000 NA NA NA NA BindingDB
PTPRC 4-Bromo-3-(carboxymethoxy)-5-phenylthiophene-2-carboxylic acid 280000 NA NA NA NA NA BindingDB
PTPRC 2-(Oxalyl-amino)-6-phenethyl-4,5,6,7-tetrahydro-thieno[2,3-c]pyridine-3-carboxylic acid 1400000 NA NA NA NA NA BindingDB|TTD
PTPRCAP Liriodenine NA 182000 NA NA NA NA BindingDB
PTPRCAP 7-Thiophosphonomethyl-naphthalene-1-carboxylic acid 200000 NA NA NA NA NA BindingDB
PTPRCAP 6-Phosphonohexanoic acid 42000000 NA NA NA NA NA BindingDB
PTPRCAP Phenylsulfanylmethyl-phosphonothioic acid 15800000 NA NA NA NA NA BindingDB
PTPRCAP 6-Thiophosphono-hexanoic acid 29000000 NA NA NA NA NA BindingDB
PTPRCAP Methylphosphonic acid 30000000 NA NA NA NA NA BindingDB|PubChem
PTPRCAP Methylphosphonothiolate 7000000 NA NA NA NA NA BindingDB
PTPRCAP (R)-Roemerine NA 107000 NA NA NA NA BindingDB
PTPRE Celastrol NA 500000 NA NA NA NA PubChem
PTPRE 2-(Oxalyl-Amino)-Benzoic Acid 130000 NA NA NA NA NA PubChem
PTPRE Cefsulodin NA 200000 NA NA NA NA PubChem