| GENE_SYMBOL |
DRUG_NAME |
Ki (nM) |
IC50 (nM) |
Kd (nM) |
EC50 (nM) |
Potency (nM) |
AC50 (nM) |
Datasource |
| PTPRF |
3-(Carboxyformamido)thiophene-2-carboxylic acid |
2000000 |
NA |
NA |
NA |
NA |
NA |
BindingDB |
| PTPRF |
6-(Oxalyl-Amino)-1h-Indole-5-Carboxylic Acid |
450000|550000 |
NA |
NA |
NA |
NA |
NA |
BindingDB |
| PTPRF |
2-(Oxalyl-Amino)-Benzoic Acid |
2000000 |
NA |
NA |
NA |
NA |
NA |
BindingDB|PubChem |
| PTPRF |
2-(Oxalyl-Amino)-4,7-Dihydro-5h-Thieno[2,3-C]Pyran-3-Carboxylic Acid |
360000 |
NA |
NA |
NA |
NA |
NA |
BindingDB |
| PTPRF |
2-[4-[3,5-Bis(trifluoromethyl)phenyl]-2-hydroxy-6-[[3-(trifluoromethyl)phenyl]methoxy]phenoxy]acetic acid |
NA |
116000 |
NA |
NA |
NA |
NA |
BindingDB |
| PTPRF |
7-(1,1-Dioxo-1h-Benzo(D)Isothiazol-3-Yloxymethyl)-2-(Oxalyl-Amino)-4,7-Dihydro-5h-Thieno(2,3-C)Pyran-3-Carboxylic Acid |
176000 |
NA |
NA |
NA |
NA |
NA |
BindingDB |
| PTPRF |
2-[(Carboxycarbonyl)amino]-4,5,6,7-tetrahydro-1-benzothiophene-3-carboxylic acid |
410000 |
NA |
NA |
NA |
NA |
NA |
BindingDB |
| PTPRF |
|
NA |
150930 |
NA |
NA |
NA |
NA |
BindingDB |
| PTPRF |
Vanadate(3-) |
NA |
141000 |
NA |
NA |
NA |
NA |
BindingDB |
| PTPRF |
Cefsulodin |
NA |
200000 |
NA |
NA |
NA |
NA |
PubChem |
| PTPRF |
(2S)-2-amino-N-[(2R)-1-[[2-(2,3-dihydro-1H-inden-1-ylamino)-2-oxoethyl]amino]-1-oxopropan-2-yl]-3-(4-hydroxyphenyl)propanamide |
NA |
111600 |
NA |
NA |
NA |
NA |
BindingDB |
| PTPRF |
[4-[3-[(S)-(3,4-dichlorophenyl)-hydroxymethyl]phenyl]benzoyl]-trihydroxyphosphanium |
390000 |
NA |
NA |
NA |
NA |
NA |
BindingDB |
| PTPRF |
[4-[3-[(R)-(3,4-dichlorophenyl)-hydroxymethyl]phenyl]benzoyl]-trihydroxyphosphanium |
360000 |
NA |
NA |
NA |
NA |
NA |
BindingDB |
| PTPRF |
ammonium N-[4-(2-{[(benzyloxy)carbonyl]amino}-3-ethoxy-2-(methoxycarbonyl)-3-oxopropyl)phenyl]sulfamate |
NA |
227000|472000 |
NA |
NA |
NA |
NA |
BindingDB |
| PTPRF |
ammonium N-{4-[4-ethoxy-2,2-bis(methoxycarbonyl)-4-oxobutyl]phenyl}sulfamate |
NA |
288000 |
NA |
NA |
NA |
NA |
BindingDB |
| PTPRF |
ammonium N-{4-[3-methoxy-2-(methoxycarbonyl)-3-oxo-2-(3-phenylpropyl)propyl]phenyl}sulfamate |
NA |
409000 |
NA |
NA |
NA |
NA |
BindingDB |
| PTPRF |
4-(Carboxyformamido)biphenyl-3-carboxylic acid |
700000 |
NA |
NA |
NA |
NA |
NA |
BindingDB |
| PTPRF |
3-(Carboxyformamido)-5-(4-fluorophenyl)thiophene-2-carboxylic acid |
110000 |
NA |
NA |
NA |
NA |
NA |
BindingDB |
| PTPRF |
2-(Oxalyl-amino)-6-phenethyl-4,5,6,7-tetrahydro-thieno[2,3-c]pyridine-3-carboxylic acid |
2100000 |
NA |
NA |
NA |
NA |
NA |
BindingDB |
| PTPRF |
3-(Carboxyformamido)-5-(3-nitrophenyl)thiophene-2-carboxylic acid |
165000 |
NA |
NA |
NA |
NA |
NA |
BindingDB |