| GENE_SYMBOL |
DRUG_NAME |
Ki (nM) |
IC50 (nM) |
Kd (nM) |
EC50 (nM) |
Potency (nM) |
AC50 (nM) |
Datasource |
| PYGB |
(2S,3R,4S,5S,6R)-3,4,5-trihydroxy-6-(hydroxymethyl)oxane-2-carbohydrazide |
3160000 |
NA |
NA |
NA |
NA |
NA |
BindingDB |
| PYGB |
3,4,5-Trihydroxy-6-hydroxymethyl-tetrahydro-pyran-2-carboxylic acid hydrazide |
398000|400000 |
NA |
NA |
NA |
NA |
NA |
BindingDB |
| PYGB |
(2S,3R,4S,5S,6R)-N-[(2,4-difluorophenyl)methyl]-3,4,5-trihydroxy-6-(hydroxymethyl)oxane-2-carboxamide |
25100000 |
NA |
NA |
NA |
NA |
NA |
BindingDB |
| PYGB |
N-(phenylcarbonyl)-beta-D-glucopyranosylamine |
144000 |
NA |
NA |
NA |
NA |
NA |
BindingDB |
| PYGB |
(2S,3R,4R,5S,6R)-2-(aminomethyl)-6-(hydroxymethyl)oxane-3,4,5-triol |
15800000 |
NA |
NA |
NA |
NA |
NA |
BindingDB |
| PYGB |
2-[(2R,3R,4S,5S,6R)-3,4,5-trihydroxy-6-(hydroxymethyl)oxan-2-yl]sulfanylacetamide |
19900000 |
NA |
NA |
NA |
NA |
NA |
BindingDB |
| PYGB |
N-(2,4-difluorophenyl)-2-[(2R,3R,4S,5S,6R)-3,4,5-trihydroxy-6-(hydroxymethyl)oxan-2-yl]sulfanylacetamide |
19900000 |
NA |
NA |
NA |
NA |
NA |
BindingDB |
| PYGB |
N-phenyl-2-[(2R,3R,4S,5S,6R)-3,4,5-trihydroxy-6-(hydroxymethyl)oxan-2-yl]sulfanylacetamide |
3980000 |
NA |
NA |
NA |
NA |
NA |
BindingDB |
| PYGB |
D-glycero-D-ido-Heptonic acid, 2,6-anhydro-, 2-methylhydrazide |
1990000 |
NA |
NA |
NA |
NA |
NA |
BindingDB |
| PYGB |
benzyl N-[(2S,3R,4S,5S,6R)-3,4,5-trihydroxy-6-(hydroxymethyl)oxan-2-yl]carbamate |
316000 |
NA |
NA |
NA |
NA |
NA |
BindingDB |
| PYGB |
2-acetamido-N-[(2S,3R,4S,5S,6R)-3,4,5-trihydroxy-6-(hydroxymethyl)oxan-2-yl]acetamide |
999000 |
NA |
NA |
NA |
NA |
NA |
BindingDB |
| PYGB |
N-[(5S,7S,8S,9S,10S)-8,9,10-trihydroxy-7-(hydroxymethyl)-2,4-dioxo-6-oxa-1,3-diazaspiro[4.5]decan-3-yl]acetamide |
501000 |
NA |
NA |
NA |
NA |
NA |
BindingDB |
| PYGB |
alpha-Isomaltose |
15800000 |
NA |
NA |
NA |
NA |
NA |
BindingDB |
| PYGB |
(R)-2-Hydroxymethyl-6-methoxy-tetrahydro-pyran-3,4,5-triol |
24700000 |
NA |
NA |
NA |
NA |
NA |
BindingDB |
| PYGB |
3,4,5-Trihydroxy-6-hydroxymethyl-tetrahydro-pyran-2-carboxylic acid methyl ester |
2800000 |
NA |
NA |
NA |
NA |
NA |
BindingDB |
| PYGB |
methyl (2S,3R,4S,5S,6R)-3,4,5-trihydroxy-6-(hydroxymethyl)oxane-2-carboxylate |
25100000 |
NA |
NA |
NA |
NA |
NA |
BindingDB |
| PYGB |
2-Aminomethyl-6-hydroxymethyl-tetrahydro-pyran-3,4,5-triol |
16800000 |
NA |
NA |
NA |
NA |
NA |
BindingDB |
| PYGB |
3,4,5-Trihydroxy-6-hydroxymethyl-tetrahydro-pyran-2-carboxylic acid phenylamide |
5400000 |
NA |
NA |
NA |
NA |
NA |
BindingDB |
| PYGB |
(3,4,5-Trihydroxy-6-hydroxymethyl-tetrahydro-pyran-2-yl)-carbamic acid benzyl ester |
350000 |
NA |
NA |
NA |
NA |
NA |
BindingDB |
| PYGB |
2-Hydroxymethyl-6-mercapto-tetrahydro-pyran-3,4,5-triol |
1000000 |
NA |
NA |
NA |
NA |
NA |
BindingDB |