| GENE_SYMBOL |
DRUG_NAME |
Ki (nM) |
IC50 (nM) |
Kd (nM) |
EC50 (nM) |
Potency (nM) |
AC50 (nM) |
Datasource |
| PYGB |
((R)-3,4,5-Trihydroxy-6-hydroxymethyl-tetrahydro-pyran-2-yl)-carbamic acid benzyl ester |
350000 |
NA |
NA |
NA |
NA |
NA |
BindingDB |
| PYGB |
2-((S)-3,4,5-Trihydroxy-6-hydroxymethyl-tetrahydro-pyran-2-yl)-ethyl-ammonium |
4500000 |
NA |
NA |
NA |
NA |
NA |
BindingDB |
| PYGB |
((S)-3,4,5-Trihydroxy-6-hydroxymethyl-tetrahydro-pyran-2-yl)-acetonitrile |
9000000 |
NA |
NA |
NA |
NA |
NA |
BindingDB |
| PYGB |
(2R)-3,4,5-trihydroxy-6-(hydroxymethyl)-N-(4-hydroxyphenyl)oxane-2-carboxamide |
4400000 |
NA |
NA |
NA |
NA |
NA |
BindingDB |
| PYGB |
(S)-2,6-Bis-hydroxymethyl-tetrahydro-pyran-2,3,4,5-tetraol |
15800000 |
NA |
NA |
NA |
NA |
NA |
BindingDB |
| PYGB |
(S)-3,4,5-Trihydroxy-6-hydroxymethyl-tetrahydro-pyran-2-carboxylic acid methylamide |
36700000 |
NA |
NA |
NA |
NA |
NA |
BindingDB |
| PYGB |
(R)-3,4,5-Trihydroxy-6-hydroxymethyl-tetrahydro-pyran-2-ylmethyl-ammonium |
34500000 |
NA |
NA |
NA |
NA |
NA |
BindingDB |
| PYGB |
((S)-2,3,4,5-Tetrahydroxy-6-hydroxymethyl-tetrahydro-pyran-2-yl)-acetonitrile |
7600000 |
NA |
NA |
NA |
NA |
NA |
BindingDB |
| PYGB |
(S)-2-Azidomethyl-6-hydroxymethyl-tetrahydro-pyran-2,3,4,5-tetraol |
7400000 |
NA |
NA |
NA |
NA |
NA |
BindingDB |
| PYGB |
(2S)-3,4,5-trihydroxy-N-(2-hydroxyethyl)-6-(hydroxymethyl)oxane-2-carboxamide |
16900000 |
NA |
NA |
NA |
NA |
NA |
BindingDB |
| PYGB |
(S)-3,4,5-Trihydroxy-6-hydroxymethyl-tetrahydro-pyran-2-ylmethyl-ammonium |
16800000 |
NA |
NA |
NA |
NA |
NA |
BindingDB |
| PYGB |
(S)-3,4,5-Trihydroxy-6-hydroxymethyl-tetrahydro-pyran-2-carboxylic acid anion |
15200000 |
NA |
NA |
NA |
NA |
NA |
BindingDB |
| PYGB |
(S)-3,4,5-Trihydroxy-6-hydroxymethyl-tetrahydro-pyran-2-carboxylic acid methyl ester |
24200000 |
NA |
NA |
NA |
NA |
NA |
BindingDB |
| PYGB |
(R)-2-Azidomethyl-6-hydroxymethyl-tetrahydro-pyran-3,4,5-triol |
22400000 |
NA |
NA |
NA |
NA |
NA |
BindingDB |
| PYGB |
(S)-2-Hydroxymethyl-6-mercapto-tetrahydro-pyran-3,4,5-triol |
1000000 |
NA |
NA |
NA |
NA |
NA |
BindingDB |
| PYGB |
(2S)-3,4,5-trihydroxy-6-(hydroxymethyl)-N-(4-hydroxyphenyl)oxane-2-carboxamide |
5600000 |
NA |
NA |
NA |
NA |
NA |
BindingDB |
| PYGB |
(R)-3,4,5-Trihydroxy-6-hydroxymethyl-tetrahydro-pyran-2-carboxylic acid phenylamide |
5400000 |
NA |
NA |
NA |
NA |
NA |
BindingDB |
| PYGB |
(R)-2,6-Bis-hydroxymethyl-tetrahydro-pyran-3,4,5-triol |
1500000 |
NA |
NA |
NA |
NA |
NA |
BindingDB |
| PYGB |
(S)-3,4,5-Trihydroxy-6-hydroxymethyl-tetrahydro-pyran-2-carboxylic acid 2,4-difluoro-benzylamide |
27200000 |
NA |
NA |
NA |
NA |
NA |
BindingDB |
| PYGB |
(2R)-3,4,5-trihydroxy-6-(hydroxymethyl)-N-(2,2,2-trifluoroethyl)oxane-2-carboxamide |
8100000 |
NA |
NA |
NA |
NA |
NA |
BindingDB |