| GENE_SYMBOL |
DRUG_NAME |
Ki (nM) |
IC50 (nM) |
Kd (nM) |
EC50 (nM) |
Potency (nM) |
AC50 (nM) |
Datasource |
| PYGB |
(2R,3R,4S,5S,6R)-3,4,5-trihydroxy-6-(hydroxymethyl)-N'-methyloxane-2-carbohydrazide |
1800000 |
NA |
NA |
NA |
NA |
NA |
BindingDB |
| PYGB |
(2R)-N-[(2R)-1-[(2-amino-2-oxoethyl)amino]-1-oxopropan-2-yl]-2-(dioxiran-3-yl)-3-phenylpropanamide |
398000 |
NA |
NA |
NA |
NA |
NA |
BindingDB |
| PYGB |
(2R,3R,4S,5S,6R)-3,4,5-trihydroxy-6-(hydroxymethyl)-N-(4-hydroxyphenyl)oxane-2-carboxamide |
3980000 |
NA |
NA |
NA |
NA |
NA |
BindingDB |
| PYGB |
(2R,3R,4S,5S,6R)-3,4,5-trihydroxy-N-(2-hydroxyethyl)-6-(hydroxymethyl)oxane-2-carboxamide |
2510000 |
NA |
NA |
NA |
NA |
NA |
BindingDB |
| PYGB |
2-Amino-N-beta-D-glucopyranosylacetamide |
398000 |
NA |
NA |
NA |
NA |
NA |
BindingDB |
| PYGB |
2-acetamido-N-[(2R,3R,4S,5S,6R)-3,4,5-trihydroxy-6-(hydroxymethyl)oxan-2-yl]acetamide |
990000 |
NA |
NA |
NA |
NA |
NA |
BindingDB |
| PYGB |
(2R,3R,4S,5S,6R)-3,4,5-trihydroxy-6-(hydroxymethyl)-N-methyloxane-2-carboxamide |
199000 |
NA |
NA |
NA |
NA |
NA |
BindingDB |
| PYGB |
methyl (2R,3R,4S,5S,6R)-3,4,5-trihydroxy-6-(hydroxymethyl)oxane-2-carboxylate |
2510000 |
NA |
NA |
NA |
NA |
NA |
BindingDB |
| PYGB |
(2S,3R,4S,5S,6R)-3,4,5-trihydroxy-6-(hydroxymethyl)-N-(4-hydroxyphenyl)oxane-2-carboxamide |
5010000 |
NA |
NA |
NA |
NA |
NA |
BindingDB |
| PYGB |
(2S,3R,4S,5S,6R)-3,4,5-trihydroxy-6-(hydroxymethyl)-N-methyloxane-2-carboxamide |
39800000 |
NA |
NA |
NA |
NA |
NA |
BindingDB |
| PYGB |
(2R,3R,4S,5S,6R)-3,4,5-trihydroxy-6-(hydroxymethyl)oxane-2-carboxamide |
398000 |
NA |
NA |
NA |
NA |
NA |
BindingDB |
| PYGB |
(2S,3R,4S,5S,6R)-3,4,5-trihydroxy-6-(hydroxymethyl)-N-phenyloxane-2-carboxamide |
12500000 |
NA |
NA |
NA |
NA |
NA |
BindingDB |
| PYGB |
(2R,3S,4S,5R,6R)-2-(hydroxymethyl)-6-(1H-indol-2-yloxy)oxane-3,4,5-triol |
2510000 |
NA |
NA |
NA |
NA |
NA |
BindingDB |
| PYGB |
2-[(2S,3R,4S,5S,6R)-2,3,4,5-tetrahydroxy-6-(hydroxymethyl)oxan-2-yl]acetonitrile |
7600000|7940000 |
NA |
NA |
NA |
NA |
NA |
BindingDB |
| PYGB |
(2S,3R,4R,5S,6R)-2-(2-aminoethyl)-6-(hydroxymethyl)oxane-3,4,5-triol |
5010000 |
NA |
NA |
NA |
NA |
NA |
BindingDB |
| PYGB |
(3,4,5-Trihydroxy-6-hydroxymethyl-tetrahydro-pyran-2-yl)-acetonitrile |
9000000|9990000 |
NA |
NA |
NA |
NA |
NA |
BindingDB |
| PYGB |
2,6-Anhydro-D-glycero-D-ido-heptonic acid |
15800000 |
NA |
NA |
NA |
NA |
NA |
BindingDB |
| PYGB |
(2R,3R,4S,5S,6R)-3,4,5-trihydroxy-6-(hydroxymethyl)-N-(3,3,3-trifluoropropyl)oxane-2-carboxamide |
7940000 |
NA |
NA |
NA |
NA |
NA |
BindingDB |
| PYGB |
(2R,3R,4R,5S,6R)-2-(aminomethyl)-6-(hydroxymethyl)oxane-3,4,5-triol |
31600000 |
NA |
NA |
NA |
NA |
NA |
BindingDB |
| PYGB |
(2S,3R,4S,5S,6R)-2,6-bis(hydroxymethyl)oxane-2,3,4,5-tetrol |
15800000 |
NA |
NA |
NA |
NA |
NA |
BindingDB |