| GENE_SYMBOL |
DRUG_NAME |
Ki (nM) |
IC50 (nM) |
Kd (nM) |
EC50 (nM) |
Potency (nM) |
AC50 (nM) |
Datasource |
| PYGB |
(2S,3R,4S,5S,6R)-3,4,5-trihydroxy-N-(2-hydroxyethyl)-6-(hydroxymethyl)oxane-2-carboxamide |
15800000 |
NA |
NA |
NA |
NA |
NA |
BindingDB |
| PYGB |
(2R,3R,4S,5S,6R)-3,4,5-trihydroxy-6-(hydroxymethyl)-N-phenyloxane-2-carboxamide |
5010000 |
NA |
NA |
NA |
NA |
NA |
BindingDB |
| PYGB |
(2R,3S,4S,5R,6S)-2-(hydroxymethyl)-6-(1H-indol-2-yloxy)oxane-3,4,5-triol |
2510000|2600000 |
NA |
NA |
NA |
NA |
NA |
BindingDB |
| PYGB |
(2R,3R,4S,5S,6R)-N-cyclopropyl-3,4,5-trihydroxy-6-(hydroxymethyl)oxane-2-carboxamide |
1250000 |
NA |
NA |
NA |
NA |
NA |
BindingDB |
| PYGB |
(2R,3R,4S,5S,6R)-3,4,5-trihydroxy-6-(hydroxymethyl)-N-(2,2,2-trifluoroethyl)oxane-2-carboxamide |
7940000 |
NA |
NA |
NA |
NA |
NA |
BindingDB |
| PYGB |
1-thio-beta-D-glucopyranose |
999000 |
NA |
NA |
NA |
NA |
NA |
BindingDB |
| PYGB |
Methyl beta-D-glucopyranoside |
25100000 |
NA |
NA |
NA |
NA |
NA |
BindingDB |
| PYGB |
Alpha-D-Glucopyranosyl-2-Carboxylic Acid Amide |
398000 |
NA |
NA |
NA |
NA |
NA |
BindingDB |
| PYGB |
3-Amino-8,9,10-trihydroxy-7-hydroxymethyl-6-oxa-1,3-diaza-spiro[4.5]decane-2,4-dione |
146000 |
NA |
NA |
NA |
NA |
NA |
BindingDB |
| PYGB |
3,4,5-Trihydroxy-6-hydroxymethyl-tetrahydro-pyran-2-carboxylic acid amide |
440000 |
NA |
NA |
NA |
NA |
NA |
BindingDB |
| PYGB |
2,6-Bis-hydroxymethyl-tetrahydro-pyran-3,4,5-triol |
1500000 |
NA |
NA |
NA |
NA |
NA |
BindingDB |
| PYGB |
5-Thio-alpha-D-glucopyranose |
1990000|2000000 |
NA |
NA |
NA |
NA |
NA |
BindingDB |
| PYGB |
D-Glucose |
1700000|7400000|7940000|7943280|1584890 |
NA |
NA |
NA |
NA |
NA |
BindingDB|PubChem |
| PYGB |
(S)-6-Hydroxymethyl-tetrahydro-pyran-2,3,4,5-tetraol |
1700000 |
NA |
NA |
NA |
NA |
NA |
BindingDB |
| PYGB |
Methyl alpha-D-glucopyranoside |
12500000 |
NA |
NA |
NA |
NA |
NA |
BindingDB |
| PYGB |
(2S,3S,4S,5S,6S)-2-(azidomethyl)-6-(hydroxymethyl)oxane-2,3,4,5-tetrol |
7400000 |
NA |
NA |
NA |
NA |
NA |
BindingDB |
| PYGB |
[(2S,3S,4S,5S,6S)-2,3,4,5-tetrahydroxy-6-(hydroxymethyl)oxan-2-yl]methyl methanesulfonate |
3700000 |
NA |
NA |
NA |
NA |
NA |
BindingDB |
| PYGB |
(2S,3S,4S,5S,6S)-2,6-bis(hydroxymethyl)oxane-2,3,4,5-tetrol |
15800000 |
NA |
NA |
NA |
NA |
NA |
BindingDB |
| PYGB |
(2S,3R,4S,5S,6R)-6-(3,4,5-Trihydroxy-6-hydroxymethyl-tetrahydro-pyran-2-yloxymethyl)-tetrahydro-pyran-2,3,4,5-tetraol |
16300000 |
NA |
NA |
NA |
NA |
NA |
BindingDB |
| PYGB |
[(2S,3R,4S,5S,6R)-3,4,5-trihydroxy-6-(hydroxymethyl)oxan-2-yl]urea |
125000 |
NA |
NA |
NA |
NA |
NA |
BindingDB |