| GENE_SYMBOL |
DRUG_NAME |
Ki (nM) |
IC50 (nM) |
Kd (nM) |
EC50 (nM) |
Potency (nM) |
AC50 (nM) |
Datasource |
| PYGM |
2-Amino-N-(3,4,5-trihydroxy-6-hydroxymethyl-tetrahydro-pyran-2-yl)-acetamide |
371535 |
NA |
NA |
NA |
NA |
NA |
BindingDB |
| PYGM |
2-(hydroxymethyl)-6-[3-[(3R,4S,5S,6R)-3,4,5-trihydroxy-6-(hydroxymethyl)oxan-2-yl]oxyindol-1-yl]oxane-3,4,5-triol |
2570396 |
NA |
NA |
NA |
NA |
NA |
BindingDB |
| PYGM |
3,4,5,6-tetrahydroxy-N-(4-hydroxyphenyl)oxane-2-carboxamide |
4365158 |
NA |
NA |
NA |
NA |
NA |
BindingDB |
| PYGM |
2-(hydroxymethyl)-6-[[(2R,3S,4S,6S)-3,4,6-trihydroxy-5-sulfanyloxan-2-yl]methoxy]oxane-3,4,5-triol |
1995262 |
NA |
NA |
NA |
NA |
NA |
BindingDB |
| PYGM |
2-[(2S,3R,4S,5S,6R)-3,4,5-trihydroxy-6-(hydroxymethyl)oxan-2-yl]sulfanylacetamide |
20892961 |
NA |
NA |
NA |
NA |
NA |
BindingDB |
| PYGM |
N-(2,4-difluorophenyl)-2-[(2S,3R,4S,5S,6R)-3,4,5-trihydroxy-6-(hydroxymethyl)oxan-2-yl]sulfanylacetamide |
19054607 |
NA |
NA |
NA |
NA |
NA |
BindingDB |
| PYGM |
(2R,3R,4R,5S,6R)-2-(azidomethyl)-6-(hydroxymethyl)oxane-3,4,5-triol |
1650000 |
NA |
NA |
NA |
NA |
NA |
BindingDB |
| PYGM |
(2S,3R,4R,5S,6R)-2-(azidomethyl)-6-(hydroxymethyl)oxane-3,4,5-triol |
1820000 |
NA |
NA |
NA |
NA |
NA |
BindingDB |
| PYGM |
N-phenyl-2-[(2S,3R,4S,5S,6R)-3,4,5-trihydroxy-6-(hydroxymethyl)oxan-2-yl]sulfanylacetamide |
3630781 |
NA |
NA |
NA |
NA |
NA |
BindingDB |
| PYGM |
(2R,3R,4S,5S,6R)-3,4,5-trihydroxy-6-(hydroxymethyl)-N'-methyloxane-2-carbohydrazide |
1778279 |
NA |
NA |
NA |
NA |
NA |
BindingDB |
| PYGM |
2-acetamido-N-[(2R,3R,4S,5S,6R)-3,4,5-trihydroxy-6-(hydroxymethyl)oxan-2-yl]acetamide |
1000000 |
NA |
NA |
NA |
NA |
NA |
BindingDB |
| PYGM |
2-[(2S,3R,4S,5S,6R)-2,3,4,5-tetrahydroxy-6-(hydroxymethyl)oxan-2-yl]acetonitrile |
2120000 |
NA |
NA |
NA |
NA |
NA |
BindingDB |
| PYGM |
(3,4,5-Trihydroxy-6-hydroxymethyl-tetrahydro-pyran-2-yl)-acetonitrile |
2040000 |
NA |
NA |
NA |
NA |
NA |
BindingDB |
| PYGM |
1-Deoxy-1-methoxycarbamido-beta-D-gluco-2-heptulopyranosonamide |
4800000 |
NA |
NA |
NA |
NA |
NA |
BindingDB |
| PYGM |
1-Deoxy-1-Methoxycarbamido-Beta-D-Glucopyranose |
4070000 |
NA |
NA |
NA |
NA |
NA |
BindingDB |
| PYGM |
3-Amino-8,9,10-trihydroxy-7-hydroxymethyl-6-oxa-1,3-diaza-spiro[4.5]decane-2,4-dione |
144544 |
NA |
NA |
NA |
NA |
NA |
BindingDB |
| PYGM |
N-[8,9,10-trihydroxy-7-(hydroxymethyl)-2,4-dioxo-6-oxa-1,3-diazaspiro[4.5]decan-3-yl]acetamide |
549541 |
NA |
NA |
NA |
NA |
NA |
BindingDB |
| PYGM |
3,4,5-Trihydroxy-6-hydroxymethyl-tetrahydro-pyran-2-carboxylic acid amide |
3360000 |
NA |
NA |
NA |
NA |
NA |
BindingDB |
| PYGM |
2,6-Bis-hydroxymethyl-tetrahydro-pyran-3,4,5-triol |
2820000 |
NA |
NA |
NA |
NA |
NA |
BindingDB |
| PYGM |
Gal(a1-6)Hex |
1790000 |
NA |
NA |
NA |
NA |
NA |
BindingDB |