| GENE_SYMBOL |
DRUG_NAME |
Ki (nM) |
IC50 (nM) |
Kd (nM) |
EC50 (nM) |
Potency (nM) |
AC50 (nM) |
Datasource |
| PYGM |
5-Ethynyl-1-(Beta-D-Glucopyranosyl)pyrimidine-2,4(1h,3h)-Dione |
NA |
291400 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| PYGM |
D-Glucose |
2770000 |
NA |
NA |
NA |
NA |
NA |
BindingDB |
| PYGM |
(2S,3S,4S,5S,6S)-2-(azidomethyl)-6-(hydroxymethyl)oxane-2,3,4,5-tetrol |
7413102 |
NA |
NA |
NA |
NA |
NA |
BindingDB |
| PYGM |
[(2S,3S,4S,5S,6S)-2,3,4,5-tetrahydroxy-6-(hydroxymethyl)oxan-2-yl]methyl methanesulfonate |
2430000 |
NA |
NA |
NA |
NA |
NA |
BindingDB |
| PYGM |
(2S,3S,4S,5S,6S)-2,6-bis(hydroxymethyl)oxane-2,3,4,5-tetrol |
1800000 |
NA |
NA |
NA |
NA |
NA |
BindingDB |
| PYGM |
alpha-D-Glucopyranose |
1700000 |
NA |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| QARS1 |
4-ammonio-5-{[(2R,6S)-6-(hydroxymethyl)piperidin-2-yl]methoxy}-5-oxopentanoate |
230000 |
NA |
NA |
NA |
NA |
NA |
BindingDB |
| QARS1 |
4-amino-5-oxo-5-[[(2R,3S,4R)-3,4,5-trihydroxyoxolan-2-yl]methoxy]pentanoic acid |
500000 |
NA |
NA |
NA |
NA |
NA |
BindingDB |
| QARS1 |
4-amino-5-oxo-5-[[(2R)-pyrrolidin-2-yl]methoxy]pentanoic acid |
380000 |
NA |
NA |
NA |
NA |
NA |
BindingDB |
| QARS1 |
4-amino-5-oxo-5-[[(2S)-pyrrolidin-2-yl]methoxy]pentanoic acid |
11400000 |
NA |
NA |
NA |
NA |
NA |
BindingDB |
| QPCT |
3-(3H-benzimidazol-5-yl)-2-sulfanylidene-4aH-quinazolin-4-one |
NA |
120800 |
NA |
NA |
NA |
NA |
BindingDB |
| QPCT |
1H-Imidazole-5-methanol, 4-methyl- |
129000 |
NA |
NA |
NA |
NA |
NA |
BindingDB |
| QPCT |
2-Thiohydantoin |
NA |
390000 |
NA |
NA |
NA |
NA |
BindingDB |
| QPCT |
4-Methylimidazole |
NA |
110000 |
NA |
NA |
NA |
NA |
BindingDB |
| QPCT |
2-Aminobenzimidazole |
1800000 |
NA |
NA |
NA |
NA |
NA |
BindingDB |
| QPCT |
5-Methyl-1-phenylimidazole |
NA |
144000 |
NA |
NA |
NA |
NA |
BindingDB |
| QPCT |
L-histidinol |
1530000 |
NA |
NA |
NA |
NA |
NA |
BindingDB |
| QPCT |
Dimethylarsinate |
1824000|6696000 |
NA |
NA |
NA |
NA |
NA |
BindingDB |
| QPCT |
N-Acetylimidazole |
107000 |
NA |
NA |
NA |
NA |
NA |
BindingDB |
| QPCT |
Oxyquinoline |
NA |
208000 |
NA |
NA |
NA |
NA |
BindingDB|PubChem |