| GENE_SYMBOL |
DRUG_NAME |
Ki (nM) |
IC50 (nM) |
Kd (nM) |
EC50 (nM) |
Potency (nM) |
AC50 (nM) |
Datasource |
| PYGL |
(2~{R},3~{S},4~{S},5~{R},6~{R})-2-(hydroxymethyl)-6-(5-phenyl-1,2,3,4-tetrazol-2-yl)oxane-3,4,5-triol |
134200 |
NA |
NA |
NA |
NA |
NA |
BindingDB |
| PYGL |
(2~{R},3~{S},4~{R},5~{R},6~{S})-2-(hydroxymethyl)-6-(2-phenyl-1,3-thiazol-4-yl)oxane-3,4,5-triol |
172200 |
NA |
NA |
NA |
NA |
NA |
BindingDB |
| PYGL |
|
179900 |
NA |
NA |
NA |
NA |
NA |
BindingDB |
| PYGL |
alpha-D-Glucopyranose |
4280000|4900000 |
NA |
NA |
NA |
NA |
NA |
BindingDB |
| PYGM |
3,4,5-Trihydroxy-6-hydroxymethyl-tetrahydro-pyran-2-carboxylic acid hydrazide |
2520000 |
NA |
NA |
NA |
NA |
NA |
BindingDB |
| PYGM |
4-[2-(3-Carboxy-benzoylamino)-phenoxy]-phthalic acid |
NA |
200000 |
NA |
NA |
NA |
NA |
TTD |
| PYGM |
3,4,5-Trihydroxy-6-hydroxymethyl-tetrahydro-pyran-2-carboxylic acid methyl ester |
2550000 |
NA |
NA |
NA |
NA |
NA |
BindingDB |
| PYGM |
2-Aminomethyl-6-hydroxymethyl-tetrahydro-pyran-3,4,5-triol |
1780000 |
NA |
NA |
NA |
NA |
NA |
BindingDB |
| PYGM |
Glc(a1-4)Glc(a1-4)Glc(a1-4)Glc(a1-4)Glc(a1-4)Glc(a1-4)Glc |
1000000 |
NA |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| PYGM |
3,4,5-Trihydroxy-6-hydroxymethyl-tetrahydro-pyran-2-carboxylic acid phenylamide |
2270000 |
NA |
NA |
NA |
NA |
NA |
BindingDB |
| PYGM |
(3,4,5-Trihydroxy-6-hydroxymethyl-tetrahydro-pyran-2-yl)-carbamic acid benzyl ester |
346737 |
NA |
NA |
NA |
NA |
NA |
BindingDB |
| PYGM |
2-Hydroxymethyl-6-mercapto-tetrahydro-pyran-3,4,5-triol |
3000000 |
NA |
NA |
NA |
NA |
NA |
BindingDB |
| PYGM |
Caffeine |
NA |
114000 |
NA |
NA |
NA |
NA |
BindingDB|PubChem|TTD |
| PYGM |
Glucosylurea |
141254 |
NA |
NA |
NA |
NA |
NA |
BindingDB |
| PYGM |
2-(2-Aminoethyl)-6-(hydroxymethyl)oxane-3,4,5-triol |
2350000 |
NA |
NA |
NA |
NA |
NA |
BindingDB |
| PYGM |
3,4,5-Trihydroxy-6-hydroxymethyl-tetrahydro-pyran-2-carboxylic acid cyclopropylamide |
1288250 |
NA |
NA |
NA |
NA |
NA |
BindingDB |
| PYGM |
3,4,5-Trihydroxy-6-hydroxymethyl-tetrahydro-pyran-2-carboxylic acid (2,2,2-trifluoro-ethyl)-amide |
8128305 |
NA |
NA |
NA |
NA |
NA |
BindingDB |
| PYGM |
Methanesulfonic acid 3,4,5-trihydroxy-6-hydroxymethyl-tetrahydro-pyran-2-ylmethyl ester |
2320000 |
NA |
NA |
NA |
NA |
NA |
BindingDB |
| PYGM |
3,4,5-Trihydroxy-6-hydroxymethyl-tetrahydro-pyran-2-carboxylic acid (2-hydroxy-ethyl)-amide |
2570396 |
NA |
NA |
NA |
NA |
NA |
BindingDB |
| PYGM |
3,4,5-Trihydroxy-6-hydroxymethyl-tetrahydro-pyran-2-carboxylic acid methylamide |
3800000 |
NA |
NA |
NA |
NA |
NA |
BindingDB |