| GENE_SYMBOL |
DRUG_NAME |
Ki (nM) |
IC50 (nM) |
Kd (nM) |
EC50 (nM) |
Potency (nM) |
AC50 (nM) |
Datasource |
| PYGB |
(S)-3,4,5-Trihydroxy-6-hydroxymethyl-tetrahydro-pyran-2-carboxylic acid phenylamide |
12600000 |
NA |
NA |
NA |
NA |
NA |
BindingDB |
| PYGB |
(S)-3,4,5-Trihydroxy-6-hydroxymethyl-tetrahydro-pyran-2-carboxylic acid hydrazide |
3000000 |
NA |
NA |
NA |
NA |
NA |
BindingDB |
| PYGB |
(R)-3,4,5-Trihydroxy-6-hydroxymethyl-tetrahydro-pyran-2-carboxylic acid methyl ester |
2800000 |
NA |
NA |
NA |
NA |
NA |
BindingDB |
| PYGB |
(2R)-3,4,5-trihydroxy-N-(2-hydroxyethyl)-6-(hydroxymethyl)oxane-2-carboxamide |
2600000 |
NA |
NA |
NA |
NA |
NA |
BindingDB |
| PYGB |
(S)-3,4,5-Trihydroxy-6-hydroxymethyl-tetrahydro-pyran-2-carboxylic acid amide |
370000 |
NA |
NA |
NA |
NA |
NA |
BindingDB |
| PYGB |
(R)-3,4,5-Trihydroxy-6-hydroxymethyl-tetrahydro-pyran-2-carboxylic acid hydrazide |
400000 |
NA |
NA |
NA |
NA |
NA |
BindingDB |
| PYGB |
((R)-3,4,5-Trihydroxy-6-hydroxymethyl-tetrahydro-pyran-2-ylcarbamoyl)-methyl-ammonium |
370000 |
NA |
NA |
NA |
NA |
NA |
BindingDB |
| PYGB |
(R)-3,4,5-Trihydroxy-6-hydroxymethyl-tetrahydro-pyran-2-carboxylic acid amide |
440000 |
NA |
NA |
NA |
NA |
NA |
BindingDB |
| PYGB |
2-(Hydroxymethyl)phenyl alpha-D-glucopyranoside |
7940000 |
NA |
NA |
NA |
NA |
NA |
BindingDB |
| PYGB |
[(2S,3R,4S,5S,6R)-2,3,4,5-tetrahydroxy-6-(hydroxymethyl)oxan-2-yl]methyl methanesulfonate |
3980000 |
NA |
NA |
NA |
NA |
NA |
BindingDB |
| PYGB |
(2S,3R,4S,5S,6R)-2-(azidomethyl)-6-(hydroxymethyl)oxane-2,3,4,5-tetrol |
7940000 |
NA |
NA |
NA |
NA |
NA |
BindingDB |
| PYGB |
2-[(2S,3R,4S,5S,6R)-3,4,5-trihydroxy-6-(hydroxymethyl)oxan-2-yl]sulfanylacetamide |
21100000 |
NA |
NA |
NA |
NA |
NA |
BindingDB |
| PYGB |
N-(2,4-difluorophenyl)-2-[(2S,3R,4S,5S,6R)-3,4,5-trihydroxy-6-(hydroxymethyl)oxan-2-yl]sulfanylacetamide |
18900000 |
NA |
NA |
NA |
NA |
NA |
BindingDB |
| PYGB |
(2R,3R,4R,5S,6R)-2-(azidomethyl)-6-(hydroxymethyl)oxane-3,4,5-triol |
22400000|25100000 |
NA |
NA |
NA |
NA |
NA |
BindingDB |
| PYGB |
(2S,3R,4R,5S,6R)-2-(azidomethyl)-6-(hydroxymethyl)oxane-3,4,5-triol |
15200000|15800000 |
NA |
NA |
NA |
NA |
NA |
BindingDB |
| PYGB |
(2R,3S,5R,6S)-2,6-bis(hydroxymethyl)oxane-3,4,5-triol |
19900000 |
NA |
NA |
NA |
NA |
NA |
BindingDB |
| PYGB |
(2R,3S,5R,6R)-2,6-bis(hydroxymethyl)oxane-3,4,5-triol |
1580000 |
NA |
NA |
NA |
NA |
NA |
BindingDB |
| PYGB |
Carba-alpha-d-glucopyranose |
50100000 |
NA |
NA |
NA |
NA |
NA |
BindingDB |
| PYGB |
[(2S,3R,4S,5S,6R)-3,4,5-trihydroxy-6-(hydroxymethyl)oxan-2-yl]methyl methanesulfonate |
5010000 |
NA |
NA |
NA |
NA |
NA |
BindingDB |
| PYGB |
N-phenyl-2-[(2S,3R,4S,5S,6R)-3,4,5-trihydroxy-6-(hydroxymethyl)oxan-2-yl]sulfanylacetamide |
3600000 |
NA |
NA |
NA |
NA |
NA |
BindingDB |