| GENE_SYMBOL |
DRUG_NAME |
Ki (nM) |
IC50 (nM) |
Kd (nM) |
EC50 (nM) |
Potency (nM) |
AC50 (nM) |
Datasource |
| PYGB |
(2R,3R,4S,5S,6R)-2-(2-hydroxyethoxy)-6-(hydroxymethyl)oxane-3,4,5-triol |
25100000 |
NA |
NA |
NA |
NA |
NA |
BindingDB |
| PYGB |
2-Deoxy-2-fluoro-alpha-d-glucopyranosyl fluoride |
199000 |
NA |
NA |
NA |
NA |
NA |
BindingDB |
| PYGB |
Glucosylurea |
140000 |
NA |
NA |
NA |
NA |
NA |
BindingDB |
| PYGB |
3,4,5-trihydroxy-6-(hydroxymethyl)-N-(4-hydroxyphenyl)oxane-2-carboxamide |
4400000 |
NA |
NA |
NA |
NA |
NA |
BindingDB |
| PYGB |
2-[3,4,5-Trihydroxy-6-(hydroxymethyl)oxan-2-yl]ethan-1-aminium |
4500000 |
NA |
NA |
NA |
NA |
NA |
BindingDB |
| PYGB |
3,4,5-Trihydroxy-6-hydroxymethyl-tetrahydro-pyran-2-carboxylic acid cyclopropylamide |
1300000 |
NA |
NA |
NA |
NA |
NA |
BindingDB |
| PYGB |
3,4,5-Trihydroxy-6-hydroxymethyl-tetrahydro-pyran-2-carboxylic acid (2,2,2-trifluoro-ethyl)-amide |
8100000 |
NA |
NA |
NA |
NA |
NA |
BindingDB |
| PYGB |
Methanesulfonic acid 3,4,5-trihydroxy-6-hydroxymethyl-tetrahydro-pyran-2-ylmethyl ester |
4800000 |
NA |
NA |
NA |
NA |
NA |
BindingDB |
| PYGB |
3,4,5-Trihydroxy-6-hydroxymethyl-tetrahydro-pyran-2-carboxylic acid (2-hydroxy-ethyl)-amide |
2600000 |
NA |
NA |
NA |
NA |
NA |
BindingDB |
| PYGB |
3,4,5-Trihydroxy-6-hydroxymethyl-tetrahydro-pyran-2-carboxylic acid methylamide |
160000 |
NA |
NA |
NA |
NA |
NA |
BindingDB |
| PYGB |
2-Amino-N-(3,4,5-trihydroxy-6-hydroxymethyl-tetrahydro-pyran-2-yl)-acetamide |
370000 |
NA |
NA |
NA |
NA |
NA |
BindingDB |
| PYGB |
(5S,8R,9S)-8,9,10-trihydroxy-6-oxa-1,3-diazaspiro[4.5]decane-2,4-dione |
11500000 |
NA |
NA |
NA |
NA |
NA |
BindingDB |
| PYGB |
(2R,4S,5S)-3,4,5-trihydroxy-6-(hydroxymethyl)oxane-2-carboxamide |
440000 |
NA |
NA |
NA |
NA |
NA |
BindingDB |
| PYGB |
2,2,2-Trifluoro-N-(3,4,5-trihydroxy-6-hydroxymethyl-tetrahydro-pyran-2-yl)-acetamide |
710000 |
NA |
NA |
NA |
NA |
NA |
BindingDB |
| PYGB |
(5R,8S,9S)-8,9,10-trihydroxy-7-(hydroxymethyl)-6-oxa-1,3-diazaspiro[4.5]decane-2,4-dione |
105000 |
NA |
NA |
NA |
NA |
NA |
BindingDB |
| PYGB |
(2S,4S,5S)-3,4,5-trihydroxy-6-(hydroxymethyl)oxane-2-carboxamide |
370000 |
NA |
NA |
NA |
NA |
NA |
BindingDB |
| PYGB |
6-Hydroxymethyl-tetrahydro-pyran-2,3,4,5-tetraol |
1700000 |
NA |
NA |
NA |
NA |
NA |
BindingDB |
| PYGB |
2,3,4,5-Tetrahydroxy-6-hydroxymethyl-tetrahydro-pyran-2-carboxylic acid amide |
3100000 |
NA |
NA |
NA |
NA |
NA |
BindingDB |
| PYGB |
(R)-3,4,5-Trihydroxy-6-hydroxymethyl-tetrahydro-pyran-2-carboxylic acid methylamide |
160000 |
NA |
NA |
NA |
NA |
NA |
BindingDB |
| PYGB |
(R)-2-Hydroxymethyl-6-methyl-tetrahydro-pyran-3,4,5-triol |
53100000 |
NA |
NA |
NA |
NA |
NA |
BindingDB |