| GENE_SYMBOL |
DRUG_NAME |
Ki (nM) |
IC50 (nM) |
Kd (nM) |
EC50 (nM) |
Potency (nM) |
AC50 (nM) |
Datasource |
| PTPRF |
5-(3-Aminophenyl)-3-(carboxyformamido)thiophene-2-carboxylic acid |
113000 |
NA |
NA |
NA |
NA |
NA |
BindingDB |
| PTPRG |
Cefsulodin |
NA |
200000 |
NA |
NA |
NA |
NA |
PubChem |
| PTPRJ |
Celastrol |
NA |
111500 |
NA |
NA |
NA |
NA |
PubChem |
| PTPRJ |
(2R,4aS,6aS,12bR,14aS,14bR)-10-Hydroxy-2,4a,6a,9,12b,14a-hexamethyl-11-oxo-1,2,3,4,4a,5,6,6a,11,12b,13,14,14a,14b-tetradecahydro-picene-2-carboxylic acid |
NA |
111500 |
NA |
NA |
NA |
NA |
BindingDB |
| PTPRM |
Cefsulodin |
NA |
200000 |
NA |
NA |
NA |
NA |
PubChem |
| PYCR1 |
N-[(4-bromophenyl)methyl]-N-methylprop-2-en-1-amine |
NA |
161000 |
NA |
NA |
NA |
NA |
ChEMBL |
| PYCR1 |
n-(2-Bromobenzyl)-n-methylprop-2-yn-1-amine |
NA |
2e+05 |
NA |
NA |
NA |
NA |
ChEMBL |
| PYCR1 |
1-[4-[[Methyl(prop-2-ynyl)amino]methyl]phenyl]ethanone |
NA |
184000 |
NA |
NA |
NA |
NA |
ChEMBL |
| PYCR1 |
N-[(2,4-dibromophenyl)methyl]-N-methylprop-2-yn-1-amine |
NA |
228000 |
NA |
NA |
NA |
NA |
ChEMBL |
| PYCR1 |
N-methyl-N-[(4-propan-2-ylphenyl)methyl]prop-2-yn-1-amine |
NA |
142000 |
NA |
NA |
NA |
NA |
ChEMBL |
| PYCR1 |
N-methyl-N-[(4-phenylphenyl)methyl]prop-2-yn-1-amine |
NA |
315000 |
NA |
NA |
NA |
NA |
ChEMBL |
| PYCR1 |
N-[(4-bromophenyl)methyl]-N-methylbut-3-yn-2-amine |
NA |
394000 |
NA |
NA |
NA |
NA |
ChEMBL |
| PYCR1 |
N-[[4-(4-fluorophenyl)phenyl]methyl]-N-methylprop-2-yn-1-amine |
NA |
211000 |
NA |
NA |
NA |
NA |
ChEMBL |
| PYCR1 |
N-[1-(4-bromophenyl)ethyl]-N-methylprop-2-yn-1-amine |
NA |
316000 |
NA |
NA |
NA |
NA |
ChEMBL |
| PYCR1 |
Chlorzymine |
NA |
139000 |
NA |
NA |
NA |
NA |
ChEMBL |
| PYCR1 |
N-[(3-bromophenyl)methyl]-N-methylprop-2-yn-1-amine |
NA |
276000 |
NA |
NA |
NA |
NA |
ChEMBL |
| PYCR1 |
Pargyline |
NA |
198000 |
NA |
NA |
NA |
NA |
ChEMBL|PubChem |
| PYCR1 |
N-[(4-fluorophenyl)methyl]-N-methylprop-2-yn-1-amine |
NA |
311000 |
NA |
NA |
NA |
NA |
ChEMBL |
| PYCR1 |
N-[(4-bromophenyl)methyl]-N-methylbut-3-yn-1-amine |
NA |
337000 |
NA |
NA |
NA |
NA |
ChEMBL |
| PYCR1 |
N-methyl-N-[(3-nitrophenyl)methyl]prop-2-yn-1-amine |
NA |
394000 |
NA |
NA |
NA |
NA |
ChEMBL |