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Drugs And Genes
Negative Drug Target Genes
GENE_SYMBOL DRUG_NAME Ki (nM) IC50 (nM) Kd (nM) EC50 (nM) Potency (nM) AC50 (nM) Datasource
PTPRF {4-[3-(4-Oxalyl-phenoxymethyl)-benzyloxy]-phenyl}-oxo-acetic acid NA 120000 NA NA NA NA BindingDB
PTPRF 2-(Carboxyformamido)-3-methylbenzoic acid 2000000 NA NA NA NA NA BindingDB
PTPRF {4-[4-(4-Oxalyl-phenoxymethyl)-benzyloxy]-phenyl}-oxo-acetic acid NA 250000 NA NA NA NA BindingDB
PTPRF {4-[2-(4-Oxalyl-phenoxymethyl)-benzyloxy]-phenyl}-oxo-acetic acid NA 120000 NA NA NA NA BindingDB
PTPRF Oleanolic Acid NA 120000 NA NA NA NA PubChem
PTPRF 2-(carboxyformamido)-5,6,7,8-tetrahydro-4H-cyclohepta[b]thiophene-3-carboxylic acid 400000 NA NA NA NA NA BindingDB
PTPRF 3-(Carboxyformamido)isonicotinic acid 2000000 NA NA NA NA NA BindingDB
PTPRF 2-(1-carboxy-N-methylformamido)benzoic acid 2000000 NA NA NA NA NA BindingDB
PTPRF 2-(Carboxyformamido)-6-methylbenzoic acid 2000000 NA NA NA NA NA BindingDB
PTPRF Benzo[b]thieno[2,3-d]thiophene-2-carboxylic acid, 3-(carboxymethoxy)- 1100000 NA NA NA NA NA BindingDB
PTPRF 3-(Carboxyformamido)-4-methylthiophene-2-carboxylic acid 2000000 NA NA NA NA NA BindingDB
PTPRF 3-(Carboxyformamido)-5-(4-chlorophenyl)thiophene-2-carboxylic acid 160000 NA NA NA NA NA BindingDB
PTPRF Novo Nordisk a/S Compound 420000 NA NA NA NA NA BindingDB
PTPRF 6-(carboxyformamido)-1H-indole-7-carboxylic acid 450000|550000 NA NA NA NA NA BindingDB
PTPRF 4-Bromo-3-(carboxymethoxy)-5-[4-[[oxo(3-pyridinyl)methyl]amino]phenyl]-2-thiophenecarboxylic acid NA|320000 320000|NA NA NA NA NA BindingDB
PTPRF 4-Hydroxyphenylglyoxylic acid NA 2300000 NA NA NA NA BindingDB
PTPRF Illudalic acid 130000 NA NA NA NA NA BindingDB
PTPRF 1-[1-[2-[2-[2-[Bis[2-hydroxy-3-[4-(2-methoxyethyl)phenoxy]propyl]amino]propoxy]propoxy]propoxy]propan-2-ylamino]-3-[4-(2-methoxyethyl)phenoxy]propan-2-ol NA 129800 NA NA NA NA BindingDB
PTPRF 2-(carboxyformamido)-5,6-dihydro-4H-cyclopenta[b]thiophene-3-carboxylic acid 900000 NA NA NA NA NA BindingDB
PTPRF 2-(Oxaloamino)thiophene-3-carboxylic acid 2000000 NA NA NA NA NA BindingDB