| GENE_SYMBOL |
DRUG_NAME |
Ki (nM) |
IC50 (nM) |
Kd (nM) |
EC50 (nM) |
Potency (nM) |
AC50 (nM) |
Datasource |
| PTPRC |
Fluoro{7-[fluoro(phosphonato)methyl]-2-naphthyl}methylphosphonate |
NA |
279000 |
NA |
NA |
NA |
NA |
BindingDB |
| PTPRC |
[Fluoro-[7-[fluoro(phosphono)methyl]naphthalen-2-yl]methyl]phosphonic acid |
NA |
279000 |
NA |
NA |
NA |
NA |
TTD |
| PTPRC |
2-(Oxaloamino)thiophene-3-carboxylic acid |
210000 |
NA |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| PTPRC |
3-(Carboxyformamido)thiophene-2-carboxylic acid |
260000 |
NA |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| PTPRC |
[[4-[4-[4-[Difluoro(phosphonato)methyl]phenyl]butyl]phenyl]-difluoromethyl]-dioxido-oxo-lambda5-phosphane |
NA |
198000 |
NA |
NA |
NA |
NA |
BindingDB |
| PTPRC |
2-(Oxalyl-Amino)-Benzoic Acid |
160000 |
NA |
NA |
NA |
NA |
NA |
BindingDB|PubChem|TTD |
| PTPRC |
((4-(4-(4-(Difluoro-Phosphono-Methyl)-Phenyl)-Butyl)-Phenyl)-Difluoro-Methyl)-Phosphonic Acid |
NA |
198000 |
NA |
NA |
NA |
NA |
TTD |
| PTPRC |
7-(1,1-Dioxo-1h-Benzo(D)Isothiazol-3-Yloxymethyl)-2-(Oxalyl-Amino)-4,7-Dihydro-5h-Thieno(2,3-C)Pyran-3-Carboxylic Acid |
489000 |
NA |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| PTPRC |
n-Acetyl-4-[(carboxycarbonyl)(2-carboxyphenyl)amino]-n-pentyl-1-naphthylalaninamide |
300000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| PTPRC |
Azane;[[7-[difluoro(phosphono)methyl]naphthalen-2-yl]-difluoromethyl]phosphonic acid |
NA |
180000 |
NA |
NA |
NA |
NA |
TTD |
| PTPRC |
Azane;[[4-[2-[[4-[difluoro(phosphono)methyl]phenyl]methoxy]ethoxymethyl]phenyl]-difluoromethyl]phosphonic acid |
NA |
236000 |
NA |
NA |
NA |
NA |
TTD |
| PTPRC |
Azane;[4-[4-ethoxy-2,2-bis(methoxycarbonyl)-4-oxobutyl]phenyl]sulfamic acid |
NA |
126000 |
NA |
NA |
NA |
NA |
TTD |
| PTPRC |
Azane;[4-[2-ethoxycarbonyl-3-methoxy-3-oxo-2-(phenylmethoxycarbonylamino)propyl]phenyl]sulfamic acid |
NA |
280000 |
NA |
NA |
NA |
NA |
TTD |
| PTPRC |
{3(S)-Methylcarbamoyl-2-[3-(3-sulfoamino-phenyl)-propionyl]-1,2,3,4-tetrahydro-isoquinolin-7-YL}-sulfamic acid |
NA |
500000 |
NA |
NA |
NA |
NA |
TTD |
| PTPRC |
3-[(3,4-Dimethylphenyl)methylsulfanyl]thiophene-2-carboxylic acid |
NA |
120000 |
NA |
NA |
NA |
NA |
TTD |
| PTPRC |
3-(Naphthalen-2-ylmethylsulfanyl)thiophene-2-carboxylic acid |
NA |
120000 |
NA |
NA |
NA |
NA |
TTD |
| PTPRC |
3-[(3,4-Dichlorophenyl)methylamino]thiophene-2-carboxylic acid |
NA |
120000 |
NA |
NA |
NA |
NA |
TTD |
| PTPRC |
3-[(3,4-Dichlorophenyl)methylsulfonyl]thiophene-2-carboxylic acid |
NA |
120000 |
NA |
NA |
NA |
NA |
TTD |
| PTPRC |
alpha,alpha-Bis(trifluoromethyl)benzyl alcohol |
NA |
500000 |
NA |
NA |
NA |
NA |
TTD |
| PTPRC |
3-[2-(3-Fluorophenyl)ethyl]-6-hydroxy-2-phenyl-benzofuran-5-carboxylic acid |
NA |
120000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |