| GENE_SYMBOL |
DRUG_NAME |
Ki (nM) |
IC50 (nM) |
Kd (nM) |
EC50 (nM) |
Potency (nM) |
AC50 (nM) |
Datasource |
| RAPGEF4 |
2-Methoxyestradiol |
NA |
NA |
NA |
NA |
125892 |
NA |
PubChem |
| RAPGEF4 |
Diphacinone |
NA |
NA |
NA |
NA |
112202 |
NA |
PubChem |
| RAPGEF4 |
Miconazole Nitrate |
NA |
NA |
NA |
NA |
112202 |
NA |
PubChem |
| RAPGEF4 |
|
NA |
127000 |
NA |
NA |
NA |
NA |
BindingDB |
| RAPGEF4 |
2-Fluoro-5-[4-(2,4,6-Trimethyl-Benzenesulfonyl)-Phenyl]-Pyridine |
NA |
300000 |
NA |
NA |
NA |
NA |
TTD |
| RAPGEF4 |
(4,5-Dimethyl-Thiazol-2-Yl)-(2,4,6-Trimethyl-Phenyl)-Amine |
NA |
300000 |
NA |
NA |
NA |
NA |
TTD |
| RAPGEF4 |
1,3,5-Trimethyl-2-(4-Pentyl-Benzenesulfonyl)-Benzene |
NA |
300000 |
NA |
NA |
NA |
NA |
TTD |
| RAPGEF4 |
2-(4-Cyclohexyl-Benzenesulfonyl)-1,3,5-Trimethyl-Benzene |
NA |
300000 |
NA |
NA |
NA |
NA |
TTD |
| RAPGEF4 |
2-(4-Cyclohexyloxy-Benzenesulfonyl)-1,3,5-Trimethyl-Benzene |
NA |
300000 |
NA |
NA |
NA |
NA |
TTD |
| RAPGEF4 |
4-[4-(2,4,6-Trimethyl-Benzenesulfonyl)-Phenoxy]-Piperidine-1-Carboxylic Acid Tert-Butyl Ester |
NA |
300000 |
NA |
NA |
NA |
NA |
TTD |
| RAPGEF4 |
4-[4-(2,4,6-Trimethylphenyl)sulfonylphenoxy]piperidine |
NA |
300000 |
NA |
NA |
NA |
NA |
TTD |
| RAPGEF4 |
2-[4-(2,4,6-Trimethyl-Benzenesulfonyl)-Phenoxy]-Ethylamine |
NA |
300000 |
NA |
NA |
NA |
NA |
TTD |
| RAPGEF4 |
2-Ethyl-1-(4-Trifluoromethyl-Benzenesulfonyl)-1H-Pyrrole |
NA |
300000 |
NA |
NA |
NA |
NA |
TTD |
| RAPGEF4 |
1-(2,4,6-Trimethyl-Benzenesulfonyl)-1H-Indole-5-Carboxylic Acid Methyl Ester |
NA |
300000 |
NA |
NA |
NA |
NA |
TTD |
| RAPGEF4 |
Parthenolide |
NA |
NA |
NA |
NA |
158489 |
NA |
PubChem |
| RAPGEF4 |
Chloranil |
NA |
NA |
NA |
NA |
125892 |
NA |
PubChem |
| RAPGEF4 |
Isopropyl Palmitate |
NA |
NA |
NA |
NA |
112202 |
NA |
PubChem |
| RAPGEF4 |
Curcumin |
NA |
NA |
NA |
NA |
112202 |
NA |
PubChem |
| RARA |
(2E,4E,6E,8E)-3,7-Dimethyl-9-(2,6,6-trimethyl-3-[1,2,4]triazol-4-yl-cyclohex-1-enyl)-nona-2,4,6,8-tetraenoic acid |
NA |
410000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| RARA |
N-(1H-imidazole-1-yl)-(E)-retinamide |
NA |
1000000 |
NA |
NA |
NA |
NA |
TTD |