| GENE_SYMBOL |
DRUG_NAME |
Ki (nM) |
IC50 (nM) |
Kd (nM) |
EC50 (nM) |
Potency (nM) |
AC50 (nM) |
Datasource |
| RARA |
Psilocin |
NA |
NA |
NA |
NA |
135464 |
NA |
PubChem |
| RARA |
Triamcinolone Acetonide |
NA |
NA |
NA |
NA |
149601 |
NA |
PubChem |
| RARA |
Miristalkonium chloride |
NA |
NA |
NA |
NA |
22387200 |
NA |
PubChem |
| RARA |
(2E,4E,6E,8E)-3,7-Dimethyl-9-(2,6,6-trimethyl-3-[1,2,4]triazol-1-yl-cyclohex-1-enyl)-nona-2,4,6,8-tetraenoic acid |
NA |
1000000 |
NA |
NA |
NA |
NA |
TTD |
| RARB |
(2E,4E,6E,8E)-3,7-Dimethyl-9-(2,6,6-trimethyl-3-[1,2,4]triazol-4-yl-cyclohex-1-enyl)-nona-2,4,6,8-tetraenoic acid |
NA |
250000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| RARB |
4-((+/-)-(1H-imidazol-1-yl)-(13Z)-retinoic acid |
NA |
175000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| RARB |
N-(1H-imidazole-1-yl)-(E)-retinamide |
NA |
500000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| RARB |
Irx-5183 |
NA |
NA |
1000000 |
NA |
NA |
NA |
PubChem |
| RARB |
(2E,4E,6E,8E)-3,7-Dimethyl-9-(2,6,6-trimethyl-3-[1,2,4]triazol-1-yl-cyclohex-1-enyl)-nona-2,4,6,8-tetraenoic acid |
NA |
1000000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| RARB |
4-((+/-)-(1H-imidazol-1-yl)-(E)-retinoic acid |
NA |
175000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| RARG |
Gka-50 |
NA |
1000000 |
NA |
NA |
NA |
NA |
TTD |
| RARG |
Irx-5183 |
NA |
NA |
1000000 |
NA |
NA |
NA |
PubChem |
| RCOR1 |
Tranylcypromine |
168000 |
NA |
NA |
NA |
NA |
NA |
BindingDB |
| RCOR1 |
(+)-Tranylcypromine |
284000 |
NA |
NA |
NA |
NA |
NA |
BindingDB |
| RCOR1 |
N~4~-(1-Benzylpiperidin-4-Yl)-N~2~-[3-(Dimethylamino)propyl]-6,7-Dimethoxyquinazoline-2,4-Diamine |
NA |
NA |
243000 |
NA |
NA |
NA |
BindingDB |
| REN |
methyl (2S)-2-[[(2S)-2-[[(2S)-2-[[(2R)-2-hydroxy-4-methylpentanoyl]amino]-4-methylpentanoyl]amino]-3-methylbutanoyl]amino]-3-phenylpropanoate |
600000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| REN |
methyl (2S)-2-[[(2S)-2-[[(2S)-2-[[(2R)-2-hydroxy-3-methylbutanoyl]amino]-4-methylpentanoyl]amino]-3-methylbutanoyl]amino]-3-phenylpropanoate |
1780000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| REN |
N-[3-[(1S,5S,6S)-3-amino-1-(methoxymethyl)-5-methyl-2-thia-4-azabicyclo[4.1.0]hept-3-en-5-yl]-4,5-difluorophenyl]-5-prop-2-ynoxypyrazine-2-carboxamide |
NA |
678000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| REN |
CID 118866986 |
NA |
214000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| REN |
Leu-Leu-Val-Phe-OCH3 |
500000|1140000 |
NA |
NA |
NA |
NA |
NA |
BindingDB|TTD |