| GENE_SYMBOL |
DRUG_NAME |
Ki (nM) |
IC50 (nM) |
Kd (nM) |
EC50 (nM) |
Potency (nM) |
AC50 (nM) |
Datasource |
| REN |
Boc-Trp-Trp-Sta-Ala-Sta-OMe |
NA |
150000 |
NA |
NA |
NA |
NA |
BindingDB |
| REN |
5-(1H-indol-7-yl)-4,6-dimethylpyridin-2-amine |
NA |
124000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| REN |
N,N'-(Iminodiethane-2,1-Diyl)bis[4-Amino-N-(2-Methylpropyl)benzenesulfonamide] |
NA |
250000 |
NA |
NA |
NA |
NA |
TTD |
| REN |
N,N'-(iminodiethane-2,1-diyl)bis(4-amino-N-benzylbenzenesulfonamide) |
NA |
250000 |
NA |
NA |
NA |
NA |
TTD |
| REN |
5,6,7,8-Tetrahydro[1]benzothieno[2,3-d]pyrimidin-4-amine |
NA |
300000 |
NA |
NA |
NA |
NA |
TTD |
| REN |
Furfurylamine |
NA |
300000 |
NA |
NA |
NA |
NA |
TTD |
| REN |
N-[2-[2-[benzenesulfonyl(benzyl)amino]ethylamino]ethyl]-N-benzylbenzenesulfonamide |
NA |
250000 |
NA |
NA |
NA |
NA |
TTD |
| REN |
N-[3-[2-[benzenesulfonyl(benzyl)amino]ethylamino]propyl]-N-benzylbenzenesulfonamide |
NA |
250000 |
NA |
NA |
NA |
NA |
TTD |
| REN |
N-[3-[3-[benzenesulfonyl(benzyl)amino]propylamino]propyl]-N-benzylbenzenesulfonamide |
NA |
250000 |
NA |
NA |
NA |
NA |
TTD |
| REN |
4-amino-N-[3-[2-[(4-aminophenyl)sulfonyl-benzylamino]ethylamino]propyl]-N-benzylbenzenesulfonamide |
NA |
250000 |
NA |
NA |
NA |
NA |
TTD |
| REN |
4-amino-N-[3-[3-[(4-aminophenyl)sulfonyl-benzylamino]propylamino]propyl]-N-benzylbenzenesulfonamide |
NA |
250000 |
NA |
NA |
NA |
NA |
TTD |
| REN |
Iso-butyl-substituted sulfonamide, 9a |
NA |
250000 |
NA |
NA |
NA |
NA |
TTD |
| REN |
Carboxamide, 12b |
NA |
250000 |
NA |
NA |
NA |
NA |
TTD |
| REN |
(1R,2R,4aR,4bS,6aS,9R,10S,10aS,12aR)-1-(carboxymethyl)-2-(2-carboxypropan-2-yl)-1,4a,4b,9,10-pentamethyl-2,3,4,5,6,7,8,9,10,10a,12,12a-dodecahydrochrysene-6a-carboxylic acid |
NA |
1991000 |
NA |
NA |
NA |
NA |
TTD |
| REN |
(2S)-N-[(2R)-1-(2,2-dimethylpropylamino)-1-oxo-3-phenylpropan-2-yl]-N'-[(2S)-1-hydroxy-4-methylpentan-2-yl]-2-(1H-imidazol-5-ylmethyl)propanediamide |
NA |
1200000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| REN |
Pro-His-Pro-Phe-Arg-Phe-Phe-Val-Tyr-Lys |
NA |
200000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| REN |
2-(2-{5-[2-Amino-3-(3H-imidazol-4-yl)-propionylamino]-7-methyl-oct-3-enoylamino}-3-methyl-butyrylamino)-3-phenyl-propionic acid methyl ester |
146000|500000 |
NA |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| REN |
His-Leu-Leu-Val-Phe-OCH3 |
540000 |
NA |
NA |
NA |
NA |
NA |
BindingDB |
| REN |
2-{2-[2-(2-Amino-4-methyl-pentanoylamino)-acetylamino]-3-methyl-butyrylamino}-3-phenyl-propionic acid methyl ester |
1000000 |
NA |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| REN |
2-[2-(5-Amino-7-methyl-oct-3-enoylamino)-3-methyl-butyrylamino]-3-phenyl-propionic acid methyl ester |
400000|800000 |
NA |
NA |
NA |
NA |
NA |
BindingDB|TTD |