| GENE_SYMBOL |
DRUG_NAME |
Ki (nM) |
IC50 (nM) |
Kd (nM) |
EC50 (nM) |
Potency (nM) |
AC50 (nM) |
Datasource |
| REN |
4-Methoxy-N-{4-[(3R,4R)-3-(naphthalen-2-ylmethoxy)-piperidin-4-yl]-benzyl}-benzamide |
NA |
1000000 |
NA |
NA |
NA |
NA |
TTD |
| REN |
(3S,4S)-4-(4-Chloro-phenyl)-3-(4-methoxy-benzyloxy)-piperidine |
NA |
1200000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| REN |
(3S,5S)-methyl 2-[1-(4-amino-2-hydroxy-6-methylheptylcarboxamido)-2-methyl-propylcarboxamido]-3-phenyl-propanoate |
170000|1180000|1600000 |
NA |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| REN |
(2R,3R,4S)-4-amino-N-butyl-5-cyclohexyl-2,3-dihydroxypentane-1-sulfonamide |
NA |
470000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| REN |
N-((1S,2R,3S)-4-Butylsulfamoyl-1-cyclohexylmethyl-2,3-dihydroxy-butyl)-acetamide |
NA |
1000000 |
NA |
NA |
NA |
NA |
TTD |
| REN |
4-(2-{4-[2-(2-tert-Butoxycarbonylamino-3-phenyl-propionylamino)-3-(3H-imidazol-4-yl)-propionylamino]-3-hydroxy-6-methyl-heptanoylamino}-propionylamino)-3-hydroxy-6-methyl-heptanoic acid methyl ester |
NA |
270000 |
NA |
NA |
NA |
NA |
BindingDB |
| REN |
4-Methyl-pentanoic acid ((1S,2R,3S)-4-butylsulfamoyl-1-cyclohexylmethyl-2,3-dihydroxy-butyl)-amide |
NA |
1000000 |
NA |
NA |
NA |
NA |
TTD |
| REN |
N-((1S,2R,3R)-4-Butylsulfamoyl-1-cyclohexylmethyl-2,3-dihydroxy-butyl)-3-(3H-imidazol-4-yl)-propionamide |
NA |
1000000 |
NA |
NA |
NA |
NA |
TTD |
| REN |
(2R,3R,4S)-N-butyl-5-cyclohexyl-2,3-dihydroxy-4-[3-(1H-imidazol-5-yl)propylamino]pentane-1-sulfonamide |
NA |
310000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| REN |
(2S)-N-[(2S,3R,4S)-5-(butylsulfamoyl)-1-cyclohexyl-3,4-dihydroxypentan-2-yl]-2-hydroxy-4-methylpentanamide |
NA |
1000000 |
NA |
NA |
NA |
NA |
TTD |
| REN |
(2S)-N-[(2S,3R,4R)-5-(butylsulfamoyl)-1-cyclohexyl-3,4-dihydroxypentan-2-yl]-2-hydroxy-4-methylpentanamide |
NA |
1000000 |
NA |
NA |
NA |
NA |
TTD |
| REN |
(2S)-2-amino-N-[(2S,3R,4R)-5-(butylsulfamoyl)-1-cyclohexyl-3,4-dihydroxypentan-2-yl]-4-methylpentanamide |
NA |
1000000 |
NA |
NA |
NA |
NA |
TTD |
| REN |
4-Methyl-pentanoic acid ((1S,2R,3R)-4-butylsulfamoyl-1-cyclohexylmethyl-2,3-dihydroxy-butyl)-amide |
NA |
1000000 |
NA |
NA |
NA |
NA |
TTD |
| REN |
(2R,3R,4S)-N-butyl-5-cyclohexyl-2,3-dihydroxy-4-(4-methylpentylamino)pentane-1-sulfonamide |
NA |
680000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| REN |
N-((1S,2R,3R)-4-Butylsulfamoyl-1-cyclohexylmethyl-2,3-dihydroxy-butyl)-acetamide |
NA |
1000000 |
NA |
NA |
NA |
NA |
TTD |
| REN |
(S)-N-[(S)-4-((S,R)-Butylsulfamoyl)-1-cyclohexylmethyl-2,3-dihydroxy-butyl]-3-(3H-imidazol-4-yl)-2-(2-phenyl-ethanesulfonylamino)-propionamide |
NA |
140000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| REN |
(S)-2-Amino-N-[4-((S,R,R)-butylsulfamoyl)-1-cyclohexylmethyl-2,3-dihydroxy-butyl]-3-(3H-imidazol-4-yl)-propionamide |
NA |
1000000 |
NA |
NA |
NA |
NA |
TTD |
| REN |
N-((1S,2R,3S)-4-Butylsulfamoyl-1-cyclohexylmethyl-2,3-dihydroxy-butyl)-3-(3H-imidazol-4-yl)-propionamide |
NA |
1000000 |
NA |
NA |
NA |
NA |
TTD |
| REN |
His-Sta-Leu-Phe-NH2 |
NA |
370000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| REN |
N-(3-{1-Hydroxy-2-[1-(3-methyl-butylcarbamoyl)-ethylcarbamoyl]-ethylamino}-1-isopropyl-2-oxo-3-phenyl-propyl)-3-methyl-butyramide |
NA |
140000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |