| GENE_SYMBOL |
DRUG_NAME |
Ki (nM) |
IC50 (nM) |
Kd (nM) |
EC50 (nM) |
Potency (nM) |
AC50 (nM) |
Datasource |
| ROCK2 |
US11078197, Example 89 |
NA |
716400 |
NA |
NA |
NA |
NA |
BindingDB |
| ROCK2 |
US11078197, Example 67 |
NA |
142000 |
NA |
NA |
NA |
NA |
BindingDB |
| ROCK2 |
US11078197, Example 87 |
NA |
156200 |
NA |
NA |
NA |
NA |
BindingDB |
| ROCK2 |
US11078197, Example 68 |
NA |
108000 |
NA |
NA |
NA |
NA |
BindingDB |
| ROCK2 |
US11078197, Example 162 |
NA |
162000 |
NA |
NA |
NA |
NA |
BindingDB |
| ROCK2 |
US11078197, Example 16 |
NA |
136700 |
NA |
NA |
NA |
NA |
BindingDB |
| ROCK2 |
N-[2-[2-(3-aminopropyl)-4-carbamoylpyrazol-1-ium-3-yl]oxyspiro[3.3]heptan-6-yl]-7-cyclopropyl-6-(2-hydroxy-2-methylpropoxy)pyrazolo[1,5-a]pyridine-3-carboxamide |
NA |
551100 |
NA |
NA |
NA |
NA |
BindingDB |
| ROCK2 |
3-[[3-fluoro-4-(5-methyl-7H-pyrrolo[2,3-d]pyrimidin-4-yl)phenyl]carbamoylamino]-N-propan-2-ylbenzamide |
NA |
781000 |
NA |
NA |
NA |
NA |
BindingDB |
| ROCK2 |
5-bromo-N-(pyridin-4-yl)nicotinamide |
NA |
357200 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| ROCK2 |
N-[3-(4-Dimethylaminomethyl-phenylcarbamoyl)-benzyl]-4-methoxy-3-trifluoromethyl-benzamide |
NA |
160000 |
NA |
NA |
NA |
NA |
BindingDB |
| ROCK2 |
N-[3-(4-Dimethylaminomethyl-phenylcarbamoyl)-benzyl]-4-methoxy-3-methyl-benzamide |
NA |
266000 |
NA |
NA |
NA |
NA |
BindingDB |
| ROCK2 |
N-[3-(4-Dimethylaminomethyl-phenylcarbamoyl)-benzyl]-4-methoxy-benzamide |
NA |
1300000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| ROCK2 |
4-Cyano-N-[3-(4-dimethylaminomethyl-phenylcarbamoyl)-benzyl]-benzamide |
NA |
1700000 |
NA |
NA |
NA |
NA |
BindingDB |
| ROCK2 |
3-Chloro-N-[3-(4-dimethylaminomethyl-phenylcarbamoyl)-benzyl]-4-trifluoromethoxy-benzamide |
NA |
670000 |
NA |
NA |
NA |
NA |
BindingDB |
| ROCK2 |
3-[3-(3,4-Dimethoxy-phenyl)-ureidomethyl]-N-(2-piperidin-3-ylethyl)-benzamide |
NA |
1600000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| ROCK2 |
N-{3-[3-(4-Cyano-phenyl)-ureidomethyl]-phenyl}-3-piperidin-3-yl-propionamide |
NA |
110000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| ROCK2 |
3,4-Dimethoxy-N-{3-[2-(1-methyl-piperidin-3-yl)-ethylcarbamoyl]-benzyl}-benzamide |
NA |
102000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| ROCK2 |
1-Amino-5-piperidin-1-yl-6,7,8,9-tetrahydrothieno[2,3-c]isoquinoline-2-carboxamide |
NA |
142800 |
NA |
NA |
NA |
NA |
BindingDB |
| ROCK2 |
N-[4-(2-amino-1,5-dicyano-4,4-diethoxy-3-azabicyclo[3.1.0]hex-2-en-6-yl)phenyl]acetamide |
NA |
445300 |
NA |
NA |
NA |
NA |
BindingDB |
| ROCK2 |
|
NA |
200000 |
NA |
NA |
NA |
NA |
BindingDB |