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Drugs And Genes
Negative Drug Target Genes
Gene
Drug
GENE_SYMBOL
DRUG_NAME
Ki (nM)
IC50 (nM)
Kd (nM)
EC50 (nM)
Potency (nM)
AC50 (nM)
Datasource
RORC
N-[(4-methylphenyl)sulfonyl]-N-[3-(trifluoromethyl)phenyl]glycine
NA
151900
NA
NA
NA
NA
TTD
RORC
N-(3-chloro-4-ethoxyphenyl)acetamide
NA
216000
NA
NA
NA
NA
ChEMBL|TTD
RORC
N-(4-carbamoylphenyl)-3-[(4-chlorophenoxy)methyl]benzamide
NA
168270
NA
NA
NA
NA
TTD
RORC
2-({4-allyl-5-[3-(1,3-dioxo-1H-benzo[de]isoquinolin-2(3H)-yl)propyl]-4H-1,2,4-triazol-3-yl}sulfanyl)-N-[4-(aminosulfonyl)phenyl]acetamide
NA
142210
NA
NA
NA
NA
TTD
RORC
Bromoethane
NA
NA
NA
NA
133332
NA
PubChem
RORC
2-(4-(Ethylsulfonyl)phenyl)acetamide
NA
500000
NA
NA
NA
NA
TTD
RORC
N-(2-benzoylphenyl)-1-ethyl-2-oxobenzo[cd]indole-6-sulfonamide
NA
156300
NA
NA
NA
NA
TTD
RORC
1-ethyl-N-[(4-methoxyphenyl)methyl]-2-oxobenzo[cd]indole-6-sulfonamide
NA
174400
NA
NA
NA
NA
TTD
RPA1
7-methyl-3-phenyl-1H-indole-2-carboxylic acid
NA
NA
640000
NA
NA
NA
ChEMBL
RPA1
5-(4-Chlorophenyl)-1H-tetrazole
NA
NA
1850000
NA
NA
NA
ChEMBL
RPA1
5-(3-Chloro-4-fluorophenyl)furan-2-carboxylic acid
NA
NA
1400000|710000
NA
NA
NA
ChEMBL
RPA1
1-(3-Methylphenyl)-5-Phenyl-1h-Pyrazole-3-Carboxylic Acid
NA
NA
580000
NA
NA
NA
ChEMBL
RPA1
3-(4-Fluorophenyl)-1H-pyrazole-5-carboxylic acid
NA
NA
1120000
NA
NA
NA
ChEMBL
RPL10
NB-124 sulfate
NA
1493000
NA
NA
NA
NA
PubChem
RPL10A
NB-124 sulfate
NA
1493000
NA
NA
NA
NA
PubChem
RPL11
NB-124 sulfate
NA
1493000
NA
NA
NA
NA
PubChem
RPL12
NB-124 sulfate
NA
1493000
NA
NA
NA
NA
PubChem
RPL13
NB-124 sulfate
NA
1493000
NA
NA
NA
NA
PubChem
RPL13A
NB-124 sulfate
NA
1493000
NA
NA
NA
NA
PubChem
RPL14
NB-124 sulfate
NA
1493000
NA
NA
NA
NA
PubChem
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