| GENE_SYMBOL |
DRUG_NAME |
Ki (nM) |
IC50 (nM) |
Kd (nM) |
EC50 (nM) |
Potency (nM) |
AC50 (nM) |
Datasource |
| ROCK2 |
4-Methoxy-N-[3-(2-pyridin-4-yl-ethylcarbamoyl)-benzyl]-benzamide |
NA |
7000000 |
NA |
NA |
NA |
NA |
TTD |
| ROCK2 |
3-Methoxy-N-[3-(2-pyridin-4-yl-ethylcarbamoyl)-benzyl]-benzamide |
NA |
7000000 |
NA |
NA |
NA |
NA |
TTD |
| ROCK2 |
1,3-Benzodioxole-5-carboxylic acid 3-(2-pyridin-4-yl-ethylcarbamoyl)-benzylamide |
NA |
7000000 |
NA |
NA |
NA |
NA |
TTD |
| ROCK2 |
3,4-Dimethyl-N-[3-(2-pyridin-4-yl-ethylcarbamoyl)-benzyl]-benzamide |
NA |
7000000 |
NA |
NA |
NA |
NA |
TTD |
| ROCK2 |
N-[3-(Isoquinolin-6-ylcarbamoyl)-benzyl]-3,4-dimethoxy-benzamide |
NA |
685000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| ROCK2 |
3-[(3,4-dimethoxyphenyl)carbamoylamino]-N-(2-piperidin-3-ylethyl)benzamide |
NA |
7000000 |
NA |
NA |
NA |
NA |
TTD |
| ROCK2 |
N-(3,4-Dimethoxy-benzyl)-N-(2-piperidin-3-yl-ethyl)-isophthalamide |
NA |
6000000 |
NA |
NA |
NA |
NA |
TTD |
| ROCK2 |
3-[2-(3,4-Dimethoxy-phenyl)-acetylamino]-N-(2-piperidin-3-ylethyl)-benzamide |
NA |
3200000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| ROCK2 |
3,4-Dimethoxy-N-[3-(2-piperidin-3-yl-ethylcarbamoyl)-phenyl]-benzamide |
NA |
6000000 |
NA |
NA |
NA |
NA |
TTD |
| ROCK2 |
3-[(3,4-Dimethoxy-benzenesulfonylamino)-methyl]-N-(2-piperidin-3-yl-ethyl)-benzamide |
NA |
6000000 |
NA |
NA |
NA |
NA |
TTD |
| ROCK2 |
3-[3-(3-Amido-phenyl)-ureidomethyl]-N-(4-dimethylaminomethylphenyl)-benzamide |
NA |
240000 |
NA |
NA |
NA |
NA |
BindingDB |
| ROCK2 |
(R)-2-(6-acetamidohexanamido)-6-amino-N-(6-((R)-1-((R)-1-amino-5-guanidino-1-oxopentan-2-ylamino)-5-guanidino-1-oxopentan-2-ylamino)-6-oxohexyl)hexanamide |
NA |
NA |
123000 |
NA |
NA |
NA |
BindingDB |
| ROCK2 |
3-methyl-N-(2-pyridin-3-yl-1,3-benzoxazol-5-yl)-1-benzofuran-2-carboxamide |
NA |
1009000 |
NA |
NA |
NA |
NA |
BindingDB |
| ROCK2 |
5-(4-fluorophenyl)-N-pyridin-4-ylpyridine-3-carboxamide |
NA |
400000 |
NA |
NA |
NA |
NA |
TTD |
| ROCK2 |
4-chloro-N-pyridin-4-ylpyridine-3-carboxamide |
NA |
221400 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| ROCK2 |
4-(4-fluorophenyl)-N-pyridin-4-ylpyridine-3-carboxamide |
NA |
400000 |
NA |
NA |
NA |
NA |
TTD |
| ROCK2 |
5-Aminoindazole |
NA |
119700 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| ROCK2 |
2-azanyl-7-oxidanyl-4-pyridin-4-yl-4H-chromene-3-carbonitrile |
NA |
126600 |
NA |
NA |
NA |
NA |
BindingDB |
| RORB |
5-[2,3-dichloro-4-[[(2S)-1,1,1-trifluoropropan-2-yl]sulfamoyl]phenyl]-4-(4-fluoropiperidine-1-carbonyl)-N-[2-methyl-2-(5-oxo-4H-1,2,4-oxadiazol-3-yl)propyl]-1,3-thiazole-2-carboxamide |
NA |
NA |
335000 |
NA |
NA |
NA |
BindingDB |
| RORC |
N-[4-(1,1,1,3,3,3-hexafluoro-2-hydroxypropan-2-yl)phenyl]-2-[N-(4-methylphenyl)sulfonyl-3-(trifluoromethyl)anilino]acetamide |
NA |
112250 |
NA |
NA |
NA |
NA |
TTD |