| GENE_SYMBOL |
DRUG_NAME |
Ki (nM) |
IC50 (nM) |
Kd (nM) |
EC50 (nM) |
Potency (nM) |
AC50 (nM) |
Datasource |
| RPS3 |
NB-124 sulfate |
NA |
1493000 |
NA |
NA |
NA |
NA |
PubChem |
| RPS3A |
NB-124 sulfate |
NA |
1493000 |
NA |
NA |
NA |
NA |
PubChem |
| RPS4X |
NB-124 sulfate |
NA |
1493000 |
NA |
NA |
NA |
NA |
PubChem |
| RPS4Y1 |
NB-124 sulfate |
NA |
1493000 |
NA |
NA |
NA |
NA |
PubChem |
| RPS5 |
NB-124 sulfate |
NA |
1493000 |
NA |
NA |
NA |
NA |
PubChem |
| RPS6 |
NB-124 sulfate |
NA |
1493000 |
NA |
NA |
NA |
NA |
PubChem |
| RPS6KA1 |
1H-Pyrrole-3-carboxamide, 5-((5-fluoro-1,2-dihydro-2-oxo-3H-indol-3-ylidene)methyl)-N-((2S)-2-hydroxy-3-(4-morpholinyl)propyl)-2,4-dimethyl- |
180000|5800000 |
NA |
NA |
NA |
NA |
NA |
BindingDB |
| RPS6KA1 |
Ruboxistaurin |
400000 |
NA |
NA |
NA |
NA |
NA |
BindingDB |
| RPS6KA1 |
Canertinib |
6200000 |
NA |
NA |
NA |
NA |
NA |
BindingDB |
| RPS6KA1 |
SB 203580 |
320000 |
NA |
NA |
NA |
NA |
NA |
BindingDB |
| RPS6KA1 |
N-[(2R,3S,4S,6S)-3-methoxy-2-methyl-16-oxo-29-oxa-1,7,17-triazaoctacyclo[12.12.2.12,6.07,28.08,13.015,19.020,27.021,26]nonacosa-8,10,12,14,19,21,23,25,27-nonaen-4-yl]-N-methylbenzamide |
690000 |
NA |
NA |
NA |
NA |
NA |
BindingDB |
| RPS6KA1 |
2-(2-chlorophenyl)-5,7-dihydroxy-8-[(3S)-3-hydroxy-1-methyl-4-piperidyl]chromone |
720000|2300000 |
NA |
NA |
NA |
NA |
NA |
BindingDB |
| RPS6KA1 |
Vandetanib |
400000 |
NA |
NA |
NA |
NA |
NA |
BindingDB |
| RPS6KA1 |
9,13-Epoxy-1H,9H-diindolo[1,2,3-gh:3',2',1'-lm]pyrrolo[3,4-j][1,7]benzodiazonin-1-one, 2,3,10,11,12,13-hexahydro-10-methoxy-9-methyl-11-(methylamino)-, (9S,10R,11R,13R)- |
1200000 |
NA |
NA |
NA |
NA |
NA |
BindingDB |
| RPS6KA1 |
4-(4-(benzo[d][1,3]dioxol-5-yl)-5-(pyridin-2-yl)-1H-imidazol-2-yl)benzamide |
1300000 |
NA |
NA |
NA |
NA |
NA |
BindingDB |
| RPS6KA1 |
Sunitinib |
140000|5000000 |
NA |
NA |
NA |
NA |
NA |
BindingDB |
| RPS6KA1 |
Jnj-7706621 |
4000000 |
NA |
NA |
NA |
NA |
NA |
BindingDB |
| RPS6KA1 |
|
170000 |
NA |
NA |
NA |
NA |
NA |
BindingDB |
| RPS6KA1 |
|
450000 |
NA |
NA |
NA |
NA |
NA |
BindingDB |
| RPS6KA2 |
1H-Pyrrole-3-carboxamide, 5-((5-fluoro-1,2-dihydro-2-oxo-3H-indol-3-ylidene)methyl)-N-((2S)-2-hydroxy-3-(4-morpholinyl)propyl)-2,4-dimethyl- |
260000|9600000 |
NA |
NA |
NA |
NA |
NA |
BindingDB |