| GENE_SYMBOL |
DRUG_NAME |
Ki (nM) |
IC50 (nM) |
Kd (nM) |
EC50 (nM) |
Potency (nM) |
AC50 (nM) |
Datasource |
| RPS6KA2 |
Ast-487 |
1100000 |
NA |
NA |
NA |
NA |
NA |
BindingDB |
| RPS6KA2 |
Synthesis of (R)-9-methyl-N-(1-((1-methylpiperidin-4-yl)methyl)-1H-pyrazol-4-yl)-6-oxo-6,7,8,9-tetrahydropyrido[3',2':4,5]pyrrolo[1,2-a]pyrazine-2-carboxamide |
NA |
124000 |
NA |
NA |
NA |
NA |
BindingDB |
| RPS6KA2 |
(R)-1-benzyl-N-(4-methyl-1-oxo-1,2,3,4-tetrahydropyrazino[1,2-a]indol-7-yl)-1H-pyrazole-4-carboxamide |
NA |
1377000 |
NA |
NA |
NA |
NA |
BindingDB |
| RPS6KA2 |
(R)-1-(3-aminobenzyl)-N-(9-methyl-6-oxo-6,7,8,9-tetrahydropyrido[3'',2'':4,5]pyrrolo[1,2-a]pyrazin-2-yl)-1H-pyrazole-4-carboxamide |
NA |
123000 |
NA |
NA |
NA |
NA |
BindingDB |
| RPS6KA2 |
Ruboxistaurin |
280000 |
NA |
NA |
NA |
NA |
NA |
BindingDB |
| RPS6KA2 |
N-[(2R,3S,4S,6S)-3-methoxy-2-methyl-16-oxo-29-oxa-1,7,17-triazaoctacyclo[12.12.2.12,6.07,28.08,13.015,19.020,27.021,26]nonacosa-8,10,12,14,19,21,23,25,27-nonaen-4-yl]-N-methylbenzamide |
730000 |
NA |
NA |
NA |
NA |
NA |
BindingDB |
| RPS6KA2 |
2-(2-chlorophenyl)-5,7-dihydroxy-8-[(3S)-3-hydroxy-1-methyl-4-piperidyl]chromone |
1500000 |
NA |
NA |
NA |
NA |
NA |
BindingDB |
| RPS6KA2 |
9,13-Epoxy-1H,9H-diindolo[1,2,3-gh:3',2',1'-lm]pyrrolo[3,4-j][1,7]benzodiazonin-1-one, 2,3,10,11,12,13-hexahydro-10-methoxy-9-methyl-11-(methylamino)-, (9S,10R,11R,13R)- |
190000 |
NA |
NA |
NA |
NA |
NA |
BindingDB |
| RPS6KA2 |
Sunitinib |
8400000 |
NA |
NA |
NA |
NA |
NA |
BindingDB |
| RPS6KA2 |
Jnj-7706621 |
410000 |
NA |
NA |
NA |
NA |
NA |
BindingDB |
| RPS6KA2 |
Tozasertib |
2000000 |
NA |
NA |
NA |
NA |
NA |
BindingDB |
| RPS6KA2 |
Pelitinib |
8700000 |
NA |
NA |
NA |
NA |
NA |
BindingDB |
| RPS6KA2 |
|
310000 |
NA |
NA |
NA |
NA |
NA |
BindingDB |
| RPS6KA2 |
Tofacitinib |
1400000 |
NA |
NA |
NA |
NA |
NA |
BindingDB |
| RPS6KA3 |
1H-Pyrrole-3-carboxamide, 5-((5-fluoro-1,2-dihydro-2-oxo-3H-indol-3-ylidene)methyl)-N-((2S)-2-hydroxy-3-(4-morpholinyl)propyl)-2,4-dimethyl- |
2100000 |
NA |
NA |
NA |
NA |
NA |
BindingDB |
| RPS6KA3 |
Synthesis of (R)-9-methyl-N-(1-((1-methylpiperidin-4-yl)methyl)-1H-pyrazol-4-yl)-6-oxo-6,7,8,9-tetrahydropyrido[3',2':4,5]pyrrolo[1,2-a]pyrazine-2-carboxamide |
NA |
124000 |
NA |
NA |
NA |
NA |
BindingDB |
| RPS6KA3 |
(R)-1-benzyl-N-(4-methyl-1-oxo-1,2,3,4-tetrahydropyrazino[1,2-a]indol-7-yl)-1H-pyrazole-4-carboxamide |
NA |
1377000 |
NA |
NA |
NA |
NA |
BindingDB |
| RPS6KA3 |
(R)-1-(3-aminobenzyl)-N-(9-methyl-6-oxo-6,7,8,9-tetrahydropyrido[3'',2'':4,5]pyrrolo[1,2-a]pyrazin-2-yl)-1H-pyrazole-4-carboxamide |
NA |
123000 |
NA |
NA |
NA |
NA |
BindingDB |
| RPS6KA3 |
Ruboxistaurin |
3600000 |
NA |
NA |
NA |
NA |
NA |
BindingDB |
| RPS6KA3 |
2-(3-bromo-4-hydroxyanilino)-5,7-dimethyl-8-(3-methylbutyl)-7H-pteridin-6-one |
NA |
141000 |
NA |
NA |
NA |
NA |
BindingDB |