| GENE_SYMBOL |
DRUG_NAME |
Ki (nM) |
IC50 (nM) |
Kd (nM) |
EC50 (nM) |
Potency (nM) |
AC50 (nM) |
Datasource |
| RPS6KA6 |
Ast-487 |
3400000 |
NA |
NA |
NA |
NA |
NA |
BindingDB |
| RPS6KA6 |
Ruboxistaurin |
2300000 |
NA |
NA |
NA |
NA |
NA |
BindingDB |
| RPS6KA6 |
SB 203580 |
250000 |
NA |
NA |
NA |
NA |
NA |
BindingDB |
| RPS6KA6 |
Sorafenib |
7500000 |
NA |
NA |
NA |
NA |
NA |
BindingDB |
| RPS6KA6 |
N-[(2R,3S,4S,6S)-3-methoxy-2-methyl-16-oxo-29-oxa-1,7,17-triazaoctacyclo[12.12.2.12,6.07,28.08,13.015,19.020,27.021,26]nonacosa-8,10,12,14,19,21,23,25,27-nonaen-4-yl]-N-methylbenzamide |
1500000 |
NA |
NA |
NA |
NA |
NA |
BindingDB |
| RPS6KA6 |
2-(2-chlorophenyl)-5,7-dihydroxy-8-[(3S)-3-hydroxy-1-methyl-4-piperidyl]chromone |
800000 |
NA |
NA |
NA |
NA |
NA |
BindingDB |
| RPS6KA6 |
Vandetanib |
240000 |
NA |
NA |
NA |
NA |
NA |
BindingDB |
| RPS6KA6 |
9,13-Epoxy-1H,9H-diindolo[1,2,3-gh:3',2',1'-lm]pyrrolo[3,4-j][1,7]benzodiazonin-1-one, 2,3,10,11,12,13-hexahydro-10-methoxy-9-methyl-11-(methylamino)-, (9S,10R,11R,13R)- |
3300000 |
NA |
NA |
NA |
NA |
NA |
BindingDB |
| RPS6KA6 |
Sunitinib |
2400000 |
NA |
NA |
NA |
NA |
NA |
BindingDB |
| RPS6KA6 |
|
270000 |
NA |
NA |
NA |
NA |
NA |
BindingDB |
| RPS6KA6 |
|
4600000 |
NA |
NA |
NA |
NA |
NA |
BindingDB |
| RPS6KA6 |
Tofacitinib |
1200000 |
NA |
NA |
NA |
NA |
NA |
BindingDB |
| RPS6KB1 |
(S)-2-(3-1H-indazol-5-ylureido)-N-(2-(dimethylamino)ethyl)-5-(1-hydroxyethyl)thiophene-3-carboxamide |
NA |
379000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| RPS6KB1 |
1-(5-tert-butyl-3-(morpholine-4-carbonyl)thiophen-2-yl)-3-(1H-indazol-5-yl)urea |
NA |
207000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| RPS6KB1 |
2-(3-1H-indazol-5-ylureido)-N-benzyl-5-tert-butylthiophene-3-carboxamide |
NA |
201000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| RPS6KB1 |
2-(3-1H-indazol-5-ylureido)-5-tert-butyl-N-(2-fluorobenzyl)thiophene-3-carboxamide |
NA |
191000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| RPS6KB1 |
2-(3-1H-indazol-5-ylureido)-N-(2-(dimethylamino)ethyl)-5-phenylthiophene-3-carboxamide |
NA |
1900000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| RPS6KB1 |
(R)-2-(3-1H-indazol-5-ylureido)-N-(2-(dimethylamino)ethyl)-5-(1-hydroxyethyl)thiophene-3-carboxamide |
NA |
196000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| RPS6KB1 |
2-(3-1H-indazol-5-ylureido)-N-(2-(dimethylamino)ethyl)-5-methylthiophene-3-carboxamide |
NA |
223000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| RPS7 |
NB-124 sulfate |
NA |
1493000 |
NA |
NA |
NA |
NA |
PubChem |